Compile Data Set for Download or QSAR
Report error Found 70 Enz. Inhib. hit(s) with all data for entry = 50031125
TargetEpidermal growth factor receptor(Human)
Curis

Curated by ChEMBL
LigandPNGBDBM50307778(7-(4-(3-Chloro-4-fluorophenylamino)-7-methoxyquina...)
Affinity DataIC50: 2nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Curis

Curated by ChEMBL
LigandPNGBDBM50307783(N1-(4-(3-chloro-4-fluorophenylamino)-7-methoxyquin...)
Affinity DataIC50: 2.10nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Curis

Curated by ChEMBL
LigandPNGBDBM50307768(7-(4-(3-Ethynylphenylamino)-7-methoxyquinazolin-6-...)
Affinity DataIC50: 2.40nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Curis

Curated by ChEMBL
LigandPNGBDBM50307775(7-(4-(3-Chloro-4-fluorophenylamino)-7-methoxyquina...)
Affinity DataIC50: 3.10nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Curis

Curated by ChEMBL
LigandPNGBDBM50307773(7-(4-(3-Chloro-4-fluorophenylamino)-7-methoxyquina...)
Affinity DataIC50: 3.40nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Curis

Curated by ChEMBL
LigandPNGBDBM50307768(7-(4-(3-Ethynylphenylamino)-7-methoxyquinazolin-6-...)
Affinity DataIC50: 4.5nMAssay Description:Inhibition of human HDAC1 expressed in Escherichia coliMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Curis

Curated by ChEMBL
LigandPNGBDBM50307774(6-(4-(3-Ethynylphenylamino)-7-methoxyquinazolin-6-...)
Affinity DataIC50: 4.60nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetHistone deacetylase 6(Human)
Curis

Curated by ChEMBL
LigandPNGBDBM50307768(7-(4-(3-Ethynylphenylamino)-7-methoxyquinazolin-6-...)
Affinity DataIC50: 5.10nMAssay Description:Inhibition of human HDAC6 expressed in Escherichia coliMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Curis

Curated by ChEMBL
LigandPNGBDBM50307790(7-(4-(3-chloro-4-fluorophenylamino)-6-methoxyquina...)
Affinity DataIC50: 7nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Curis

Curated by ChEMBL
LigandPNGBDBM50307769(3-(4-(3-chloro-4-fluorophenylamino)-7-methoxyquina...)
Affinity DataIC50: 7.10nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Curis

Curated by ChEMBL
LigandPNGBDBM50307770(4-(4-(3-Chloro-4-fluorophenylamino)-7-methoxyquina...)
Affinity DataIC50: 7.80nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Curis

Curated by ChEMBL
LigandPNGBDBM50307791(7-(4-(3-Ethynylphenylamino)-6-methoxyquinazolin-7-...)
Affinity DataIC50: 8.20nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Curis

Curated by ChEMBL
LigandPNGBDBM50307777(7-(4-(3-Chloro-4-(3-fluorobenzyloxy)phenylamino)-7...)
Affinity DataIC50: 9.10nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetHistone deacetylase 3(Human)
Curis

Curated by ChEMBL
LigandPNGBDBM50307768(7-(4-(3-Ethynylphenylamino)-7-methoxyquinazolin-6-...)
Affinity DataIC50: 9.10nMAssay Description:Inhibition of human HDAC3 expressed in Escherichia coliMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Curis

Curated by ChEMBL
LigandPNGBDBM50307771(5-(4-(3-Chloro-4-fluorophenylamino)-7-methoxyquina...)
Affinity DataIC50: 9.40nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
LigandPNGBDBM5445(N-{3-chloro-4-[(3-fluorophenyl)methoxy]phenyl}-6-(...)
Affinity DataIC50: 10nMAssay Description:Inhibition of HER2More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
LigandPNGBDBM50307777(7-(4-(3-Chloro-4-(3-fluorobenzyloxy)phenylamino)-7...)
Affinity DataIC50: 10nMAssay Description:Inhibition of HER2More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Curis

Curated by ChEMBL
LigandPNGBDBM50307782(7-(4-(3-Chloro-4-fluorophenylamino)-7-(2-methoxyet...)
Affinity DataIC50: 10nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
LigandPNGBDBM50307769(3-(4-(3-chloro-4-fluorophenylamino)-7-methoxyquina...)
Affinity DataIC50: 11nMAssay Description:Inhibition of HER2More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetHistone deacetylase 5(Human)
Curis

Curated by ChEMBL
LigandPNGBDBM50307768(7-(4-(3-Ethynylphenylamino)-7-methoxyquinazolin-6-...)
Affinity DataIC50: 11nMAssay Description:Inhibition of human HDAC5 expressed in Escherichia coliMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Curis

Curated by ChEMBL
LigandPNGBDBM5445(N-{3-chloro-4-[(3-fluorophenyl)methoxy]phenyl}-6-(...)
Affinity DataIC50: 11nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
LigandPNGBDBM50307770(4-(4-(3-Chloro-4-fluorophenylamino)-7-methoxyquina...)
Affinity DataIC50: 12nMAssay Description:Inhibition of HER2More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetHistone deacetylase 2(Human)
Curis

Curated by ChEMBL
LigandPNGBDBM50307768(7-(4-(3-Ethynylphenylamino)-7-methoxyquinazolin-6-...)
Affinity DataIC50: 13nMAssay Description:Inhibition of human HDAC2 expressed in Escherichia coliMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetHistone deacetylase 4(Human)
Curis

Curated by ChEMBL
LigandPNGBDBM50307768(7-(4-(3-Ethynylphenylamino)-7-methoxyquinazolin-6-...)
Affinity DataIC50: 13nMAssay Description:Inhibition of human HDAC4 expressed in Escherichia coliMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Curis

Curated by ChEMBL
LigandPNGBDBM50307787((R)-N-Hydroxy-7-(7-methoxy-4-(1-phenylethylamino)q...)
Affinity DataIC50: 13nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Curis

Curated by ChEMBL
LigandPNGBDBM50307772(5-(4-(3-Ethynylphenylamino)-7-methoxyquinazolin-6-...)
Affinity DataIC50: 15nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
LigandPNGBDBM50307771(5-(4-(3-Chloro-4-fluorophenylamino)-7-methoxyquina...)
Affinity DataIC50: 15nMAssay Description:Inhibition of HER2More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Curis

Curated by ChEMBL
LigandPNGBDBM50307779(7-(4-(3-chloro-4-fluorophenylamino)-7-methoxyquina...)
Affinity DataIC50: 15nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
LigandPNGBDBM50307768(7-(4-(3-Ethynylphenylamino)-7-methoxyquinazolin-6-...)
Affinity DataIC50: 16nMAssay Description:Inhibition of HER2More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
LigandPNGBDBM50307775(7-(4-(3-Chloro-4-fluorophenylamino)-7-methoxyquina...)
Affinity DataIC50: 19nMAssay Description:Inhibition of HER2More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
LigandPNGBDBM50307773(7-(4-(3-Chloro-4-fluorophenylamino)-7-methoxyquina...)
Affinity DataIC50: 20nMAssay Description:Inhibition of HER2More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
LigandPNGBDBM50307783(N1-(4-(3-chloro-4-fluorophenylamino)-7-methoxyquin...)
Affinity DataIC50: 20nMAssay Description:Inhibition of HER2More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
LigandPNGBDBM50307778(7-(4-(3-Chloro-4-fluorophenylamino)-7-methoxyquina...)
Affinity DataIC50: 24nMAssay Description:Inhibition of HER2More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
LigandPNGBDBM50307782(7-(4-(3-Chloro-4-fluorophenylamino)-7-(2-methoxyet...)
Affinity DataIC50: 24nMAssay Description:Inhibition of HER2More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetPolyamine deacetylase HDAC10(Human)
Curis

Curated by ChEMBL
LigandPNGBDBM50307768(7-(4-(3-Ethynylphenylamino)-7-methoxyquinazolin-6-...)
Affinity DataIC50: 26nMAssay Description:Inhibition of human HDAC10 expressed in Escherichia coliMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
LigandPNGBDBM50307787((R)-N-Hydroxy-7-(7-methoxy-4-(1-phenylethylamino)q...)
Affinity DataIC50: 28nMAssay Description:Inhibition of HER2More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Curis

Curated by ChEMBL
LigandPNGBDBM50307776(7-(4-(3-Ethynyl-4-fluorophenylamino)-7-methoxyquin...)
Affinity DataIC50: 29nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
LigandPNGBDBM50307774(6-(4-(3-Ethynylphenylamino)-7-methoxyquinazolin-6-...)
Affinity DataIC50: 38nMAssay Description:Inhibition of HER2More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
LigandPNGBDBM50307772(5-(4-(3-Ethynylphenylamino)-7-methoxyquinazolin-6-...)
Affinity DataIC50: 38nMAssay Description:Inhibition of HER2More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
LigandPNGBDBM50307781(7-(4-(3-Chloro-4-fluorophenylamino)quinazolin-6-yl...)
Affinity DataIC50: 44nMAssay Description:Inhibition of HER2More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Curis

Curated by ChEMBL
LigandPNGBDBM5446(Erlotinib | OSI-774 | N-(3-ethynylphenyl)-6,7-bis(...)
Affinity DataIC50: 48nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM50307791(7-(4-(3-Ethynylphenylamino)-6-methoxyquinazolin-7-...)
Affinity DataIC50: 52nMAssay Description:Inhibition of HER2More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetHistone deacetylase 9(Human)
Curis

Curated by ChEMBL
LigandPNGBDBM50307768(7-(4-(3-Ethynylphenylamino)-7-methoxyquinazolin-6-...)
Affinity DataIC50: 67nMAssay Description:Inhibition of human HDAC9 expressed in Escherichia coliMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
LigandPNGBDBM50307790(7-(4-(3-chloro-4-fluorophenylamino)-6-methoxyquina...)
Affinity DataIC50: 71nMAssay Description:Inhibition of HER2More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Curis

Curated by ChEMBL
LigandPNGBDBM50307780(7-(4-(3-Chloro-4-fluorobenzylamino)-7-methoxyquina...)
Affinity DataIC50: 72nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
LigandPNGBDBM50307776(7-(4-(3-Ethynyl-4-fluorophenylamino)-7-methoxyquin...)
Affinity DataIC50: 77nMAssay Description:Inhibition of HER2More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetHistone deacetylase 8(Human)
Curis

Curated by ChEMBL
LigandPNGBDBM50307768(7-(4-(3-Ethynylphenylamino)-7-methoxyquinazolin-6-...)
Affinity DataIC50: 80nMAssay Description:Inhibition of human HDAC8 expressed in Escherichia coliMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Curis

Curated by ChEMBL
LigandPNGBDBM50307781(7-(4-(3-Chloro-4-fluorophenylamino)quinazolin-6-yl...)
Affinity DataIC50: 84nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Curis

Curated by ChEMBL
LigandPNGBDBM50307784(7-(4-(Benzylamino)-7-methoxyquinazolin-6-yloxy)-N-...)
Affinity DataIC50: 99nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Curis

Curated by ChEMBL
LigandPNGBDBM50307788((R)-7-(4-(1-(4-Fluorophenyl)ethylamino)-7-methoxyq...)
Affinity DataIC50: 126nMAssay Description:Inhibition of EGFRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
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