Compile Data Set for Download or QSAR
Report error Found 23 Enz. Inhib. hit(s) with all data for entry = 50031855
TargetHistone deacetylase 2(Human)
University of Poitiers

Curated by ChEMBL
LigandPNGBDBM50320524((E)-N-(2-amino-5-(thiophen-2-yl)phenyl)-4-(2-imino...)
Affinity DataIC50: 20nMAssay Description:Inhibition of recombinant HDAC2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
University of Poitiers

Curated by ChEMBL
LigandPNGBDBM19423(N-[2-amino-5-(thiophen-2-yl)phenyl]-4-acetamidoben...)
Affinity DataIC50: 40nMAssay Description:Inhibition of recombinant HDAC1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetPolyamine deacetylase HDAC10(Human)
University of Poitiers

Curated by ChEMBL
LigandPNGBDBM50140882(3-(5-benzoyl-1-methyl-1H-pyrrol-3-yl)-N-hydroxyacr...)
Affinity DataIC50: 50nMAssay Description:Inhibition of HDAC10More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
University of Poitiers

Curated by ChEMBL
LigandPNGBDBM19427(N-[2-amino-5-(thiophen-2-yl)phenyl]-4-methoxybenza...)
Affinity DataIC50: 50nMAssay Description:Inhibition of recombinant HDAC1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
University of Poitiers

Curated by ChEMBL
LigandPNGBDBM50320524((E)-N-(2-amino-5-(thiophen-2-yl)phenyl)-4-(2-imino...)
Affinity DataIC50: 60nMAssay Description:Inhibition of recombinant HDAC1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetHistone deacetylase 2(Human)
University of Poitiers

Curated by ChEMBL
LigandPNGBDBM19423(N-[2-amino-5-(thiophen-2-yl)phenyl]-4-acetamidoben...)
Affinity DataIC50: 100nMAssay Description:Inhibition of recombinant HDAC2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetHistone deacetylase 2(Human)
University of Poitiers

Curated by ChEMBL
LigandPNGBDBM19427(N-[2-amino-5-(thiophen-2-yl)phenyl]-4-methoxybenza...)
Affinity DataIC50: 200nMAssay Description:Inhibition of recombinant HDAC2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetPolyamine deacetylase HDAC10(Human)
University of Poitiers

Curated by ChEMBL
LigandPNGBDBM50140883(3-(5-benzoyl-1-methyl-1H-pyrrol-2-yl)-N-hydroxyacr...)
Affinity DataIC50: 280nMAssay Description:Inhibition of HDAC10More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetHistone deacetylase 3(Human)
University of Poitiers

Curated by ChEMBL
LigandPNGBDBM50320524((E)-N-(2-amino-5-(thiophen-2-yl)phenyl)-4-(2-imino...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of recombinant HDAC3More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetHistone deacetylase 3(Human)
University of Poitiers

Curated by ChEMBL
LigandPNGBDBM19423(N-[2-amino-5-(thiophen-2-yl)phenyl]-4-acetamidoben...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of recombinant HDAC3More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetHistone deacetylase 3(Human)
University of Poitiers

Curated by ChEMBL
LigandPNGBDBM19427(N-[2-amino-5-(thiophen-2-yl)phenyl]-4-methoxybenza...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of recombinant HDAC3More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetHistone deacetylase 6(Human)
University of Poitiers

Curated by ChEMBL
LigandPNGBDBM19423(N-[2-amino-5-(thiophen-2-yl)phenyl]-4-acetamidoben...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of recombinant HDAC6More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetHistone deacetylase 6(Human)
University of Poitiers

Curated by ChEMBL
LigandPNGBDBM19427(N-[2-amino-5-(thiophen-2-yl)phenyl]-4-methoxybenza...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of recombinant HDAC6More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetHistone deacetylase 6(Human)
University of Poitiers

Curated by ChEMBL
LigandPNGBDBM50320524((E)-N-(2-amino-5-(thiophen-2-yl)phenyl)-4-(2-imino...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of recombinant HDAC6More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetHistone deacetylase 8(Human)
University of Poitiers

Curated by ChEMBL
LigandPNGBDBM19423(N-[2-amino-5-(thiophen-2-yl)phenyl]-4-acetamidoben...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of recombinant HDAC8More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetHistone deacetylase 8(Human)
University of Poitiers

Curated by ChEMBL
LigandPNGBDBM19427(N-[2-amino-5-(thiophen-2-yl)phenyl]-4-methoxybenza...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of recombinant HDAC8More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetHistone deacetylase 8(Human)
University of Poitiers

Curated by ChEMBL
LigandPNGBDBM50320524((E)-N-(2-amino-5-(thiophen-2-yl)phenyl)-4-(2-imino...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of recombinant HDAC8More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
University of Poitiers

Curated by ChEMBL
LigandPNGBDBM19130(CHEMBL99 | (2E,4E,6R)-7-[4-(dimethylamino)phenyl]-...)
Affinity DataKi:  0.230nMAssay Description:Inhibition of recombinant HDAC1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetHistone deacetylase 3(Human)
University of Poitiers

Curated by ChEMBL
LigandPNGBDBM19130(CHEMBL99 | (2E,4E,6R)-7-[4-(dimethylamino)phenyl]-...)
Affinity DataKi:  0.580nMAssay Description:Inhibition of recombinant HDAC3More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetHistone deacetylase 2(Human)
University of Poitiers

Curated by ChEMBL
LigandPNGBDBM19130(CHEMBL99 | (2E,4E,6R)-7-[4-(dimethylamino)phenyl]-...)
Affinity DataKi:  0.760nMAssay Description:Inhibition of recombinant HDAC2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetHistone deacetylase 6(Human)
University of Poitiers

Curated by ChEMBL
LigandPNGBDBM19130(CHEMBL99 | (2E,4E,6R)-7-[4-(dimethylamino)phenyl]-...)
Affinity DataKi:  0.990nMAssay Description:Inhibition of recombinant HDAC6More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetPolyamine deacetylase HDAC10(Human)
University of Poitiers

Curated by ChEMBL
LigandPNGBDBM19130(CHEMBL99 | (2E,4E,6R)-7-[4-(dimethylamino)phenyl]-...)
Affinity DataKi:  7nMAssay Description:Inhibition of HDAC10More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetHistone deacetylase 8(Human)
University of Poitiers

Curated by ChEMBL
LigandPNGBDBM19130(CHEMBL99 | (2E,4E,6R)-7-[4-(dimethylamino)phenyl]-...)
Affinity DataKi:  130nMAssay Description:Inhibition of recombinant HDAC8More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed