Compile Data Set for Download or QSAR
Report error Found 2 Enz. Inhib. hit(s) with all data for entry = 50041809
TargetPeroxisome proliferator-activated receptor gamma(Human)
Rikkyo University

Curated by ChEMBL
LigandPNGBDBM28681(cid_5281055 | [3H]rosiglitazone | CHEMBL121 | ROSI...)
Affinity DataEC50:  89.1nMAssay Description:Transactivation of PPARgamma assessed as induction of alkaline phosphatase activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Rikkyo University

Curated by ChEMBL
LigandPNGBDBM50085044(2-(2-Benzoyl-phenylamino)-3-{4-[2-(5-methyl-2-phen...)
Affinity DataEC50:  0.339nMAssay Description:Transactivation of PPARgamma assessed as induction of alkaline phosphatase activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed