Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) with all data for entry = 50031466
TargetTyrosine-protein kinase JAK2(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50182010(7-(pyridin-2-yl)-N-(2,4,6-trimethoxyphenyl)-7H-pyr...)
Affinity DataIC50: 5.90nMAssay Description:Inhibition of recombinant GST tagged JAK2 after 60 mins by Caliper mobility shift assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetTyrosine-protein kinase JAK2(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50312975(7-phenyl-N-(3,4,5-trimethoxyphenyl)benzo[d]oxazol-...)
Affinity DataIC50: 15nMAssay Description:Inhibition of recombinant GST tagged JAK2 after 60 mins by Caliper mobility shift assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed
TargetTyrosine-protein kinase JAK2(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50313807(N-methyl-4-[3-(3,4,5-trimethoxyphenyl)quinoxalin-5...)
Affinity DataIC50: 42nMAssay Description:Inhibition of recombinant GST tagged JAK2 after 60 mins by Caliper mobility shift assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2010
Entry Details Article
PubMed