Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with all data for entry = 50031278
TargetLysophosphatidic acid receptor 1(Human)
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50148348(lysophosphatidic acid | 1-oleoyl lysophosphatidic ...)
Affinity DataEC50:  31nMAssay Description:Agonist activity at LPA1 expressed in human chem1 cells assessed as intracellular calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 3(Human)
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50148348(lysophosphatidic acid | 1-oleoyl lysophosphatidic ...)
Affinity DataEC50:  120nMAssay Description:Agonist activity at LPA3 expressed in human chem1 cells assessed as intracellular calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 5(Human)
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50148348(lysophosphatidic acid | 1-oleoyl lysophosphatidic ...)
Affinity DataEC50:  12nMAssay Description:Agonist activity at LPA5 expressed in human chem1 cells assessed as intracellular calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50170859(3-(4-(4-((1-(2-chlorophenyl)ethoxy)carbonylamino)-...)
Affinity DataIC50: 46nMAssay Description:Antagonist activity at LPA1 expressed in human chem1 cells assessed as effect on intracellular calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed