Compile Data Set for Download or QSAR
Report error Found 17 Enz. Inhib. hit(s) with all data for entry = 50031707
TargetHistone deacetylase 3(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50317647((3S,6S,9S,14aR)-6-((1H-indol-3-yl)methyl)-9-benzyl...)
Affinity DataIC50: 25nMAssay Description:Inhibition of full length HDAC3 expressed in HEK293 cells after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50317647((3S,6S,9S,14aR)-6-((1H-indol-3-yl)methyl)-9-benzyl...)
Affinity DataIC50: 68nMAssay Description:Inhibition of full length HDAC1 expressed in HEK293 cells after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetHistone deacetylase 2(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50317647((3S,6S,9S,14aR)-6-((1H-indol-3-yl)methyl)-9-benzyl...)
Affinity DataIC50: 179nMAssay Description:Inhibition of full length HDAC2 expressed in HEK293 cells after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetHistone deacetylase 6(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50317649(6-((3S,6S,9S,14aR)-6-((1H-indol-3-yl)methyl)-9-ben...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of full length HDAC6 expressed in HEK293 cells after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetHistone deacetylase 6(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50317647((3S,6S,9S,14aR)-6-((1H-indol-3-yl)methyl)-9-benzyl...)
Affinity DataIC50: 9.40E+3nMAssay Description:Inhibition of full length HDAC6 expressed in HEK293 cells after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetHistone deacetylase 4(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50317649(6-((3S,6S,9S,14aR)-6-((1H-indol-3-yl)methyl)-9-ben...)
Affinity DataIC50: 9.60E+3nMAssay Description:Inhibition of human HDAC4 catalytic domain expressed in Escherichia coli BL21 after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50317648(6-((3S,6S,9S,14aR)-6-((1H-indol-3-yl)methyl)-9-ben...)
Affinity DataIC50: 1.02E+4nMAssay Description:Inhibition of full length HDAC1 expressed in HEK293 cells after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetHistone deacetylase 4(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50317650(6-((3S,6S,9S,14aR)-3,9-bis((1H-indol-3-yl)methyl)-...)
Affinity DataIC50: 1.07E+4nMAssay Description:Inhibition of human HDAC4 catalytic domain expressed in Escherichia coli BL21 after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetHistone deacetylase 2(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50317648(6-((3S,6S,9S,14aR)-6-((1H-indol-3-yl)methyl)-9-ben...)
Affinity DataIC50: 1.14E+4nMAssay Description:Inhibition of full length HDAC2 expressed in HEK293 cells after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetHistone deacetylase 3(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50317648(6-((3S,6S,9S,14aR)-6-((1H-indol-3-yl)methyl)-9-ben...)
Affinity DataIC50: 2.20E+4nMAssay Description:Inhibition of full length HDAC3 expressed in HEK293 cells after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetHistone deacetylase 8(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50317648(6-((3S,6S,9S,14aR)-6-((1H-indol-3-yl)methyl)-9-ben...)
Affinity DataIC50: 2.30E+4nMAssay Description:Inhibition of human full length HDAC8 expressed in Escherichia coli after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetHistone deacetylase 6(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50317650(6-((3S,6S,9S,14aR)-3,9-bis((1H-indol-3-yl)methyl)-...)
Affinity DataIC50: 2.47E+4nMAssay Description:Inhibition of full length HDAC6 expressed in HEK293 cells after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetHistone deacetylase 8(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50317650(6-((3S,6S,9S,14aR)-3,9-bis((1H-indol-3-yl)methyl)-...)
Affinity DataIC50: 2.76E+4nMAssay Description:Inhibition of human full length HDAC8 expressed in Escherichia coli after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetHistone deacetylase 5(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50317650(6-((3S,6S,9S,14aR)-3,9-bis((1H-indol-3-yl)methyl)-...)
Affinity DataIC50: 3.10E+4nMAssay Description:Inhibition of HDAC5 catalytic domain expressed in Escherichia coli after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetHistone deacetylase 5(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50317649(6-((3S,6S,9S,14aR)-6-((1H-indol-3-yl)methyl)-9-ben...)
Affinity DataIC50: 3.10E+4nMAssay Description:Inhibition of HDAC5 catalytic domain expressed in Escherichia coli after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetHistone deacetylase 6(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50317648(6-((3S,6S,9S,14aR)-6-((1H-indol-3-yl)methyl)-9-ben...)
Affinity DataIC50: 3.36E+4nMAssay Description:Inhibition of full length HDAC6 expressed in HEK293 cells after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
University of Salerno

Curated by ChEMBL
LigandPNGBDBM50317650(6-((3S,6S,9S,14aR)-3,9-bis((1H-indol-3-yl)methyl)-...)
Affinity DataIC50: 7.30E+4nMAssay Description:Inhibition of full length HDAC1 expressed in HEK293 cells after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed