Compile Data Set for Download or QSAR
Report error Found 28 Enz. Inhib. hit(s) with all data for entry = 50031102
TargetCoagulation factor X(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM19023(BMS-562247 | CHEMBL231779 | 1-(4-methoxyphenyl)-7-...)
Affinity DataKi:  0.0800nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM12657(CHEMBL559015 | 1-[3-(Aminomethyl)phenyl]-N-[3-fluo...)
Affinity DataKi:  0.150nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM12676(DPC 906 | 1-(3-Aminobenzisoxazol-5-yl)-3-trifluoro...)
Affinity DataKi:  0.190nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50307102(7-oxo-1-(3-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-y...)
Affinity DataKi:  0.25nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50307100(1-(3-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)phen...)
Affinity DataKi:  0.400nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50307093(N-(3-fluoro-2'-(methylsulfonyl)biphenyl-4-yl)-1-(3...)
Affinity DataKi:  0.5nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50307099(6-(2'-(((R)-3-hydroxypyrrolidin-1-yl)methyl)biphen...)
Affinity DataKi:  0.840nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50307098(6-(2'-((dimethylamino)methyl)biphenyl-4-yl)-1-(3-(...)
Affinity DataKi:  1.10nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50307097(6-(4-(2-((dimethylamino)methyl)-1H-imidazol-1-yl)p...)
Affinity DataKi:  2nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50307096(6-(2'-(methylsulfonyl)biphenyl-4-yl)-1-(3-(5-oxo-4...)
Affinity DataKi:  2.20nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50307101(3-methyl-1-(3-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-...)
Affinity DataKi:  8.10nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50307092(1-(3-((2-aminoacetamido)methyl)phenyl)-N-(3-fluoro...)
Affinity DataKi:  9nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50307095(1-(3-(5-amino-4H-1,2,4-triazol-3-yl)phenyl)-N-(3-f...)
Affinity DataKi:  15nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50307094(1-(3-(5-amino-1,3,4-thiadiazol-2-yl)phenyl)-N-(3-f...)
Affinity DataKi:  46nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetProthrombin(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM12676(DPC 906 | 1-(3-Aminobenzisoxazol-5-yl)-3-trifluoro...)
Affinity DataKi:  540nMAssay Description:Inhibition of human factor 2aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetProthrombin(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM19023(BMS-562247 | CHEMBL231779 | 1-(4-methoxyphenyl)-7-...)
Affinity DataKi:  3.10E+3nMAssay Description:Inhibition of human factor 2aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetProthrombin(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50307095(1-(3-(5-amino-4H-1,2,4-triazol-3-yl)phenyl)-N-(3-f...)
Affinity DataKi:  4.90E+3nMAssay Description:Inhibition of human factor 2aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetProthrombin(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50307098(6-(2'-((dimethylamino)methyl)biphenyl-4-yl)-1-(3-(...)
Affinity DataKi: >6.00E+3nMAssay Description:Inhibition of human factor 2aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetProthrombin(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50307099(6-(2'-(((R)-3-hydroxypyrrolidin-1-yl)methyl)biphen...)
Affinity DataKi: >6.00E+3nMAssay Description:Inhibition of human factor 2aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetProthrombin(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50307097(6-(4-(2-((dimethylamino)methyl)-1H-imidazol-1-yl)p...)
Affinity DataKi: >6.00E+3nMAssay Description:Inhibition of human factor 2aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetProthrombin(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50307100(1-(3-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)phen...)
Affinity DataKi: >6.00E+3nMAssay Description:Inhibition of human factor 2aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetProthrombin(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50307096(6-(2'-(methylsulfonyl)biphenyl-4-yl)-1-(3-(5-oxo-4...)
Affinity DataKi: >6.00E+3nMAssay Description:Inhibition of human factor 2aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetProthrombin(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50307101(3-methyl-1-(3-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-...)
Affinity DataKi: >6.00E+3nMAssay Description:Inhibition of human factor 2aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetProthrombin(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50307102(7-oxo-1-(3-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-y...)
Affinity DataKi: >6.00E+3nMAssay Description:Inhibition of human factor 2aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetProthrombin(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM12657(CHEMBL559015 | 1-[3-(Aminomethyl)phenyl]-N-[3-fluo...)
Affinity DataKi:  6.00E+3nMAssay Description:Inhibition of human factor 2aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetProthrombin(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50307094(1-(3-(5-amino-1,3,4-thiadiazol-2-yl)phenyl)-N-(3-f...)
Affinity DataKi: >2.10E+4nMAssay Description:Inhibition of human factor 2aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetProthrombin(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50307093(N-(3-fluoro-2'-(methylsulfonyl)biphenyl-4-yl)-1-(3...)
Affinity DataKi: >2.10E+4nMAssay Description:Inhibition of human factor 2aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetProthrombin(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50307092(1-(3-((2-aminoacetamido)methyl)phenyl)-N-(3-fluoro...)
Affinity DataKi: >2.10E+4nMAssay Description:Inhibition of human factor 2aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed