Compile Data Set for Download or QSAR
Report error Found 35 Enz. Inhib. hit(s) with all data for entry = 50001013
TargetPlatelet-activating factor receptor(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50011872(CHEMBL34461 | 4-(2-Chloro-phenyl)-9-methyl-2-[2-(5...)
Affinity DataIC50: 8nMAssay Description:In vitro for platelet activating factor receptor antagonist activity in a binding assay using washed whole dog platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50011876(CHEMBL286217 | 4-(2-Chloro-phenyl)-2-ethynyl-9-met...)
Affinity DataIC50: 10nMAssay Description:In vitro for platelet activating factor receptor antagonist activity in a binding assay using washed whole dog platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50011862(CHEMBL430919 | 2-[2-(4-Butyl-phenyl)-vinyl]-4-(2-c...)
Affinity DataIC50: 10nMAssay Description:In vitro for platelet activating factor receptor antagonist activity in a binding assay using washed whole dog platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50011866(CHEMBL442259 | 2-[2-(4-Butyl-phenyl)-ethyl]-4-(2-c...)
Affinity DataIC50: 10nMAssay Description:In vitro for platelet activating factor receptor antagonist activity in a binding assay using washed whole dog platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50011877(CHEMBL32475 | 4-(2-Chloro-phenyl)-9-methyl-2-trime...)
Affinity DataIC50: 20nMAssay Description:In vitro for platelet activating factor receptor antagonist activity in a binding assay using washed whole dog platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50011852(CHEMBL289463 | 4-(2-Chloro-phenyl)-2-(2-indan-5-yl...)
Affinity DataIC50: 20nMAssay Description:In vitro for platelet activating factor receptor antagonist activity in a binding assay using washed whole dog platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50011864(CHEMBL287465 | 4-(2-Chloro-phenyl)-2-[2-(2,3-dihyd...)
Affinity DataIC50: 20nMAssay Description:In vitro for platelet activating factor receptor antagonist activity in a binding assay using washed whole dog platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50011853(CHEMBL32942 | 4-(2-Chloro-phenyl)-2-[2-(4-isobutyl...)
Affinity DataIC50: 30nMAssay Description:In vitro for platelet activating factor receptor antagonist activity in a binding assay using washed whole dog platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50011868(CHEMBL432850 | 4-(2-Chloro-phenyl)-2-[2-(4-cyclohe...)
Affinity DataIC50: 35nMAssay Description:In vitro for platelet activating factor receptor antagonist activity in a binding assay using washed whole dog platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50011861(CHEMBL284079 | 4-(2-Chloro-phenyl)-9-methyl-2-(5-p...)
Affinity DataIC50: 60nMAssay Description:In vitro for platelet activating factor receptor antagonist activity in a binding assay using washed whole dog platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50011857(CHEMBL286229 | 4-(2-Chloro-phenyl)-2-[2-(4-isobuty...)
Affinity DataIC50: 80nMAssay Description:In vitro for platelet activating factor receptor antagonist activity in a binding assay using washed whole dog platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50011871(CHEMBL33139 | 4-(2-Chloro-phenyl)-2-(4-isobutyl-ph...)
Affinity DataIC50: 100nMAssay Description:Compound tested in vitro for Platelet activating factor receptor antagonist activity in a binding assay using washed whole dog plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50011878(CHEMBL288098 | 4-(2-Chloro-phenyl)-9-methyl-2-phen...)
Affinity DataIC50: 100nMAssay Description:Compound tested in vitro for Platelet activating factor receptor antagonist activity in a binding assay using washed whole dog plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50011879(CHEMBL369194 | 4-(2-Chloro-phenyl)-2-[2-(4-imidazo...)
Affinity DataIC50: 100nMAssay Description:In vitro for platelet activating factor receptor antagonist activity in a binding assay using washed whole dog platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50011860(CHEMBL286762 | 4-(2-Chloro-phenyl)-2-(2-indan-5-yl...)
Affinity DataIC50: 110nMAssay Description:In vitro for platelet activating factor receptor antagonist activity in a binding assay using washed whole dog platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50011880(CHEMBL32389 | 4-(2-Chloro-phenyl)-2-[2-(4-cyclohex...)
Affinity DataIC50: 120nMAssay Description:In vitro for platelet activating factor receptor antagonist activity in a binding assay using washed whole dog platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50011855(CHEMBL32110 | 4-(2-Chloro-phenyl)-9-methyl-2-napht...)
Affinity DataIC50: 150nMAssay Description:Compound tested in vitro for Platelet activating factor receptor antagonist activity in a binding assay using washed whole dog plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50011881(CHEMBL286557 | 3-[4-(2-Chloro-phenyl)-9-methyl-6H-...)
Affinity DataIC50: 180nMAssay Description:In vitro for platelet activating factor receptor antagonist activity in a binding assay using washed whole dog platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50011858(CHEMBL32327 | 3-[4-(2-Chloro-phenyl)-9-methyl-6H-1...)
Affinity DataIC50: 180nMAssay Description:In vitro for platelet activating factor receptor antagonist activity in a binding assay using washed whole dog platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50000714(3-[4-(2-Chloro-phenyl)-9-methyl-6H-1-thia-5,7,8,9a...)
Affinity DataIC50: 200nMAssay Description:In vitro for platelet activating factor receptor antagonist activity in a binding assay using washed whole dog platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50011883(CHEMBL285035 | 4-(2-Chloro-phenyl)-9-methyl-2-pyri...)
Affinity DataIC50: 250nMAssay Description:In vitro for platelet activating factor receptor antagonist activity in a binding assay using washed whole dog platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50011865(CHEMBL287380 | 3-[4-(2-Chloro-phenyl)-9-methyl-6H-...)
Affinity DataIC50: 260nMAssay Description:Compound tested in vitro for Platelet activating factor receptor antagonist activity in a binding assay using washed whole dog plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50011874(CHEMBL33857 | 4-(2-Chloro-phenyl)-2-(4-cyclohexyl-...)
Affinity DataIC50: 300nMAssay Description:In vitro for platelet activating factor receptor antagonist activity in a binding assay using washed whole dog platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50011875(2-Bromo-4-(2-chloro-phenyl)-9-methyl-6H-1-thia-5,7...)
Affinity DataIC50: 300nMAssay Description:In vitro for platelet activating factor receptor antagonist activity in a binding assay using washed whole dog platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50011628(CHEMBL20359 | 4-(2-Chloro-phenyl)-2-iodo-9-methyl-...)
Affinity DataIC50: 370nMAssay Description:In vitro for platelet activating factor receptor antagonist activity in a binding assay using washed whole dog platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50011854(CHEMBL284280 | 4-(2-Chloro-phenyl)-2-indan-5-yleth...)
Affinity DataIC50: 380nMAssay Description:In vitro for platelet activating factor receptor antagonist activity in a binding assay using washed whole dog platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50011863(CHEMBL285926 | 4-(2-Chloro-phenyl)-9-methyl-2-(2-p...)
Affinity DataIC50: 400nMAssay Description:Compound tested in vitro for Platelet activating factor receptor antagonist activity in a binding assay using washed whole dog plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50011873(CHEMBL286337 | 4-(2-Chloro-phenyl)-9-methyl-2-[2-(...)
Affinity DataIC50: 400nMAssay Description:In vitro for platelet activating factor receptor antagonist activity in a binding assay using washed whole dog platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50011867(CHEMBL32932 | 4-(2-Chloro-phenyl)-9-methyl-2-(2,2,...)
Affinity DataIC50: 400nMAssay Description:In vitro for platelet activating factor receptor antagonist activity in a binding assay using washed whole dog platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50011884(CHEMBL34796 | 4-(2-Chloro-phenyl)-2-(2,3-dihydro-b...)
Affinity DataIC50: 420nMAssay Description:In vitro for platelet activating factor receptor antagonist activity in a binding assay using washed whole dog platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50011882(CHEMBL285199 | 3-[4-(2-Chloro-phenyl)-9-methyl-6H-...)
Affinity DataIC50: 420nMAssay Description:In vitro for platelet activating factor receptor antagonist activity in a binding assay using washed whole dog platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50011870(CHEMBL285067 | 3-[4-(2-Chloro-phenyl)-9-methyl-6H-...)
Affinity DataIC50: 450nMAssay Description:In vitro for platelet activating factor receptor antagonist activity in a binding assay using washed whole dog platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50011869(CHEMBL32767 | 2-(4-Butyl-phenylethynyl)-4-(2-chlor...)
Affinity DataIC50: 650nMAssay Description:In vitro for platelet activating factor receptor antagonist activity in a binding assay using washed whole dog platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50011859(CHEMBL32303 | 5-[4-(2-Chloro-phenyl)-9-methyl-6H-1...)
Affinity DataIC50: 1.00E+3nMAssay Description:In vitro for platelet activating factor receptor antagonist activity in a binding assay using washed whole dog platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50011856(CHEMBL33217 | {5-[4-(2-Chloro-phenyl)-9-methyl-6H-...)
Affinity DataIC50: 1.00E+3nMAssay Description:In vitro for platelet activating factor receptor antagonist activity in a binding assay using washed whole dog platelets.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed