Compile Data Set for Download or QSAR
Report error Found 54 Enz. Inhib. hit(s) with all data for entry = 50032023
TargetMitogen-activated protein kinase 14(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50323438(4-(3-(3-tert-butyl-5-(3-naphthalen-1-ylureido)-1H-...)
Affinity DataIC50: 5nMAssay Description:Inhibition of unactive p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50323438(4-(3-(3-tert-butyl-5-(3-naphthalen-1-ylureido)-1H-...)
Affinity DataIC50: 6nMAssay Description:Inhibition of active p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50323416(2-acetamido-N-(3-(3-tert-butyl-5-(3-phenylureido)-...)
Affinity DataIC50: 6nMAssay Description:Inhibition of unactive p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50323437((1R)-6-(3-(3-tert-butyl-5-(3-phenylureido)-1H-pyra...)
Affinity DataIC50: 14nMAssay Description:Inhibition of unactive p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50323427(N-(3-(3-tert-butyl-5-(3-phenylureido)-1H-pyrazol-1...)
Affinity DataIC50: 16nMAssay Description:Inhibition of unactive p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50323420(N-(2-(3-(3-tert-butyl-5-(3-phenylureido)-1H-pyrazo...)
Affinity DataIC50: 18nMAssay Description:Inhibition of unactive p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50323431(N-(3-(3-tert-butyl-5-(3-phenylureido)-1H-pyrazol-1...)
Affinity DataIC50: 27.9nMAssay Description:Inhibition of unactive p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50323435((1R)-2-(3-(3-tert-butyl-5-(3-phenylureido)-1H-pyra...)
Affinity DataIC50: 30nMAssay Description:Inhibition of unactive p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50323416(2-acetamido-N-(3-(3-tert-butyl-5-(3-phenylureido)-...)
Affinity DataIC50: 34nMAssay Description:Inhibition of active p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50323433(4-(3-(3-tert-butyl-5-(3-phenylureido)-1H-pyrazol-1...)
Affinity DataIC50: 37nMAssay Description:Inhibition of unactive p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50323419(N-(2-(3-(3-tert-butyl-5-(3-phenylureido)-1H-pyrazo...)
Affinity DataIC50: 38nMAssay Description:Inhibition of unactive p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50323434(4-(3-(3-tert-butyl-5-(3-phenylureido)-1H-pyrazol-1...)
Affinity DataIC50: 39nMAssay Description:Inhibition of unactive p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50323430(N-(3-(3-tert-butyl-5-(3-phenylureido)-1H-pyrazol-1...)
Affinity DataIC50: 48.8nMAssay Description:Inhibition of unactive p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50323418(N-(2-(3-(3-tert-butyl-5-(3-phenylureido)-1H-pyrazo...)
Affinity DataIC50: 51nMAssay Description:Inhibition of unactive p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50323436((1R)-2-(3-(3-tert-butyl-5-(3-phenylureido)-1H-pyra...)
Affinity DataIC50: 57nMAssay Description:Inhibition of unactive p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50323427(N-(3-(3-tert-butyl-5-(3-phenylureido)-1H-pyrazol-1...)
Affinity DataIC50: 63nMAssay Description:Inhibition of active p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50323425(N-(3-(3-tert-butyl-5-(3-phenylureido)-1H-pyrazol-1...)
Affinity DataIC50: 68nMAssay Description:Inhibition of unactive p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50323415(N-(3-(3-tert-butyl-5-(3-phenylureido)-1H-pyrazol-1...)
Affinity DataIC50: 68nMAssay Description:Inhibition of unactive p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50323432(N-(3-(3-tert-butyl-5-(3-phenylureido)-1H-pyrazol-1...)
Affinity DataIC50: 78.2nMAssay Description:Inhibition of unactive p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50323420(N-(2-(3-(3-tert-butyl-5-(3-phenylureido)-1H-pyrazo...)
Affinity DataIC50: 88nMAssay Description:Inhibition of active p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50323423(N-(3-(3-tert-butyl-5-(3-phenylureido)-1H-pyrazol-1...)
Affinity DataIC50: 108nMAssay Description:Inhibition of unactive p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50323429(N-(3-(3-tert-butyl-5-(3-phenylureido)-1H-pyrazol-1...)
Affinity DataIC50: 132nMAssay Description:Inhibition of unactive p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50323430(N-(3-(3-tert-butyl-5-(3-phenylureido)-1H-pyrazol-1...)
Affinity DataIC50: 135nMAssay Description:Inhibition of active p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50323421(2-acetamido-N-(3-(3-tert-butyl-5-(3-phenylureido)-...)
Affinity DataIC50: 168nMAssay Description:Inhibition of unactive p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50323417(N-(2-(3-(3-tert-butyl-5-(3-phenylureido)-1H-pyrazo...)
Affinity DataIC50: 169nMAssay Description:Inhibition of unactive p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50323413(2-amino-N-(3-(3-tert-butyl-5-(3-phenylureido)-1H-p...)
Affinity DataIC50: 176nMAssay Description:Inhibition of unactive p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50323414(methyl 2-(3-(3-tert-butyl-5-(3-phenylureido)-1H-py...)
Affinity DataIC50: 176nMAssay Description:Inhibition of unactive p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50323426(N-(3-(3-tert-butyl-5-(3-phenylureido)-1H-pyrazol-1...)
Affinity DataIC50: 185nMAssay Description:Inhibition of unactive p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50323431(N-(3-(3-tert-butyl-5-(3-phenylureido)-1H-pyrazol-1...)
Affinity DataIC50: 201nMAssay Description:Inhibition of active p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50323418(N-(2-(3-(3-tert-butyl-5-(3-phenylureido)-1H-pyrazo...)
Affinity DataIC50: 205nMAssay Description:Inhibition of active p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50323424(2-acetamido-N-(3-(3-tert-butyl-5-(3-phenylureido)-...)
Affinity DataIC50: 211nMAssay Description:Inhibition of unactive p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50323428(N-(3-(3-tert-butyl-5-(3-phenylureido)-1H-pyrazol-1...)
Affinity DataIC50: 231nMAssay Description:Inhibition of unactive p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50323419(N-(2-(3-(3-tert-butyl-5-(3-phenylureido)-1H-pyrazo...)
Affinity DataIC50: 243nMAssay Description:Inhibition of active p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50323414(methyl 2-(3-(3-tert-butyl-5-(3-phenylureido)-1H-py...)
Affinity DataIC50: 287nMAssay Description:Inhibition of active p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50323425(N-(3-(3-tert-butyl-5-(3-phenylureido)-1H-pyrazol-1...)
Affinity DataIC50: 296nMAssay Description:Inhibition of active p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50323432(N-(3-(3-tert-butyl-5-(3-phenylureido)-1H-pyrazol-1...)
Affinity DataIC50: 331nMAssay Description:Inhibition of active p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50323415(N-(3-(3-tert-butyl-5-(3-phenylureido)-1H-pyrazol-1...)
Affinity DataIC50: 332nMAssay Description:Inhibition of active p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50323433(4-(3-(3-tert-butyl-5-(3-phenylureido)-1H-pyrazol-1...)
Affinity DataIC50: 393nMAssay Description:Inhibition of active p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50323417(N-(2-(3-(3-tert-butyl-5-(3-phenylureido)-1H-pyrazo...)
Affinity DataIC50: 441nMAssay Description:Inhibition of active p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50323421(2-acetamido-N-(3-(3-tert-butyl-5-(3-phenylureido)-...)
Affinity DataIC50: 480nMAssay Description:Inhibition of active p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50323428(N-(3-(3-tert-butyl-5-(3-phenylureido)-1H-pyrazol-1...)
Affinity DataIC50: 536nMAssay Description:Inhibition of active p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50323426(N-(3-(3-tert-butyl-5-(3-phenylureido)-1H-pyrazol-1...)
Affinity DataIC50: 599nMAssay Description:Inhibition of active p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50323423(N-(3-(3-tert-butyl-5-(3-phenylureido)-1H-pyrazol-1...)
Affinity DataIC50: 649nMAssay Description:Inhibition of active p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50323429(N-(3-(3-tert-butyl-5-(3-phenylureido)-1H-pyrazol-1...)
Affinity DataIC50: 677nMAssay Description:Inhibition of active p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50323422(1-acetamido-N-(3-(3-tert-butyl-5-(3-phenylureido)-...)
Affinity DataIC50: 715nMAssay Description:Inhibition of unactive p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50323437((1R)-6-(3-(3-tert-butyl-5-(3-phenylureido)-1H-pyra...)
Affinity DataIC50: 737nMAssay Description:Inhibition of active p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50323435((1R)-2-(3-(3-tert-butyl-5-(3-phenylureido)-1H-pyra...)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of active p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50323424(2-acetamido-N-(3-(3-tert-butyl-5-(3-phenylureido)-...)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of active p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50323413(2-amino-N-(3-(3-tert-butyl-5-(3-phenylureido)-1H-p...)
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of active p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50323412(1-(1-(3-(aminomethyl)phenyl)-3-tert-butyl-1H-pyraz...)
Affinity DataIC50: 2.85E+3nMAssay Description:Inhibition of unactive p38alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
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