Compile Data Set for Download or QSAR
Report error Found 122 Enz. Inhib. hit(s) with all data for entry = 50031578
TargetAdenosine receptor A3(Human)
National University of Singapore

Curated by ChEMBL
LigandPNGBDBM50315643(N-[2-(Phenyl)-8-methylpyrazolo[4,3-e][1,2,4]triazo...)
Affinity DataKi:  0.108nMAssay Description:Displacement of [3H]NECA from human cloned adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
National University of Singapore

Curated by ChEMBL
LigandPNGBDBM50315644(N-[2-(4-Fluorophenyl)-8-methylpyrazolo[4,3-e][1,2,...)
Affinity DataKi:  0.201nMAssay Description:Displacement of [3H]NECA from human cloned adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
National University of Singapore

Curated by ChEMBL
LigandPNGBDBM50315647(N-[2-(4-Methoxyphenyl)-8-methylpyrazolo[4,3-e][1,2...)
Affinity DataKi:  0.241nMAssay Description:Displacement of [3H]NECA from human cloned adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
National University of Singapore

Curated by ChEMBL
LigandPNGBDBM50315645(N-[2-(4-Chlorophenyl)-8-methylpyrazolo[4,3-e][1,2,...)
Affinity DataKi:  0.248nMAssay Description:Displacement of [3H]NECA from human cloned adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
National University of Singapore

Curated by ChEMBL
LigandPNGBDBM50315646(N-[2-(4-Bromophenyl)-8-methylpyrazolo[4,3-e][1,2,4...)
Affinity DataKi:  0.345nMAssay Description:Displacement of [3H]NECA from human cloned adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
National University of Singapore

Curated by ChEMBL
LigandPNGBDBM50315648(N-[2-(4-Nitrophenyl)-8-methylpyrazolo[4,3-e][1,2,4...)
Affinity DataKi:  0.624nMAssay Description:Displacement of [3H]NECA from human cloned adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
National University of Singapore

Curated by ChEMBL
LigandPNGBDBM50109453(N-(2-Furan-2-yl-8-methyl-8H-pyrazolo[4,3-e][1,2,4]...)
Affinity DataKi:  0.810nMAssay Description:Displacement of [3H]NECA from human cloned adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
National University of Singapore

Curated by ChEMBL
LigandPNGBDBM50315637(N-[2-(4-Methoxyphenyl)-8-methylpyrazolo[4,3-e][1,2...)
Affinity DataKi:  2.10nMAssay Description:Displacement of [3H]NECA from human cloned adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
National University of Singapore

Curated by ChEMBL
LigandPNGBDBM50315635(N-[2-(4-Chlorophenyl)-8-methylpyrazolo[4,3-e][1,2,...)
Affinity DataKi:  2.82nMAssay Description:Displacement of [3H]NECA from human cloned adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
National University of Singapore

Curated by ChEMBL
LigandPNGBDBM50315634(N-[2-(4-Fluorophenyl)-8-methylpyrazolo[4,3-e][1,2,...)
Affinity DataKi:  3.43nMAssay Description:Displacement of [3H]NECA from human cloned adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
National University of Singapore

Curated by ChEMBL
LigandPNGBDBM50315633(N-[2-(Phenyl)-8-methylpyrazolo[4,3-e][1,2,4]triazo...)
Affinity DataKi:  5nMAssay Description:Displacement of [3H]NECA from human cloned adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
National University of Singapore

Curated by ChEMBL
LigandPNGBDBM50315636(N-[2-(4-Bromophenyl)-8-methylpyrazolo[4,3-e][1,2,4...)
Affinity DataKi:  5.24nMAssay Description:Displacement of [3H]NECA from human cloned adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
National University of Singapore

Curated by ChEMBL
LigandPNGBDBM50315639(N-Benzoyl-N-[8-methyl-2-(4-methoxyphenyl)-8H-pyraz...)
Affinity DataKi:  6.88nMAssay Description:Displacement of [3H]NECA from human cloned adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
National University of Singapore

Curated by ChEMBL
LigandPNGBDBM50315640(N-Benzoyl-N-[8-methyl-2-(4-chlorophenyl)-8H-pyrazo...)
Affinity DataKi:  6.94nMAssay Description:Displacement of [3H]NECA from human cloned adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
National University of Singapore

Curated by ChEMBL
LigandPNGBDBM50315624(2-(4-Methoxyphenyl)-8-methylpyrazolo[4,3-e]1,2,4-t...)
Affinity DataKi:  16.7nMAssay Description:Displacement of [3H]NECA from human cloned adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
National University of Singapore

Curated by ChEMBL
LigandPNGBDBM50315641(N-[2-(Phenyl)-8-phenylethyl-pyrazolo[4,3-e][1,2,4]...)
Affinity DataKi:  23.9nMAssay Description:Displacement of [3H]NECA from human cloned adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
National University of Singapore

Curated by ChEMBL
LigandPNGBDBM50315632(2-(4-Methoxyphenyl)-8-phenylethylpyrazolo[4,3-e]1,...)
Affinity DataKi:  25nMAssay Description:Displacement of [3H]NECA from human cloned adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
National University of Singapore

Curated by ChEMBL
LigandPNGBDBM50315621(2-(4-Fluorophenyl)-8-methylpyrazolo[4,3-e]1,2,4-tr...)
Affinity DataKi:  31.4nMAssay Description:Displacement of [3H]NECA from human cloned adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
National University of Singapore

Curated by ChEMBL
LigandPNGBDBM50315623(2-(4-Bromophenyl)-8-methylpyrazolo[4,3-e]1,2,4-tri...)
Affinity DataKi:  38.6nMAssay Description:Displacement of [3H]NECA from human cloned adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
National University of Singapore

Curated by ChEMBL
LigandPNGBDBM50315629(2-(4-Fluorophenyl)-8-phenylethylpyrazolo[4,3-e]1,2...)
Affinity DataKi:  39.1nMAssay Description:Displacement of [3H]CCPA from human cloned adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
National University of Singapore

Curated by ChEMBL
LigandPNGBDBM50315629(2-(4-Fluorophenyl)-8-phenylethylpyrazolo[4,3-e]1,2...)
Affinity DataKi:  50.6nMAssay Description:Displacement of [3H]NECA from human cloned adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
National University of Singapore

Curated by ChEMBL
LigandPNGBDBM50315638(N-[2-(4-Nitrophenyl)-8-methylpyrazolo[4,3-e][1,2,4...)
Affinity DataKi:  56.4nMAssay Description:Displacement of [3H]NECA from human cloned adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
National University of Singapore

Curated by ChEMBL
LigandPNGBDBM50315627(2-(4-Chlorophenyl)-8-ethylpyrazolo[4,3-e]1,2,4-tri...)
Affinity DataKi:  68.7nMAssay Description:Displacement of [3H]NECA from human cloned adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
National University of Singapore

Curated by ChEMBL
LigandPNGBDBM50315622(2-(4-Chlorophenyl)-8-methylpyrazolo[4,3-e]1,2,4-tr...)
Affinity DataKi:  72.4nMAssay Description:Displacement of [3H]NECA from human cloned adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
National University of Singapore

Curated by ChEMBL
LigandPNGBDBM50315628(2-(Phenyl)-8-phenylethylpyrazolo[4,3-e]1,2,4-triaz...)
Affinity DataKi:  74.8nMAssay Description:Displacement of [3H]CCPA from human cloned adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
National University of Singapore

Curated by ChEMBL
LigandPNGBDBM50315620(2-(Phenyl)-8-methylpyrazolo[4,3-e]1,2,4-triazolo[1...)
Affinity DataKi:  75nMAssay Description:Displacement of [3H]NECA from human cloned adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
National University of Singapore

Curated by ChEMBL
LigandPNGBDBM50315628(2-(Phenyl)-8-phenylethylpyrazolo[4,3-e]1,2,4-triaz...)
Affinity DataKi:  76.7nMAssay Description:Displacement of [3H]NECA from human cloned adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
National University of Singapore

Curated by ChEMBL
LigandPNGBDBM50315630(2-(4-Chlorophenyl)-8-phenylethylpyrazolo[4,3-e]1,2...)
Affinity DataKi:  79.7nMAssay Description:Displacement of [3H]NECA from human cloned adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
National University of Singapore

Curated by ChEMBL
LigandPNGBDBM50315626(2-(4-Chlorophenyl)-7-ethylpyrazolo[4,3-e]1,2,4-tri...)
Affinity DataKi:  83.8nMAssay Description:Displacement of [3H]NECA from human cloned adenosine A2a receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
National University of Singapore

Curated by ChEMBL
LigandPNGBDBM50315626(2-(4-Chlorophenyl)-7-ethylpyrazolo[4,3-e]1,2,4-tri...)
Affinity DataKi:  121nMAssay Description:Displacement of [3H]CCPA from human cloned adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
National University of Singapore

Curated by ChEMBL
LigandPNGBDBM50315620(2-(Phenyl)-8-methylpyrazolo[4,3-e]1,2,4-triazolo[1...)
Affinity DataKi:  121nMAssay Description:Displacement of [3H]NECA from human cloned adenosine A2a receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
National University of Singapore

Curated by ChEMBL
LigandPNGBDBM50315629(2-(4-Fluorophenyl)-8-phenylethylpyrazolo[4,3-e]1,2...)
Affinity DataKi:  127nMAssay Description:Displacement of [3H]NECA from human cloned adenosine A2a receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
National University of Singapore

Curated by ChEMBL
LigandPNGBDBM50315642(N-[2-(4-Bromophenyl)-8-phenylethyl-pyrazolo[4,3-e]...)
Affinity DataKi:  153nMAssay Description:Displacement of [3H]NECA from human cloned adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
National University of Singapore

Curated by ChEMBL
LigandPNGBDBM50315628(2-(Phenyl)-8-phenylethylpyrazolo[4,3-e]1,2,4-triaz...)
Affinity DataKi:  196nMAssay Description:Displacement of [3H]NECA from human cloned adenosine A2a receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
National University of Singapore

Curated by ChEMBL
LigandPNGBDBM50315630(2-(4-Chlorophenyl)-8-phenylethylpyrazolo[4,3-e]1,2...)
Affinity DataKi:  204nMAssay Description:Displacement of [3H]CCPA from human cloned adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
National University of Singapore

Curated by ChEMBL
LigandPNGBDBM50315631(2-(4-Bromophenyl)-8-phenylethylpyrazolo[4,3-e]1,2,...)
Affinity DataKi:  221nMAssay Description:Displacement of [3H]NECA from human cloned adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
National University of Singapore

Curated by ChEMBL
LigandPNGBDBM50315642(N-[2-(4-Bromophenyl)-8-phenylethyl-pyrazolo[4,3-e]...)
Affinity DataKi:  270nMAssay Description:Displacement of [3H]CCPA from human cloned adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
National University of Singapore

Curated by ChEMBL
LigandPNGBDBM50315632(2-(4-Methoxyphenyl)-8-phenylethylpyrazolo[4,3-e]1,...)
Affinity DataKi:  289nMAssay Description:Displacement of [3H]CCPA from human cloned adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
National University of Singapore

Curated by ChEMBL
LigandPNGBDBM50094701(2-Furan-2-yl-8-methyl-8H-pyrazolo[4,3-e][1,2,4]tri...)
Affinity DataKi:  300nMAssay Description:Displacement of [3H]NECA from human cloned adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
National University of Singapore

Curated by ChEMBL
LigandPNGBDBM50315641(N-[2-(Phenyl)-8-phenylethyl-pyrazolo[4,3-e][1,2,4]...)
Affinity DataKi:  313nMAssay Description:Displacement of [3H]CCPA from human cloned adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
National University of Singapore

Curated by ChEMBL
LigandPNGBDBM50315633(N-[2-(Phenyl)-8-methylpyrazolo[4,3-e][1,2,4]triazo...)
Affinity DataKi:  324nMAssay Description:Displacement of [3H]NECA from human cloned adenosine A2a receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
National University of Singapore

Curated by ChEMBL
LigandPNGBDBM50315620(2-(Phenyl)-8-methylpyrazolo[4,3-e]1,2,4-triazolo[1...)
Affinity DataKi:  339nMAssay Description:Displacement of [3H]CCPA from human cloned adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
National University of Singapore

Curated by ChEMBL
LigandPNGBDBM50315621(2-(4-Fluorophenyl)-8-methylpyrazolo[4,3-e]1,2,4-tr...)
Affinity DataKi:  355nMAssay Description:Displacement of [3H]NECA from human cloned adenosine A2a receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
National University of Singapore

Curated by ChEMBL
LigandPNGBDBM50315631(2-(4-Bromophenyl)-8-phenylethylpyrazolo[4,3-e]1,2,...)
Affinity DataKi:  498nMAssay Description:Displacement of [3H]CCPA from human cloned adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
National University of Singapore

Curated by ChEMBL
LigandPNGBDBM50315643(N-[2-(Phenyl)-8-methylpyrazolo[4,3-e][1,2,4]triazo...)
Affinity DataKi:  562nMAssay Description:Displacement of [3H]CCPA from human cloned adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
National University of Singapore

Curated by ChEMBL
LigandPNGBDBM50315626(2-(4-Chlorophenyl)-7-ethylpyrazolo[4,3-e]1,2,4-tri...)
Affinity DataKi:  565nMAssay Description:Displacement of [3H]NECA from human cloned adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
National University of Singapore

Curated by ChEMBL
LigandPNGBDBM50315633(N-[2-(Phenyl)-8-methylpyrazolo[4,3-e][1,2,4]triazo...)
Affinity DataKi:  622nMAssay Description:Displacement of [3H]CCPA from human cloned adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
National University of Singapore

Curated by ChEMBL
LigandPNGBDBM50315625(2-(4-Nitrophenyl)-8-methylpyrazolo[4,3-e]1,2,4-tri...)
Affinity DataKi:  655nMAssay Description:Displacement of [3H]NECA from human cloned adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
National University of Singapore

Curated by ChEMBL
LigandPNGBDBM50315643(N-[2-(Phenyl)-8-methylpyrazolo[4,3-e][1,2,4]triazo...)
Affinity DataKi:  778nMAssay Description:Displacement of [3H]NECA from human cloned adenosine A2a receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
National University of Singapore

Curated by ChEMBL
LigandPNGBDBM50315627(2-(4-Chlorophenyl)-8-ethylpyrazolo[4,3-e]1,2,4-tri...)
Affinity DataKi:  843nMAssay Description:Displacement of [3H]NECA from human cloned adenosine A2a receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
Displayed 1 to 50 (of 122 total ) | Next | Last >>
Jump to: