Compile Data Set for Download or QSAR
Report error Found 22 Enz. Inhib. hit(s) with all data for entry = 50031829
TargetKappa-type opioid receptor(Guinea pig)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50320092((1R,5S,10R,18S)-15-hydroxy-9-methyl-6,19-dioxa-9-a...)
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [3H]U69493 from kappa opioid receptor in Hartley guinea pig cerebellum by liquid scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50320091((1R,5S,10R,18S)-9-(cyclopropylmethyl)-15-hydroxy-6...)
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [3H]U69493 from kappa opioid receptor in Hartley guinea pig cerebellum by liquid scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50320092((1R,5S,10R,18S)-15-hydroxy-9-methyl-6,19-dioxa-9-a...)
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in Hartley guinea pig forebrain by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50320083((2R,2aR,2a1S,5aR)-7-hydroxy-2-(methylamino)-2,2a,2...)
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [3H]U69493 from kappa opioid receptor in Hartley guinea pig cerebellum by liquid scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50320089((2R,2aS,2a1S,5aR)-2-(dimethylamino)-2a,7-dihydroxy...)
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [3H]U69493 from kappa opioid receptor in Hartley guinea pig cerebellum by liquid scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50320085((2R,2aR,2a1S,5aR)-2-(dimethylamino)-7-hydroxy-2,2a...)
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [3H]U69493 from kappa opioid receptor in Hartley guinea pig cerebellum by liquid scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50320087((2R,2aS,2a1S,5aR)-2a,7-dihydroxy-2-(methylamino)-2...)
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [3H]U69493 from kappa opioid receptor in Hartley guinea pig cerebellum by liquid scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50320090((2R,2aS,2a1S,5aR)-2-((cyclopropylmethyl)(methyl)am...)
Affinity DataKi:  1.17nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in Hartley guinea pig forebrain by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50320086((2R,2aR,2a1S,5aR)-2-((cyclopropylmethyl)(methyl)am...)
Affinity DataKi:  3.36nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in Hartley guinea pig forebrain by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50320090((2R,2aS,2a1S,5aR)-2-((cyclopropylmethyl)(methyl)am...)
Affinity DataKi:  5.10nMAssay Description:Displacement of [3H]U69493 from kappa opioid receptor in Hartley guinea pig cerebellum by liquid scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50320086((2R,2aR,2a1S,5aR)-2-((cyclopropylmethyl)(methyl)am...)
Affinity DataKi:  8.81nMAssay Description:Displacement of [3H]U69493 from kappa opioid receptor in Hartley guinea pig cerebellum by liquid scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50320089((2R,2aS,2a1S,5aR)-2-(dimethylamino)-2a,7-dihydroxy...)
Affinity DataKi:  8.95nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in Hartley guinea pig forebrain by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50320088((2R,2aS,2a1S,5aR)-2-(cyclopropylmethylamino)-2a,7-...)
Affinity DataKi:  24.7nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in Hartley guinea pig forebrain by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50320084((2R,2aR,2a1S,5aR)-2-(cyclopropylmethylamino)-7-hyd...)
Affinity DataKi:  30.3nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in Hartley guinea pig forebrain by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50320084((2R,2aR,2a1S,5aR)-2-(cyclopropylmethylamino)-7-hyd...)
Affinity DataKi:  32.2nMAssay Description:Displacement of [3H]U69493 from kappa opioid receptor in Hartley guinea pig cerebellum by liquid scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50320085((2R,2aR,2a1S,5aR)-2-(dimethylamino)-7-hydroxy-2,2a...)
Affinity DataKi:  50.9nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in Hartley guinea pig forebrain by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50320088((2R,2aS,2a1S,5aR)-2-(cyclopropylmethylamino)-2a,7-...)
Affinity DataKi:  68.4nMAssay Description:Displacement of [3H]U69493 from kappa opioid receptor in Hartley guinea pig cerebellum by liquid scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50320093((1S,5R,13S,20R)-8-hydroxy-6,19-dioxa-16-azahexacyc...)
Affinity DataKi:  72.6nMAssay Description:Displacement of [3H]U69493 from kappa opioid receptor in Hartley guinea pig cerebellum by liquid scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50320093((1S,5R,13S,20R)-8-hydroxy-6,19-dioxa-16-azahexacyc...)
Affinity DataKi:  86nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in Hartley guinea pig forebrain by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50320087((2R,2aS,2a1S,5aR)-2a,7-dihydroxy-2-(methylamino)-2...)
Affinity DataKi:  118nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in Hartley guinea pig forebrain by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50320083((2R,2aR,2a1S,5aR)-7-hydroxy-2-(methylamino)-2,2a,2...)
Affinity DataKi:  164nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in Hartley guinea pig forebrain by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50320091((1R,5S,10R,18S)-9-(cyclopropylmethyl)-15-hydroxy-6...)
Affinity DataKi:  294nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in Hartley guinea pig forebrain by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed