Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50001043
TargetAromatase(Human)
Marion Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50012199(CHEMBL48460 | (R isomer)10-(1-Hydroxy-2-iodo-ethyl...)
Affinity DataKi:  11nMAssay Description:Inhibition of binding to human Placental Cytochrome P450 19A1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAromatase(Human)
Marion Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50012198(CHEMBL48160 | (R isomer)10-(2-Chloro-1-hydroxy-eth...)
Affinity DataKi:  63nMAssay Description:Inhibition of binding to human Placental Cytochrome P450 19A1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAromatase(Human)
Marion Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50012196(CHEMBL300921 | 5-methylpentacyclo[14.2.1.01,13.02,...)
Affinity DataKi:  70nMAssay Description:Inhibition of binding to human Placental Cytochrome P450 19A1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAromatase(Human)
Marion Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50012194(CHEMBL416282 | 10-(2-Bromo-acetyl)-13-methyl-1,6,7...)
Affinity DataKi:  190nMAssay Description:Inhibition of binding to human Placental Cytochrome P450 19A1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAromatase(Human)
Marion Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50012193(CHEMBL297073 | (R isomer)18-hydroxy-5-methylpentac...)
Affinity DataKi:  870nMAssay Description:Inhibition of binding to human Placental Cytochrome P450 19A1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAromatase(Human)
Marion Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50012195(CHEMBL296617 | (S isomer)18-hydroxy-5-methylpentac...)
Affinity DataKi:  926nMAssay Description:Inhibition of binding to human Placental Cytochrome P450 19A1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAromatase(Human)
Marion Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50012197(CHEMBL298172 | (R isomer)10-(2-Bromo-1-hydroxy-eth...)
Affinity DataKi:  1.13E+3nMAssay Description:Inhibition of binding to human Placental Cytochrome P450 19A1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAromatase(Human)
Marion Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50012197(CHEMBL298172 | (R isomer)10-(2-Bromo-1-hydroxy-eth...)
Affinity DataKi:  1.13E+3nMAssay Description:Inhibition of binding to human Placental Cytochrome P450 19A1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed