Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with all data for entry = 50039053
TargetProgesterone receptor(Human)
University of Quebec At Trois-Rivieres

Curated by ChEMBL
LigandPNGBDBM18627(Mifeprex | (10S,11S,14S,15S,17R)-17-[4-(dimethylam...)
Affinity DataIC50: 0.0500nMAssay Description:Antiprogestagenic activity at progesterone receptor in human T47D cells assessed as inhibition of progesterone-induced alkaline phosphatase activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2012
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
University of Quebec At Trois-Rivieres

Curated by ChEMBL
LigandPNGBDBM50292750(17beta-Hydroxy-11beta-[4-(methylamino)-phenyl]-17a...)
Affinity DataIC50: 0.170nMAssay Description:Antiprogestagenic activity at progesterone receptor in human T47D cells assessed as inhibition of progesterone-induced alkaline phosphatase activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2012
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
University of Quebec At Trois-Rivieres

Curated by ChEMBL
LigandPNGBDBM50292761(17beta-Hydroxy-11beta-[4-(5-carboxy-N-methylpentyl...)
Affinity DataIC50: 0.440nMAssay Description:Antiprogestagenic activity at progesterone receptor in human T47D cells assessed as inhibition of progesterone-induced alkaline phosphatase activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2012
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
University of Quebec At Trois-Rivieres

Curated by ChEMBL
LigandPNGBDBM50292760(3-N-Methyl-N-[4-(11beta,17beta)-17-hydroxy-3-oxo-1...)
Affinity DataIC50: 34nMAssay Description:Antiprogestagenic activity at progesterone receptor in human T47D cells assessed as inhibition of progesterone-induced alkaline phosphatase activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2012
Entry Details Article
PubMed