Compile Data Set for Download or QSAR
Report error Found 28 Enz. Inhib. hit(s) with all data for entry = 50039108
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50423773(A-1544750 | CEP-701 | KT-5555 | SP924 | LESTAURTIN...)
Affinity DataIC50: 5nMAssay Description:Inhibition of FLT3 by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50313606(Sodium-3-[hydroxyimino]-2'-oxo-1,3,1',2'-tetrahydr...)
Affinity DataIC50: 9nMAssay Description:Inhibition of FLT3 by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50313604(5'-Fluoro-1H,1'H-[2,3']biindolylidene-3,2'-dione 3...)
Affinity DataIC50: 15nMAssay Description:Inhibition of FLT3 by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50313610(5'-Methyl-1H,1'H-[2,3']biindolylidene-3,2'-dione 3...)
Affinity DataIC50: 28nMAssay Description:Inhibition of FLT3 by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM7393(Indirubin-3 -monoxime | 3-[(2Z,3E)-3-(hydroxyimino...)
Affinity DataIC50: 33nMAssay Description:Inhibition of FLT3 by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50304109(5'-Nitro-1H,1'H-[2,3']biindolylidene-3,2'-dione 3-...)
Affinity DataIC50: 62nMAssay Description:Inhibition of FLT3 by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50313609(5'-Chloro-1H,1'H-[2,3']biindolylidene-3,2'-dione 3...)
Affinity DataIC50: 82nMAssay Description:Inhibition of FLT3 by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50304112((Z)-5'-Amino-1H,1'H-[2,3']biindolylidene-3,2'-dion...)
Affinity DataIC50: 128nMAssay Description:Inhibition of FLT3 by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50313614(5'-Methyl-1H,1'H-[2,3']biindolylidene-3,2'-dione |...)
Affinity DataIC50: 209nMAssay Description:Inhibition of FLT3 by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50313613(5'-Chloro-1H,1'H-[2,3']biindolylidene-3,2'-dione |...)
Affinity DataIC50: 212nMAssay Description:Inhibition of FLT3 by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50313615(Sodium-3,2'-dioxo-1,3,1',2'-tetrahydro-[2,3']biind...)
Affinity DataIC50: 280nMAssay Description:Inhibition of FLT3 by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50304110((Z)-5'-Amino-1H,1'H-[2,3']biindolylidene-3,2'-dion...)
Affinity DataIC50: 359nMAssay Description:Inhibition of FLT3 by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM7492(3-[(2Z,3E)-3-(hydroxyimino)-2,3-dihydro-1H-indol-2...)
Affinity DataIC50: 418nMAssay Description:Inhibition of FLT3 by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50313608(5',7'-Dimethyl-1H,1'H-[2,3']biindolylidene-3,2'-di...)
Affinity DataIC50: 952nMAssay Description:Inhibition of FLT3 by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50313604(5'-Fluoro-1H,1'H-[2,3']biindolylidene-3,2'-dione 3...)
Affinity DataIC50: 1.27E+3nMAssay Description:Inhibition of Aurora A by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50313604(5'-Fluoro-1H,1'H-[2,3']biindolylidene-3,2'-dione 3...)
Affinity DataIC50: 1.53E+3nMAssay Description:Inhibition of VEGFR2 by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50313612(5'-Iodo-1H,1'H-[2,3']biindolylidene-3,2'-dione | C...)
Affinity DataIC50: 4.72E+3nMAssay Description:Inhibition of FLT3 by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50304116((Z)-5'-Nitro-1H,1'H-[2,3']biindolylidene-3,2'-dion...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of FLT3 by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50313617(1-Acetyl-1H,1'H-[2,3']biindolylidene-3,2'-dione | ...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of FLT3 by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50349806(INDIRUBIN)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of FLT3 by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed
TargetMacrophage-stimulating protein receptor(Human)
Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50313604(5'-Fluoro-1H,1'H-[2,3']biindolylidene-3,2'-dione 3...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Ron by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed
TargetInsulin receptor(Human)
Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50313604(5'-Fluoro-1H,1'H-[2,3']biindolylidene-3,2'-dione 3...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of insulin receptor by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50313611(5'-Trifluoromethoxy-1H,1'H-[2,3']biindolylidene-3,...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of FLT3 by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50313607(5'-Chloro-7'-methyl-1H,1'H-[2,3']biindolylidene-3,...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of FLT3 by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50313604(5'-Fluoro-1H,1'H-[2,3']biindolylidene-3,2'-dione 3...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of EGFR by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50304121((Z)-5-Bromo-5'-nitro-1H,1'H-[2,3']biindolylidene-3...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of FLT3 by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50313604(5'-Fluoro-1H,1'H-[2,3']biindolylidene-3,2'-dione 3...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Met by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Institute of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50313616(5'-Fluoro-1H,1'H-[2,3']biindolylidene-3,2'-dione |...)
Affinity DataIC50: 1.01E+4nMAssay Description:Inhibition of FLT3 by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed