Compile Data Set for Download or QSAR
Report error Found 49 Enz. Inhib. hit(s) with all data for entry = 50031665
TargetBombesin receptor subtype-3(Mouse)
Amri

Curated by ChEMBL
LigandPNGBDBM50316914(5-((4'-(2-(4-(2,2-dimethylbutyl)-1H-imidazol-2-yl)...)
Affinity DataEC50:  2.90nMAssay Description:Agonist activity at mouse BRS3More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Mouse)
Amri

Curated by ChEMBL
LigandPNGBDBM50316912(5-((4'-(2-(4-(2,2-dimethylbutyl)-1H-imidazol-2-yl)...)
Affinity DataEC50:  4.60nMAssay Description:Agonist activity at mouse BRS3More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50316914(5-((4'-(2-(4-(2,2-dimethylbutyl)-1H-imidazol-2-yl)...)
Affinity DataIC50: 5.30nMAssay Description:Binding affinity to human BRS3More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50316905((R)-1-(4-(2-(4-(2,2-dimethylbutyl)-1H-imidazol-2-y...)
Affinity DataIC50: 5.30nMAssay Description:Binding affinity to human BRS3More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Mouse)
Amri

Curated by ChEMBL
LigandPNGBDBM50316911(5-((4'-(2-(4-(2,2-dimethylbutyl)-1H-imidazol-2-yl)...)
Affinity DataEC50:  5.80nMAssay Description:Agonist activity at mouse BRS3More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50316911(5-((4'-(2-(4-(2,2-dimethylbutyl)-1H-imidazol-2-yl)...)
Affinity DataIC50: 6.10nMAssay Description:Binding affinity to human BRS3More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50316906((R)-1-(4-(2-(4-(2,2-dimethylbutyl)-1H-imidazol-2-y...)
Affinity DataIC50: 6.20nMAssay Description:Binding affinity to human BRS3More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Mouse)
Amri

Curated by ChEMBL
LigandPNGBDBM50313751(4'-(2-(4-(2,2-dimethylbutyl)-1H-imidazol-2-yl)ethy...)
Affinity DataEC50:  9.60nMAssay Description:Agonist activity at mouse BRS3More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50316915(9-(2-(4-(2,2-dimethylbutyl)-1H-imidazol-2-yl)ethyl...)
Affinity DataIC50: 10nMAssay Description:Binding affinity to human BRS3More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Mouse)
Amri

Curated by ChEMBL
LigandPNGBDBM50316915(9-(2-(4-(2,2-dimethylbutyl)-1H-imidazol-2-yl)ethyl...)
Affinity DataEC50:  11nMAssay Description:Agonist activity at mouse BRS3More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50313751(4'-(2-(4-(2,2-dimethylbutyl)-1H-imidazol-2-yl)ethy...)
Affinity DataIC50: 11nMAssay Description:Binding affinity to human BRS3More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Mouse)
Amri

Curated by ChEMBL
LigandPNGBDBM50316905((R)-1-(4-(2-(4-(2,2-dimethylbutyl)-1H-imidazol-2-y...)
Affinity DataEC50:  12nMAssay Description:Agonist activity at mouse BRS3More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Mouse)
Amri

Curated by ChEMBL
LigandPNGBDBM50316913(5-((4'-(2-(4-(2,2-dimethylbutyl)-1H-imidazol-2-yl)...)
Affinity DataEC50:  12nMAssay Description:Agonist activity at mouse BRS3More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Mouse)
Amri

Curated by ChEMBL
LigandPNGBDBM50316908(7-(4-(2-(4-(2,2-dimethylbutyl)-1H-imidazol-2-yl)et...)
Affinity DataEC50:  13nMAssay Description:Agonist activity at mouse BRS3More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Mouse)
Amri

Curated by ChEMBL
LigandPNGBDBM50316907((R)-1-(4-(2-(4-(2,2-dimethylbutyl)-1H-imidazol-2-y...)
Affinity DataEC50:  13nMAssay Description:Agonist activity at mouse BRS3More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50316906((R)-1-(4-(2-(4-(2,2-dimethylbutyl)-1H-imidazol-2-y...)
Affinity DataEC50:  15nMAssay Description:Agonist activity at human BRS3More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50316909(5-(4'-(2-(4-(cyclopentylmethyl)-2H-imidazol-2-yl)e...)
Affinity DataIC50: 15nMAssay Description:Binding affinity to human BRS3More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Mouse)
Amri

Curated by ChEMBL
LigandPNGBDBM50316906((R)-1-(4-(2-(4-(2,2-dimethylbutyl)-1H-imidazol-2-y...)
Affinity DataEC50:  16nMAssay Description:Agonist activity at mouse BRS3More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Mouse)
Amri

Curated by ChEMBL
LigandPNGBDBM50316909(5-(4'-(2-(4-(cyclopentylmethyl)-2H-imidazol-2-yl)e...)
Affinity DataEC50:  16nMAssay Description:Agonist activity at mouse BRS3More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50316908(7-(4-(2-(4-(2,2-dimethylbutyl)-1H-imidazol-2-yl)et...)
Affinity DataIC50: 18nMAssay Description:Binding affinity to human BRS3More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50316904(9-(2-(4-(2,2-dimethylbutyl)-1H-imidazol-2-yl)ethyl...)
Affinity DataIC50: 20nMAssay Description:Binding affinity to human BRS3More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50316918(5-((4'-(2-(4-(2,2-dimethylbutyl)-1H-imidazol-2-yl)...)
Affinity DataIC50: 22nMAssay Description:Binding affinity to human BRS3More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50316905((R)-1-(4-(2-(4-(2,2-dimethylbutyl)-1H-imidazol-2-y...)
Affinity DataEC50:  24nMAssay Description:Agonist activity at human BRS3More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50313751(4'-(2-(4-(2,2-dimethylbutyl)-1H-imidazol-2-yl)ethy...)
Affinity DataEC50:  25nMAssay Description:Agonist activity at human BRS3More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50316907((R)-1-(4-(2-(4-(2,2-dimethylbutyl)-1H-imidazol-2-y...)
Affinity DataIC50: 26nMAssay Description:Binding affinity to human BRS3More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Mouse)
Amri

Curated by ChEMBL
LigandPNGBDBM50316904(9-(2-(4-(2,2-dimethylbutyl)-1H-imidazol-2-yl)ethyl...)
Affinity DataEC50:  27nMAssay Description:Agonist activity at mouse BRS3More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50316912(5-((4'-(2-(4-(2,2-dimethylbutyl)-1H-imidazol-2-yl)...)
Affinity DataIC50: 27nMAssay Description:Binding affinity to human BRS3More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50316915(9-(2-(4-(2,2-dimethylbutyl)-1H-imidazol-2-yl)ethyl...)
Affinity DataEC50:  29nMAssay Description:Agonist activity at human BRS3More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50316914(5-((4'-(2-(4-(2,2-dimethylbutyl)-1H-imidazol-2-yl)...)
Affinity DataEC50:  30nMAssay Description:Agonist activity at human BRS3More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50316919(5-((4'-(2-(4-(2,2-dimethylbutyl)-1H-imidazol-2-yl)...)
Affinity DataIC50: 31nMAssay Description:Binding affinity to human BRS3More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50316910(4'-(2-(4-(2,2-dimethylbutyl)-1H-imidazol-2-yl)ethy...)
Affinity DataIC50: 31nMAssay Description:Binding affinity to human BRS3More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Mouse)
Amri

Curated by ChEMBL
LigandPNGBDBM50316910(4'-(2-(4-(2,2-dimethylbutyl)-1H-imidazol-2-yl)ethy...)
Affinity DataEC50:  34nMAssay Description:Agonist activity at mouse BRS3More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50316911(5-((4'-(2-(4-(2,2-dimethylbutyl)-1H-imidazol-2-yl)...)
Affinity DataEC50:  41nMAssay Description:Agonist activity at human BRS3More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50316908(7-(4-(2-(4-(2,2-dimethylbutyl)-1H-imidazol-2-yl)et...)
Affinity DataEC50:  42nMAssay Description:Agonist activity at human BRS3More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50316907((R)-1-(4-(2-(4-(2,2-dimethylbutyl)-1H-imidazol-2-y...)
Affinity DataEC50:  42nMAssay Description:Agonist activity at human BRS3More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50316917(2-(4'-(2-(4-(2,2-dimethylbutyl)-1H-imidazol-2-yl)e...)
Affinity DataEC50:  54nMAssay Description:Agonist activity at human BRS3More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50316904(9-(2-(4-(2,2-dimethylbutyl)-1H-imidazol-2-yl)ethyl...)
Affinity DataEC50:  56nMAssay Description:Agonist activity at human BRS3More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50316909(5-(4'-(2-(4-(cyclopentylmethyl)-2H-imidazol-2-yl)e...)
Affinity DataEC50:  56nMAssay Description:Agonist activity at human BRS3More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50316912(5-((4'-(2-(4-(2,2-dimethylbutyl)-1H-imidazol-2-yl)...)
Affinity DataEC50:  78nMAssay Description:Agonist activity at human BRS3More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50316920(5-((4'-(2-(4-(2,2-dimethylbutyl)-1H-imidazol-2-yl)...)
Affinity DataIC50: 83nMAssay Description:Binding affinity to human BRS3More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50316917(2-(4'-(2-(4-(2,2-dimethylbutyl)-1H-imidazol-2-yl)e...)
Affinity DataIC50: 103nMAssay Description:Binding affinity to human BRS3More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50316913(5-((4'-(2-(4-(2,2-dimethylbutyl)-1H-imidazol-2-yl)...)
Affinity DataIC50: 127nMAssay Description:Binding affinity to human BRS3More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50316913(5-((4'-(2-(4-(2,2-dimethylbutyl)-1H-imidazol-2-yl)...)
Affinity DataEC50:  129nMAssay Description:Agonist activity at human BRS3More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50316910(4'-(2-(4-(2,2-dimethylbutyl)-1H-imidazol-2-yl)ethy...)
Affinity DataEC50:  133nMAssay Description:Agonist activity at human BRS3More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50316918(5-((4'-(2-(4-(2,2-dimethylbutyl)-1H-imidazol-2-yl)...)
Affinity DataEC50:  172nMAssay Description:Agonist activity at human BRS3More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50316916(5-(4'-(2-(4-(cyclopentylmethyl)-2H-imidazol-2-yl)e...)
Affinity DataIC50: 287nMAssay Description:Binding affinity to human BRS3More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50316919(5-((4'-(2-(4-(2,2-dimethylbutyl)-1H-imidazol-2-yl)...)
Affinity DataEC50:  336nMAssay Description:Agonist activity at human BRS3More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50316920(5-((4'-(2-(4-(2,2-dimethylbutyl)-1H-imidazol-2-yl)...)
Affinity DataEC50:  399nMAssay Description:Agonist activity at human BRS3More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed
TargetBombesin receptor subtype-3(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50316916(5-(4'-(2-(4-(cyclopentylmethyl)-2H-imidazol-2-yl)e...)
Affinity DataEC50:  1.77E+3nMAssay Description:Agonist activity at human BRS3More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2010
Entry Details Article
PubMed