Compile Data Set for Download or QSAR
Report error Found 40 Enz. Inhib. hit(s) with all data for entry = 50031505
TargetEukaryotic elongation factor 2 kinase(Human)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50314444(2-(4-chlorophenyl)-10-thia-5,7,12-triazatetracyclo...)
Affinity DataIC50: 110nMAssay Description:Inhibition of GST tagged eEf2K expressed in Escherichia coli by fluorometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50314436(3-amino-4-(furan-2-yl)-6,7,8,9,10,11-hexahydro-5H-...)
Affinity DataIC50: 170nMAssay Description:Inhibition of GST tagged eEf2K expressed in Escherichia coli by fluorometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50314406(8-(morpholin-4-yl)-11-thia-9,14,16-triazatetracycl...)
Affinity DataIC50: 220nMAssay Description:Inhibition of GST tagged eEf2K expressed in Escherichia coli by fluorometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50314427(3-amino-4-(5-chlorofuran-2-yl)-5,6,7,8,9,10-hexahy...)
Affinity DataIC50: 280nMAssay Description:Inhibition of GST tagged eEf2K expressed in Escherichia coli by fluorometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50314428(3-amino-4-(5-(trifluoromethyl)furan-2-yl)-5,6,7,8,...)
Affinity DataIC50: 300nMAssay Description:Inhibition of GST tagged eEf2K expressed in Escherichia coli by fluorometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50314419((E)-3-amino-4-(2-(furan-2-yl)vinyl)-5,6,7,8,9,10-h...)
Affinity DataIC50: 320nMAssay Description:Inhibition of GST tagged eEf2K expressed in Escherichia coli by fluorometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50314429(3-amino-4-(benzofuran-2-yl)-5,6,7,8,9,10-hexahydro...)
Affinity DataIC50: 330nMAssay Description:Inhibition of GST tagged eEf2K expressed in Escherichia coli by fluorometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50314442(2-(furan-2-yl)-10-thia-5,7,12-triazatetracyclo[11....)
Affinity DataIC50: 350nMAssay Description:Inhibition of GST tagged eEf2K expressed in Escherichia coli by fluorometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50314420(3-amino-4-(3-methylthiophen-2-yl)-5,6,7,8,9,10-hex...)
Affinity DataIC50: 460nMAssay Description:Inhibition of GST tagged eEf2K expressed in Escherichia coli by fluorometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50314418(3-amino-4-(furan-2-yl)-5,6,7,8,9,10-hexahydrocyclo...)
Affinity DataIC50: 640nMAssay Description:Inhibition of GST tagged eEf2K expressed in Escherichia coli by fluorometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50314430(3-amino-4-(5-ethylfuran-2-yl)-5,6,7,8,9,10-hexahyd...)
Affinity DataIC50: 660nMAssay Description:Inhibition of GST tagged eEf2K expressed in Escherichia coli by fluorometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50314431(3-amino-4-(5-(hydroxymethyl)furan-2-yl)-5,6,7,8,9,...)
Affinity DataIC50: 800nMAssay Description:Inhibition of GST tagged eEf2K expressed in Escherichia coli by fluorometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50314415(4-(3-amino-2-carbamoyl-5,6,7,8,9,10-hexahydrocyclo...)
Affinity DataIC50: 860nMAssay Description:Inhibition of GST tagged eEf2K expressed in Escherichia coli by fluorometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50314409(3-amino-4-isobutyl-5,6,7,8,9,10-hexahydrocycloocta...)
Affinity DataIC50: 860nMAssay Description:Inhibition of GST tagged eEf2K expressed in Escherichia coli by fluorometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50314421(3-amino-4-(pyridin-3-yl)-5,6,7,8,9,10-hexahydrocyc...)
Affinity DataIC50: 940nMAssay Description:Inhibition of GST tagged eEf2K expressed in Escherichia coli by fluorometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50314412(3-amino-4-(3,4-dichlorophenyl)-5,6,7,8,9,10-hexahy...)
Affinity DataIC50: 990nMAssay Description:Inhibition of GST tagged eEf2K expressed in Escherichia coli by fluorometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50314422(3-amino-4-(1-methyl-1H-pyrrol-2-yl)-5,6,7,8,9,10-h...)
Affinity DataIC50: 990nMAssay Description:Inhibition of GST tagged eEf2K expressed in Escherichia coli by fluorometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50314432(3-amino-4-(4,5-dimethylfuran-2-yl)-5,6,7,8,9,10-he...)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of GST tagged eEf2K expressed in Escherichia coli by fluorometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50314435(3-amino-4-(furan-2-yl)-6,7,8,9-tetrahydro-5H-cyclo...)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of GST tagged eEf2K expressed in Escherichia coli by fluorometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50314423(3-amino-4-(furan-3-yl)-5,6,7,8,9,10-hexahydrocyclo...)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of GST tagged eEf2K expressed in Escherichia coli by fluorometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50314413(3-amino-4-(4-chlorophenyl)-5,6,7,8,9,10-hexahydroc...)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of GST tagged eEf2K expressed in Escherichia coli by fluorometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50314408(3-amino-4-methyl-5,6,7,8,9,10-hexahydrocycloocta[b...)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of GST tagged eEf2K expressed in Escherichia coli by fluorometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50314417(3-amino-4-m-tolyl-5,6,7,8,9,10-hexahydrocycloocta[...)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of GST tagged eEf2K expressed in Escherichia coli by fluorometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50314416(3-amino-4-(2-fluoro-5-methoxyphenyl)-5,6,7,8,9,10-...)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of GST tagged eEf2K expressed in Escherichia coli by fluorometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50314424(3-amino-4-(thiazol-2-yl)-5,6,7,8,9,10-hexahydrocyc...)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of GST tagged eEf2K expressed in Escherichia coli by fluorometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50314410(3-amino-4-cyclopropyl-5,6,7,8,9,10-hexahydrocycloo...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of GST tagged eEf2K expressed in Escherichia coli by fluorometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50314407(3-amino-5,6,7,8,9,10-hexahydrocycloocta[b]thieno[3...)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of GST tagged eEf2K expressed in Escherichia coli by fluorometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50314441(10-thia-5,7,12-triazatetracyclo[11.7.0.0^{3,11}.0^...)
Affinity DataIC50: 3.70E+3nMAssay Description:Inhibition of GST tagged eEf2K expressed in Escherichia coli by fluorometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50314445(5-Furan-2-yl-7,8,9,10-tetrahydro-6H-12-thia-2,4,11...)
Affinity DataIC50: 4.70E+3nMAssay Description:Inhibition of GST tagged eEf2K expressed in Escherichia coli by fluorometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50314438(3-amino-6-(2,4-dimethoxyphenyl)-4-(furan-2-yl)thie...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of GST tagged eEf2K expressed in Escherichia coli by fluorometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50314439(3-amino-6-(2,4-dimethoxybenzyl)-4-(furan-2-yl)thie...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of GST tagged eEf2K expressed in Escherichia coli by fluorometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50314440(3-amino-6-(cyclohexylmethyl)-4-(furan-2-yl)thieno[...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of GST tagged eEf2K expressed in Escherichia coli by fluorometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50314411(rac-3-amino-4-(6-methylhept-5-en-2-yl)-5,6,7,8,9,1...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of GST tagged eEf2K expressed in Escherichia coli by fluorometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50314434(rac-3-amino-4-(furan-2-yl)-8-methyl-5,6,7,8-tetrah...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of GST tagged eEf2K expressed in Escherichia coli by fluorometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50314433(methyl 5-(3-amino-2-carbamoyl-5,6,7,8,9,10-hexahyd...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of GST tagged eEf2K expressed in Escherichia coli by fluorometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50314437(3-amino-4-(furan-2-yl)-5,6,7,8,9,10,11,12-octahydr...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of GST tagged eEf2K expressed in Escherichia coli by fluorometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50314426(3-amino-4-phenethyl-5,6,7,8,9,10-hexahydrocyclooct...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of GST tagged eEf2K expressed in Escherichia coli by fluorometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50314425(3-amino-4-(3-methylpyridin-2-yl)-5,6,7,8,9,10-hexa...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of GST tagged eEf2K expressed in Escherichia coli by fluorometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50314443(2-(1-benzofuran-2-yl)-10-thia-5,7,12-triazatetracy...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of GST tagged eEf2K expressed in Escherichia coli by fluorometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetEukaryotic elongation factor 2 kinase(Human)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50314414(3-amino-4-phenyl-5,6,7,8,9,10-hexahydrocycloocta[b...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of GST tagged eEf2K expressed in Escherichia coli by fluorometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed