Compile Data Set for Download or QSAR
Report error Found 13 Enz. Inhib. hit(s) with all data for entry = 50032071
TargetCannabinoid receptor 1(Rat)
Clemson University

Curated by ChEMBL
LigandPNGBDBM50323910(CP-47,497 | 5-(1,1-Dimethyl-heptyl)-2-(3-hydroxy-c...)
Affinity DataKi:  9.54nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptor in Sprague-Dawley rat brain cortex membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Clemson University

Curated by ChEMBL
LigandPNGBDBM60994((10R,10aR)-6,6,9-Trimethyl-3-pentyl-6a,7,8,10a-tet...)
Affinity DataKi:  36nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cells after 1 hr by liquid scintillation spectrometry analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Clemson University

Curated by ChEMBL
LigandPNGBDBM60994((10R,10aR)-6,6,9-Trimethyl-3-pentyl-6a,7,8,10a-tet...)
Affinity DataKi:  41nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptor in Sprague-Dawley rat brain cortex membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Clemson University

Curated by ChEMBL
LigandPNGBDBM50323909(JWH-342 | (1S,3S)3-[4-(1,1-dimethylheptyl)phenyl]c...)
Affinity DataKi:  178nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cells after 1 hr by liquid scintillation spectrometry analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Clemson University

Curated by ChEMBL
LigandPNGBDBM50323907(JWH-324 | (1R*,3S*)-3-[4-(1,1-dimethylheptyl)pheny...)
Affinity DataKi:  231nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cells after 1 hr by liquid scintillation spectrometry analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Clemson University

Curated by ChEMBL
LigandPNGBDBM50323906(JWH-440 | (1R,3S)3-[2-Methoxy-4-(1,1-dimethylhexyl...)
Affinity DataKi:  553nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cells after 1 hr by liquid scintillation spectrometry analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Clemson University

Curated by ChEMBL
LigandPNGBDBM50323909(JWH-342 | (1S,3S)3-[4-(1,1-dimethylheptyl)phenyl]c...)
Affinity DataKi:  645nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptor in Sprague-Dawley rat brain cortex membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Clemson University

Curated by ChEMBL
LigandPNGBDBM50323905(JWH-442 | (1S,3S)3-[2-Methoxy-4-(1,1-dimethylhexyl...)
Affinity DataKi:  693nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cells after 1 hr by liquid scintillation spectrometry analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Clemson University

Curated by ChEMBL
LigandPNGBDBM50323908((1R,3S)3-[2-Methoxy-4-(1,1-dimethylheptyl)phenyl]c...)
Affinity DataKi:  808nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cells after 1 hr by liquid scintillation spectrometry analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Clemson University

Curated by ChEMBL
LigandPNGBDBM50323907(JWH-324 | (1R*,3S*)-3-[4-(1,1-dimethylheptyl)pheny...)
Affinity DataKi:  2.95E+3nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptor in Sprague-Dawley rat brain cortex membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Clemson University

Curated by ChEMBL
LigandPNGBDBM50323905(JWH-442 | (1S,3S)3-[2-Methoxy-4-(1,1-dimethylhexyl...)
Affinity DataKi:  4.12E+3nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptor in Sprague-Dawley rat brain cortex membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Clemson University

Curated by ChEMBL
LigandPNGBDBM50323906(JWH-440 | (1R,3S)3-[2-Methoxy-4-(1,1-dimethylhexyl...)
Affinity DataKi:  4.41E+3nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptor in Sprague-Dawley rat brain cortex membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Clemson University

Curated by ChEMBL
LigandPNGBDBM50323908((1R,3S)3-[2-Methoxy-4-(1,1-dimethylheptyl)phenyl]c...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptor in Sprague-Dawley rat brain cortex membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed