Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) with all data for entry = 50039104
TargetPeroxisome proliferator-activated receptor alpha(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM28681(cid_5281055 | [3H]rosiglitazone | CHEMBL121 | ROSI...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human recombinant PPARalpha LBD expressed in african green monkey COS7 cells coexpressing GAL4 by luciferase reporter gene transa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50313117((Z)-5-(4-(3-(Piperidin-1-yl)propoxy)benzylidene)-2...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human recombinant PPARalpha LBD expressed in african green monkey COS7 cells coexpressing GAL4 by luciferase reporter gene transa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM28681(cid_5281055 | [3H]rosiglitazone | CHEMBL121 | ROSI...)
Affinity DataEC50:  30nMAssay Description:Agonist activity at human recombinant PPARgamma1 LBD expressed in african green monkey COS7 cells coexpressing GAL4 by luciferase reporter gene trans...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM28681(cid_5281055 | [3H]rosiglitazone | CHEMBL121 | ROSI...)
Affinity DataEC50:  100nMAssay Description:Agonist activity at human recombinant PPARgamma2 LBD expressed in african green monkey COS7 cells coexpressing GAL4 by luciferase reporter gene trans...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50313117((Z)-5-(4-(3-(Piperidin-1-yl)propoxy)benzylidene)-2...)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human recombinant PPARgamma LBD expressed in african green monkey COS7 cells coexpressing GAL4 by luciferase reporter gene transa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2012
Entry Details Article
PubMed