Compile Data Set for Download or QSAR
Report error Found 70 Enz. Inhib. hit(s) with all data for entry = 50031847
TargetCollagenase 3(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50320443(4-(4-(4-(4-(2,3-dimethylphenyl)piperazine-1-carbon...)
Affinity DataIC50: 4nMAssay Description:Inhibition of MMP13More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50320424(4-(4-(4-(3,5-dimethylpiperazine-1-carbonyl)piperid...)
Affinity DataIC50: 4.40nMAssay Description:Inhibition of MMP13More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50320435(4-(4-(4-(4-(4-fluorophenyl)piperazine-1-carbonyl)p...)
Affinity DataIC50: 6nMAssay Description:Inhibition of MMP13More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50320423(4-(4-(4-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinol...)
Affinity DataIC50: 6.20nMAssay Description:Inhibition of MMP13More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50320439(N-hydroxy-4-(4-(4-(4-(pyrimidin-2-yl)piperazine-1-...)
Affinity DataIC50: 6.40nMAssay Description:Inhibition of MMP13More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50320436(4-(4-(4-(4-(4-acetylphenyl)piperazine-1-carbonyl)p...)
Affinity DataIC50: 6.70nMAssay Description:Inhibition of MMP13More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50320433(4-(4-(4-(4-(2-fluorophenyl)piperazine-1-carbonyl)p...)
Affinity DataIC50: 6.70nMAssay Description:Inhibition of MMP13More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50320422(N-hydroxy-4-(4-(4-(1,2,3,4-tetrahydroisoquinoline-...)
Affinity DataIC50: 9nMAssay Description:Inhibition of MMP13More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50320442(N-hydroxy-1-(2-methoxyethyl)-4-(4-(4-(phenylcarbam...)
Affinity DataIC50: 9nMAssay Description:Inhibition of MMP13More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50320438(N-hydroxy-4-(4-(4-(4-(pyridin-2-yl)piperazine-1-ca...)
Affinity DataIC50: 11nMAssay Description:Inhibition of MMP13More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50320437(4-(4-(4-(4-(2,4-dimethylphenyl)piperazine-1-carbon...)
Affinity DataIC50: 12nMAssay Description:Inhibition of MMP13More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50320426(cis-4-(4-(4-(3,5-dimethylmorpholine-4-carbonyl)pip...)
Affinity DataIC50: 18nMAssay Description:Inhibition of MMP13More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50320434(N-hydroxy-4-(4-(4-(4-(2-methoxyphenyl)piperazine-1...)
Affinity DataIC50: 18nMAssay Description:Inhibition of MMP13More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50320421(N-benzyl-1-(4-(1-cyclopropyl-4-(hydroxycarbamoyl)p...)
Affinity DataIC50: 20nMAssay Description:Inhibition of MMP13More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50320420(1-(4-(4-(hydroxycarbamoyl)tetrahydro-2H-pyran-4-yl...)
Affinity DataIC50: 25nMAssay Description:Inhibition of MMP13More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50320430(N-hydroxy-4-(4-(4-(4-phenethylpiperazine-1-carbony...)
Affinity DataIC50: 25nMAssay Description:Inhibition of MMP13More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50320441(N-hydroxy-4-(4-(4-(4-(pyrazin-2-yl)piperazine-1-ca...)
Affinity DataIC50: 27nMAssay Description:Inhibition of MMP13More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50320428(N-hydroxy-4-(4-(4-(4-isopropylpiperazine-1-carbony...)
Affinity DataIC50: 28nMAssay Description:Inhibition of MMP13More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50320444(1-cyclopropyl-4-(4-(4-(4-(2,3-dimethylphenyl)piper...)
Affinity DataIC50: 28nMAssay Description:Inhibition of MMP13More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50320440(N-hydroxy-4-(4-(4-(4-(pyridin-4-yl)piperazine-1-ca...)
Affinity DataIC50: 30nMAssay Description:Inhibition of MMP13More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50320419(N-allyl-1-(4-(4-(hydroxycarbamoyl)tetrahydro-2H-py...)
Affinity DataIC50: 35nMAssay Description:Inhibition of MMP13More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50320431(N-hydroxy-4-(4-(4-(4-(2-hydroxyethyl)piperazine-1-...)
Affinity DataIC50: 40nMAssay Description:Inhibition of MMP13More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50320429(N-hydroxy-4-(4-(4-(4-(2-methoxyethyl)piperazine-1-...)
Affinity DataIC50: 45nMAssay Description:Inhibition of MMP13More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50320427(4-(4-(4-(4-acetylpiperazine-1-carbonyl)piperidin-1...)
Affinity DataIC50: 50nMAssay Description:Inhibition of MMP13More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50320425(4-(4-(4-(3,5-dimethylpiperazine-1-carbonyl)piperid...)
Affinity DataIC50: 50nMAssay Description:Inhibition of MMP13More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50320445(4-(4-(4-(4-(2,3-dimethylphenyl)piperazine-1-carbon...)
Affinity DataIC50: 70nMAssay Description:Inhibition of MMP13More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetCollagenase 3(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50320432(4-(4-(4-(4-(2-(dimethylamino)ethyl)piperazine-1-ca...)
Affinity DataIC50: 90nMAssay Description:Inhibition of MMP13More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetStromelysin-1(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50320443(4-(4-(4-(4-(2,3-dimethylphenyl)piperazine-1-carbon...)
Affinity DataIC50: 160nMAssay Description:Inhibition of MMP3More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetStromelysin-1(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50320442(N-hydroxy-1-(2-methoxyethyl)-4-(4-(4-(phenylcarbam...)
Affinity DataIC50: 370nMAssay Description:Inhibition of MMP3More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50320445(4-(4-(4-(4-(2,3-dimethylphenyl)piperazine-1-carbon...)
Affinity DataIC50: 400nMAssay Description:Inhibition of MMP2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50320442(N-hydroxy-1-(2-methoxyethyl)-4-(4-(4-(phenylcarbam...)
Affinity DataIC50: 400nMAssay Description:Inhibition of MMP2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetStromelysin-1(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50320444(1-cyclopropyl-4-(4-(4-(4-(2,3-dimethylphenyl)piper...)
Affinity DataIC50: 550nMAssay Description:Inhibition of MMP3More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50320436(4-(4-(4-(4-(4-acetylphenyl)piperazine-1-carbonyl)p...)
Affinity DataIC50: 700nMAssay Description:Inhibition of MMP2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50320441(N-hydroxy-4-(4-(4-(4-(pyrazin-2-yl)piperazine-1-ca...)
Affinity DataIC50: 900nMAssay Description:Inhibition of MMP2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50320430(N-hydroxy-4-(4-(4-(4-phenethylpiperazine-1-carbony...)
Affinity DataIC50: 900nMAssay Description:Inhibition of MMP2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50320442(N-hydroxy-1-(2-methoxyethyl)-4-(4-(4-(phenylcarbam...)
Affinity DataIC50: 1.23E+3nMAssay Description:Inhibition of MMP9More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50320433(4-(4-(4-(4-(2-fluorophenyl)piperazine-1-carbonyl)p...)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of MMP2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50320439(N-hydroxy-4-(4-(4-(4-(pyrimidin-2-yl)piperazine-1-...)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of MMP2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50320435(4-(4-(4-(4-(4-fluorophenyl)piperazine-1-carbonyl)p...)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of MMP2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50320425(4-(4-(4-(3,5-dimethylpiperazine-1-carbonyl)piperid...)
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of MMP2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50320440(N-hydroxy-4-(4-(4-(4-(pyridin-4-yl)piperazine-1-ca...)
Affinity DataIC50: 1.75E+3nMAssay Description:Inhibition of MMP2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50320422(N-hydroxy-4-(4-(4-(1,2,3,4-tetrahydroisoquinoline-...)
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of MMP2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50320420(1-(4-(4-(hydroxycarbamoyl)tetrahydro-2H-pyran-4-yl...)
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of MMP2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50320423(4-(4-(4-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinol...)
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of MMP2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50320427(4-(4-(4-(4-acetylpiperazine-1-carbonyl)piperidin-1...)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of MMP2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50320419(N-allyl-1-(4-(4-(hydroxycarbamoyl)tetrahydro-2H-py...)
Affinity DataIC50: 2.90E+3nMAssay Description:Inhibition of MMP2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50320421(N-benzyl-1-(4-(1-cyclopropyl-4-(hydroxycarbamoyl)p...)
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibition of MMP2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50320438(N-hydroxy-4-(4-(4-(4-(pyridin-2-yl)piperazine-1-ca...)
Affinity DataIC50: 3.60E+3nMAssay Description:Inhibition of MMP2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50320434(N-hydroxy-4-(4-(4-(4-(2-methoxyphenyl)piperazine-1...)
Affinity DataIC50: 4.50E+3nMAssay Description:Inhibition of MMP2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50320428(N-hydroxy-4-(4-(4-(4-isopropylpiperazine-1-carbony...)
Affinity DataIC50: 5.50E+3nMAssay Description:Inhibition of MMP2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
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