Compile Data Set for Download or QSAR
Report error Found 43 Enz. Inhib. hit(s) with all data for entry = 50001019
TargetGastrin/cholecystokinin type B receptor(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50006878(1-(1-Methyl-2-oxo-5-phenyl-2,3-dihydro-1H-benzo[e]...)
Affinity DataIC50: 2.90nMAssay Description:Inhibition of [125I]-labeled gastrin binding to gastrin receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50006878(1-(1-Methyl-2-oxo-5-phenyl-2,3-dihydro-1H-benzo[e]...)
Affinity DataIC50: 5.30nMAssay Description:Inhibition of [125I]-labeled CCK-8 sulfate binding to CCK-B receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50006878(1-(1-Methyl-2-oxo-5-phenyl-2,3-dihydro-1H-benzo[e]...)
Affinity DataIC50: 7.30nMAssay Description:Inhibition of [125I]-labeled CCK-8 sulfate binding to CCK-B receptor in mouse brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50006842(CHEMBL37312 | 2-[2-(5-Bromo-1H-indol-3-yl)-ethyl]-...)
Affinity DataIC50: 9.30nMAssay Description:Inhibition of [125I]CCK-8 sulfate binding to cholecystokinin type B receptor in mouse brain membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50011943(CHEMBL37096 | 2-[2-(5-Bromo-1H-indol-3-yl)-ethyl]-...)
Affinity DataIC50: 16nMAssay Description:Inhibition of [125I]CCK-8 sulfate binding to cholecystokinin type B receptor in mouse brain membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50006838(CHEMBL36206 | 2-[2-(1H-Indol-3-yl)-ethyl]-3-(3-iso...)
Affinity DataIC50: 26nMAssay Description:Inhibition of [125I]CCK-8 sulfate binding to cholecystokinin type B receptor in mouse brain membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50011957(CHEMBL290897 | 2-[2-(5-Bromo-1H-indol-3-yl)-ethyl]...)
Affinity DataIC50: 28nMAssay Description:Inhibition of [125I]CCK-8 sulfate binding to cholecystokinin type B receptor in mouse brain membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50011939(CHEMBL285707 | 2-[2-(5-Bromo-1H-indol-3-yl)-ethyl]...)
Affinity DataIC50: 31nMAssay Description:Inhibition of [125I]CCK-8 sulfate binding to cholecystokinin type B receptor in mouse brain membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50011953(CHEMBL284853 | 2-[2-(5-Bromo-1H-indol-3-yl)-ethyl]...)
Affinity DataIC50: 33nMAssay Description:Inhibition of [125I]CCK-8 sulfate binding to cholecystokinin type B receptor in mouse brain membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50011965(CHEMBL417876 | 2-[2-(5-Bromo-1H-indol-3-yl)-ethyl]...)
Affinity DataIC50: 37nMAssay Description:Inhibition of [125I]CCK-8 sulfate binding to cholecystokinin type B receptor in mouse brain membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50011954(CHEMBL285940 | 2-[2-(5-Bromo-1H-indol-3-yl)-ethyl]...)
Affinity DataIC50: 37nMAssay Description:Inhibition of [125I]CCK-8 sulfate binding to cholecystokinin type B receptor in mouse brain membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50011942(CHEMBL37699 | 2-[2-(5-Bromo-1H-indol-3-yl)-ethyl]-...)
Affinity DataIC50: 38nMAssay Description:Inhibition of [125I]CCK-8 sulfate binding to cholecystokinin type B receptor in mouse brain membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50011942(CHEMBL37699 | 2-[2-(5-Bromo-1H-indol-3-yl)-ethyl]-...)
Affinity DataIC50: 38nMAssay Description:Inhibition of [125I]CCK-8 sulfate binding to cholecystokinin type B receptor in mouse brain membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50011948(CHEMBL36779 | 2-[2-(5-Bromo-1H-indol-3-yl)-ethyl]-...)
Affinity DataIC50: 46nMAssay Description:Inhibition of [125I]CCK-8 sulfate binding to cholecystokinin type B receptor in mouse brain membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50011940(CHEMBL36436 | 2-[2-(5-Bromo-1H-indol-3-yl)-ethyl]-...)
Affinity DataIC50: 46nMAssay Description:Inhibition of [125I]CCK-8 sulfate binding to cholecystokinin type B receptor in mouse brain membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50011945(CHEMBL37758 | 2-[2-(5-Chloro-1H-indol-3-yl)-ethyl]...)
Affinity DataIC50: 47nMAssay Description:Inhibition of [125I]CCK-8 sulfate binding to cholecystokinin type B receptor in mouse brain membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50011946(CHEMBL287739 | 3-(3-Methoxy-phenyl)-2-[2-(5-methyl...)
Affinity DataIC50: 55nMAssay Description:Inhibition of [125I]CCK-8 sulfate binding to cholecystokinin type B receptor in mouse brain membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50011950(CHEMBL34198 | 2-[2-(5-Bromo-1H-indol-3-yl)-ethyl]-...)
Affinity DataIC50: 58nMAssay Description:Inhibition of [125I]CCK-8 sulfate binding to cholecystokinin type B receptor in mouse brain membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50011966(CHEMBL287740 | 2-[2-(5-Bromo-1H-indol-3-yl)-ethyl]...)
Affinity DataIC50: 67nMAssay Description:Inhibition of [125I]CCK-8 sulfate binding to cholecystokinin type B receptor in mouse brain membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50011958(CHEMBL37990 | 2-[2-(5-Methoxy-1H-indol-3-yl)-ethyl...)
Affinity DataIC50: 67nMAssay Description:Inhibition of [125I]CCK-8 sulfate binding to cholecystokinin type B receptor in mouse brain membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50011962(CHEMBL38330 | 3-(3-Ethyl-phenyl)-2-[2-(1H-indol-3-...)
Affinity DataIC50: 72nMAssay Description:Inhibition of [125I]CCK-8 sulfate binding to cholecystokinin type B receptor in mouse brain membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50006842(CHEMBL37312 | 2-[2-(5-Bromo-1H-indol-3-yl)-ethyl]-...)
Affinity DataIC50: 81nMAssay Description:Inhibition of [125I]-labeled CCK-8 sulfate binding to Cholecystokinin type B receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50011961(CHEMBL34547 | 2-[2-(5-Bromo-1H-indol-3-yl)-ethyl]-...)
Affinity DataIC50: 88nMAssay Description:Inhibition of [125I]CCK-8 sulfate binding to cholecystokinin type B receptor in mouse brain membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50011952(CHEMBL36634 | 2-[2-(5-Bromo-1H-indol-3-yl)-propyl]...)
Affinity DataIC50: 100nMAssay Description:Inhibition of [125I]CCK-8 sulfate binding to cholecystokinin type B receptor in mouse brain membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50011947(CHEMBL33948 | 2-[2-(5-Bromo-1H-indol-3-yl)-ethyl]-...)
Affinity DataIC50: 110nMAssay Description:Inhibition of [125I]CCK-8 sulfate binding to cholecystokinin type B receptor in mouse brain membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50011941(CHEMBL287914 | 2-[2-(5-Fluoro-1H-indol-3-yl)-ethyl...)
Affinity DataIC50: 110nMAssay Description:Inhibition of [125I]CCK-8 sulfate binding to cholecystokinin type B receptor in mouse brain membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50011964(CHEMBL34979 | 2-[2-(5-Bromo-1H-indol-3-yl)-ethyl]-...)
Affinity DataIC50: 130nMAssay Description:Inhibition of [125I]CCK-8 sulfate binding to cholecystokinin type B receptor in mouse brain membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50011949(CHEMBL289053 | 2-[2-(1H-Indol-3-yl)-ethyl]-3-m-tol...)
Affinity DataIC50: 150nMAssay Description:Inhibition of [125I]CCK-8 sulfate binding to cholecystokinin type B receptor in mouse brain membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50006842(CHEMBL37312 | 2-[2-(5-Bromo-1H-indol-3-yl)-ethyl]-...)
Affinity DataIC50: 160nMAssay Description:Inhibition of [125I]-labeled CCK-8 sulfate binding to Cholecystokinin type B receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50011956(CHEMBL37829 | 2-[2-(1H-Indol-3-yl)-ethyl]-3-(3-met...)
Affinity DataIC50: 160nMAssay Description:Inhibition of [125I]CCK-8 sulfate binding to cholecystokinin type B receptor in mouse brain membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50011963(CHEMBL287913 | 3-Benzo[1,3]dioxol-5-yl-2-[2-(1H-in...)
Affinity DataIC50: 190nMAssay Description:Inhibition of [125I]CCK-8 sulfate binding to cholecystokinin type B receptor in mouse brain membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50011960(CHEMBL284317 | 2-[2-(5-Bromo-1H-indol-3-yl)-ethyl]...)
Affinity DataIC50: 230nMAssay Description:Inhibition of [125I]CCK-8 sulfate binding to cholecystokinin type B receptor in mouse brain membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50011940(CHEMBL36436 | 2-[2-(5-Bromo-1H-indol-3-yl)-ethyl]-...)
Affinity DataIC50: 330nMAssay Description:Inhibition of [125I]-labeled CCK-8 sulfate binding to Cholecystokinin type B receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50011942(CHEMBL37699 | 2-[2-(5-Bromo-1H-indol-3-yl)-ethyl]-...)
Affinity DataIC50: 360nMAssay Description:Inhibition of [125I]-labeled CCK-8 sulfate binding to Cholecystokinin type B receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50011959(CHEMBL37887 | 3-(3-Bromo-phenyl)-2-[2-(1H-indol-3-...)
Affinity DataIC50: 370nMAssay Description:Inhibition of [125I]CCK-8 sulfate binding to cholecystokinin type B receptor in mouse brain membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50011955(CHEMBL37439 | 2-[2-(1H-Indol-3-yl)-ethyl]-3-(3-tri...)
Affinity DataIC50: 480nMAssay Description:Inhibition of [125I]CCK-8 sulfate binding to cholecystokinin type B receptor in mouse brain membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50006837(CHEMBL37653 | 2-[2-(1H-Indol-3-yl)-ethyl]-3-phenyl...)
Affinity DataIC50: 670nMAssay Description:Inhibition of [125I]CCK-8 sulfate binding to cholecystokinin type B receptor in mouse brain membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50011944(CHEMBL34185 | 3-(3-Chloro-phenyl)-2-[2-(1H-indol-3...)
Affinity DataIC50: 690nMAssay Description:Inhibition of [125I]CCK-8 sulfate binding to cholecystokinin type B receptor in mouse brain membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Mouse)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50011951(CHEMBL38176 | 3-(3-Fluoro-phenyl)-2-[2-(1H-indol-3...)
Affinity DataIC50: 730nMAssay Description:Inhibition of [125I]CCK-8 sulfate binding to cholecystokinin type B receptor in mouse brain membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50011940(CHEMBL36436 | 2-[2-(5-Bromo-1H-indol-3-yl)-ethyl]-...)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of [125I]-labeled CCK-8 sulfate binding to Cholecystokinin type B receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50011942(CHEMBL37699 | 2-[2-(5-Bromo-1H-indol-3-yl)-ethyl]-...)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of [125I]-labeled CCK-8 sulfate binding to Cholecystokinin type B receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50011952(CHEMBL36634 | 2-[2-(5-Bromo-1H-indol-3-yl)-propyl]...)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of [125I]-labeled CCK-8 sulfate binding to Cholecystokinin type B receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50011955(CHEMBL37439 | 2-[2-(1H-Indol-3-yl)-ethyl]-3-(3-tri...)
Affinity DataIC50: 8.20E+3nMAssay Description:Inhibition of [125I]-labeled CCK-8 sulfate binding to Cholecystokinin type B receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed