Compile Data Set for Download or QSAR
Report error Found 34 Enz. Inhib. hit(s) with all data for entry = 50031100
TargetC-C chemokine receptor type 4(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50307035(5,7-Dihydroxy-4-methyl-3-(4-methylpiperazin-1-yl)-...)
Affinity DataIC50: 21.2nMAssay Description:Displacement of FITC-CKLF1-C27 from human CCR4 receptor expressed in human HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetC-C chemokine receptor type 4(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50307033(4-(5,7-Dihydroxy-4-methyl-2-oxo-2H-chromen-3-yl)-N...)
Affinity DataIC50: 110nMAssay Description:Displacement of FITC-CKLF1-C27 from human CCR4 receptor expressed in human HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetC-C chemokine receptor type 4(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50307036(3-(4-Ethylpiperazin-1-yl)-5,7-dihydroxy-4-methyl-2...)
Affinity DataIC50: 131nMAssay Description:Displacement of FITC-CKLF1-C27 from human CCR4 receptor expressed in human HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetC-C chemokine receptor type 4(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50307054(4-Methyl-3-(4-methylpiperazin-1-yl)-7-(2-(piperidi...)
Affinity DataIC50: 196nMAssay Description:Displacement of FITC-CKLF1-C27 from human CCR4 receptor expressed in human HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetC-C chemokine receptor type 4(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50307045(5-Hydroxy-7-methoxy-4-methyl-3-(4-methylpiperazin-...)
Affinity DataIC50: 389nMAssay Description:Displacement of FITC-CKLF1-C27 from human CCR4 receptor expressed in human HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetC-C chemokine receptor type 4(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50307044(8-Methyl-7-(4-methylpiperazin-1-yl)-6H-[1,3]dioxol...)
Affinity DataIC50: 420nMAssay Description:Displacement of FITC-CKLF1-C27 from human CCR4 receptor expressed in human HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetC-C chemokine receptor type 4(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50307046(5,7-Dimethoxy-4-methyl-3-(4-methylpiperazin-1-yl)-...)
Affinity DataIC50: 478nMAssay Description:Displacement of FITC-CKLF1-C27 from human CCR4 receptor expressed in human HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetC-C chemokine receptor type 4(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50307052(4-Methyl-3-(4-methylpiperazin-1-yl)-7-(2-(thiophen...)
Affinity DataIC50: 527nMAssay Description:Displacement of FITC-CKLF1-C27 from human CCR4 receptor expressed in human HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetC-C chemokine receptor type 4(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50307031(4-(5,7-Dihydroxy-4-methyl-2-oxo-2H-chromen-3-yl)-N...)
Affinity DataIC50: 539nMAssay Description:Displacement of FITC-CKLF1-C27 from human CCR4 receptor expressed in human HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetC-C chemokine receptor type 4(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50307053(4-Methyl-3-(4-methylpiperazin-1-yl)-7-(2-morpholin...)
Affinity DataIC50: 671nMAssay Description:Displacement of FITC-CKLF1-C27 from human CCR4 receptor expressed in human HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetC-C chemokine receptor type 4(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50307042(7-Hydroxy-4-methyl-3-(4-methylpiperazin-1-yl)-2H-c...)
Affinity DataIC50: 775nMAssay Description:Displacement of FITC-CKLF1-C27 from human CCR4 receptor expressed in human HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetC-C chemokine receptor type 4(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50307043(5-Hydroxy-4,7-dimethyl-3-(4-methylpiperazin-1-yl)-...)
Affinity DataIC50: 1.13E+3nMAssay Description:Displacement of FITC-CKLF1-C27 from human CCR4 receptor expressed in human HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetC-C chemokine receptor type 4(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50307030(4-(5,7-Dihydroxy-4-methyl-2-oxo-2H-chromen-3-yl)-N...)
Affinity DataIC50: 1.32E+3nMAssay Description:Displacement of FITC-CKLF1-C27 from human CCR4 receptor expressed in human HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetC-C chemokine receptor type 4(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50307055(4-Methyl-3-(4-methylpiperazin-1-yl)-7-(2-(pyrrolid...)
Affinity DataIC50: 1.51E+3nMAssay Description:Displacement of FITC-CKLF1-C27 from human CCR4 receptor expressed in human HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetC-C chemokine receptor type 4(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50307024(3-(4-cinnamoylpiperazin-1-yl)-5,7-dihydroxy-4-meth...)
Affinity DataIC50: 1.57E+3nMAssay Description:Displacement of FITC-CKLF1-C27 from human CCR4 receptor expressed in human HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetC-C chemokine receptor type 4(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50307034(N-Benzyl-4-(5,7-dihydroxy-4-methyl-2-oxo-2H-chrome...)
Affinity DataIC50: 1.59E+3nMAssay Description:Displacement of FITC-CKLF1-C27 from human CCR4 receptor expressed in human HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetC-C chemokine receptor type 4(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50307049(7-Ethoxy-4-methyl-3-(4-methylpiperazin-1-yl)-2H-ch...)
Affinity DataIC50: 1.64E+3nMAssay Description:Displacement of FITC-CKLF1-C27 from human CCR4 receptor expressed in human HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetC-C chemokine receptor type 4(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50307029(N-(4-(4-(5,7-Dihydroxy-4-methyl-2-oxo-2H-chromen-3...)
Affinity DataIC50: 2.56E+3nMAssay Description:Displacement of FITC-CKLF1-C27 from human CCR4 receptor expressed in human HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetC-C chemokine receptor type 4(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50307050(7-(4-Ethylcyclohexyloxy)-4-methyl-3-(4-methylpiper...)
Affinity DataIC50: 3.12E+3nMAssay Description:Displacement of FITC-CKLF1-C27 from human CCR4 receptor expressed in human HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetC-C chemokine receptor type 4(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50307025(3-(4-Acryloylpiperazin-1-yl)-5,7-dihydroxy-4-methy...)
Affinity DataIC50: 4.24E+3nMAssay Description:Displacement of FITC-CKLF1-C27 from human CCR4 receptor expressed in human HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetC-C chemokine receptor type 4(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50307056(5,7-Dihydroxy-4-methyl-3-(piperazin-1-yl)-2H-chrom...)
Affinity DataIC50: 4.36E+3nMAssay Description:Displacement of FITC-CKLF1-C27 from human CCR4 receptor expressed in human HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetC-C chemokine receptor type 4(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50307027(3-(4-benzoylpiperazin-1-yl)-5,7-dihydroxy-4-methyl...)
Affinity DataIC50: 4.36E+3nMAssay Description:Displacement of FITC-CKLF1-C27 from human CCR4 receptor expressed in human HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetC-C chemokine receptor type 4(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50307047(7-(Dimethylamino)-4-methyl-3-(4-methylpiperazin-1-...)
Affinity DataIC50: 4.76E+3nMAssay Description:Displacement of FITC-CKLF1-C27 from human CCR4 receptor expressed in human HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetC-C chemokine receptor type 4(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50307048(7-Methoxy-4-methyl-3-(4-methylpiperazin-1-yl)-2H-c...)
Affinity DataIC50: 5.21E+3nMAssay Description:Displacement of FITC-CKLF1-C27 from human CCR4 receptor expressed in human HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetC-C chemokine receptor type 4(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50307032(4-(5,7-Dihydroxy-4-methyl-2-oxo-2H-chromen-3-yl)-N...)
Affinity DataIC50: 6.00E+3nMAssay Description:Displacement of FITC-CKLF1-C27 from human CCR4 receptor expressed in human HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetC-C chemokine receptor type 4(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50307028(5,7-Dihydroxy-4-methyl-3-(4-(phenylsulfonyl)pipera...)
Affinity DataIC50: 6.04E+3nMAssay Description:Displacement of FITC-CKLF1-C27 from human CCR4 receptor expressed in human HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetC-C chemokine receptor type 4(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50307051(7-(4-Methoxybenzyloxy)-4-methyl-3-(4-methylpiperaz...)
Affinity DataIC50: 7.32E+3nMAssay Description:Displacement of FITC-CKLF1-C27 from human CCR4 receptor expressed in human HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetC-C chemokine receptor type 4(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50307026(3-(4-(2-Chloroacetyl)piperazin-1-yl)-5,7-dihydroxy...)
Affinity DataIC50: 8.58E+3nMAssay Description:Displacement of FITC-CKLF1-C27 from human CCR4 receptor expressed in human HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetC-C chemokine receptor type 4(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50307041(3-(4-(2-Ethylbutyl)piperazin-1-yl)-5,7-dihydroxy-4...)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of FITC-CKLF1-C27 from human CCR4 receptor expressed in human HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetC-C chemokine receptor type 4(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50307038(5,7-Dihydroxy-3-(4-(2-methoxyphenyl)piperazin-1-yl...)
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of FITC-CKLF1-C27 from human CCR4 receptor expressed in human HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetC-C chemokine receptor type 4(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50307037(5,7-Dihydroxy-4-methyl-3-(4-(3-(trifluoromethyl)ph...)
Affinity DataIC50: 1.51E+4nMAssay Description:Displacement of FITC-CKLF1-C27 from human CCR4 receptor expressed in human HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetC-C chemokine receptor type 4(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50307040(3-(4-(2,3-Dimethylphenyl)piperazin-1-yl)-5,7-dihyd...)
Affinity DataIC50: 3.13E+4nMAssay Description:Displacement of FITC-CKLF1-C27 from human CCR4 receptor expressed in human HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetC-C chemokine receptor type 4(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50307039(3-(4-(4-Fluorophenyl)piperazin-1-yl)-5,7-dihydroxy...)
Affinity DataIC50: 5.85E+4nMAssay Description:Displacement of FITC-CKLF1-C27 from human CCR4 receptor expressed in human HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetC-C chemokine receptor type 4(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50307057(2-amino-N-((2S,3R)-1-(2,6-dioxopiperidin-3-ylamino...)
Affinity DataIC50: 8.36E+5nMAssay Description:Displacement of FITC-CKLF1-C27 from human CCR4 receptor expressed in human HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed