Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 50031589
TargetSigma non-opioid intracellular receptor 1(Rat)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50315831(1-(3-Phenylpropyl)-4-(3-pyridyl)piperazine | CHEMB...)
Affinity DataKi:  21nMAssay Description:Displacement of [3H](+)-pentazocine from rat brain membrane sigma 1receptor after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Rat)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50315829(1-(3-Phenylpropyl)-4-(4-pyridyl)piperazine | CHEMB...)
Affinity DataKi:  34nMAssay Description:Displacement of [3H](+)-pentazocine from rat brain membrane sigma 1receptor after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Rat)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50315828(1-(2-Phenylethyl)-4-(4-pyridyl)piperazine | CHEMBL...)
Affinity DataKi:  42nMAssay Description:Displacement of [3H](+)-pentazocine from rat brain membrane sigma 1receptor after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Rat)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50109383(1-(3-phenylpropyl)-4-(pyridin-2-yl)piperazine | 1-...)
Affinity DataKi:  83nMAssay Description:Displacement of [3H](+)-pentazocine from rat brain membrane sigma 1receptor after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Rat)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50315830(1-(2-Phenylethyl)-4-(3-pyridyl)piperazine | CHEMBL...)
Affinity DataKi:  97nMAssay Description:Displacement of [3H](+)-pentazocine from rat brain membrane sigma 1receptor after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Rat)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50109388(1-Phenethyl-4-pyridin-2-yl-piperazine | 1-phenethy...)
Affinity DataKi:  326nMAssay Description:Displacement of [3H](+)-pentazocine from rat brain membrane sigma 1receptor after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed