Compile Data Set for Download or QSAR
Report error Found 62 Enz. Inhib. hit(s) with all data for entry = 50030910
TargetDelta-type opioid receptor(Human)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50037134((-)-trans-3-Cyclopropylmethyl-2,3,4,4aalpha,5,6,7,...)
Affinity DataKd:  20nMAssay Description:Binding affinity to human delta opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50037134((-)-trans-3-Cyclopropylmethyl-2,3,4,4aalpha,5,6,7,...)
Affinity DataKd:  0.220nMAssay Description:Binding affinity to human mu opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50037134((-)-trans-3-Cyclopropylmethyl-2,3,4,4aalpha,5,6,7,...)
Affinity DataKi:  0.0800nMAssay Description:Displacement of [125I]OXY from human mu opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50037134((-)-trans-3-Cyclopropylmethyl-2,3,4,4aalpha,5,6,7,...)
Affinity DataKi:  0.100nMAssay Description:Displacement of [125I]OXY from human kappa opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50037134((-)-trans-3-Cyclopropylmethyl-2,3,4,4aalpha,5,6,7,...)
Affinity DataKi:  0.100nMAssay Description:Displacement of [125I]OXY from human kappa opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50303852((-)-trans-3-(2-Phenylethyl)-2,3,4,4aalpha,5,6,7,7a...)
Affinity DataKi:  0.300nMAssay Description:Displacement of [125I]OXY from human mu opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50303852((-)-trans-3-(2-Phenylethyl)-2,3,4,4aalpha,5,6,7,7a...)
Affinity DataKi:  0.300nMAssay Description:Binding affinity to human mu opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50303848((-)-trans-3-Methyl-2,3,4,4aalpha,5,6,7,7aalpha-oct...)
Affinity DataKi:  0.650nMAssay Description:Displacement of [125I]OXY from human mu opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50303848((-)-trans-3-Methyl-2,3,4,4aalpha,5,6,7,7aalpha-oct...)
Affinity DataKi:  0.650nMAssay Description:Binding affinity to human mu opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50000788([17-(2,3-3H-2-propenyl)]-4, 5a -epoxy-3,14-dihydro...)
Affinity DataKi:  0.980nMAssay Description:Binding affinity to human mu opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetDelta-type opioid receptor(Human)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50037134((-)-trans-3-Cyclopropylmethyl-2,3,4,4aalpha,5,6,7,...)
Affinity DataKi:  2nMAssay Description:Displacement of [125I]OXY from human delta opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50001033(3-But-2-enyl-6,11-dimethyl-1,2,3,4,5,6-hexahydro-2...)
Affinity DataKi:  2.20nMAssay Description:Displacement of [125I]OXY from human kappa opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50000788([17-(2,3-3H-2-propenyl)]-4, 5a -epoxy-3,14-dihydro...)
Affinity DataKi:  3nMAssay Description:Displacement of [125I]OXY from human kappa opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50001033(3-But-2-enyl-6,11-dimethyl-1,2,3,4,5,6-hexahydro-2...)
Affinity DataKi:  3.90nMAssay Description:Displacement of [125I]OXY from human mu opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50303852((-)-trans-3-(2-Phenylethyl)-2,3,4,4aalpha,5,6,7,7a...)
Affinity DataKi:  6nMAssay Description:Displacement of [125I]OXY from human delta opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Rat)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50035131((1S,9S,13S)-1,13-dimethyl-10-(3-methylbut-2-enyl)-...)
Affinity DataKi:  6nMAssay Description:Displacement of [3H](+)-pentazocine from sigma1 receptor in rat brain homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50303848((-)-trans-3-Methyl-2,3,4,4aalpha,5,6,7,7aalpha-oct...)
Affinity DataKi:  14nMAssay Description:Displacement of [125I]OXY from human kappa opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50303848((-)-trans-3-Methyl-2,3,4,4aalpha,5,6,7,7aalpha-oct...)
Affinity DataKi:  14nMAssay Description:Displacement of [125I]OXY from human kappa opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50303852((-)-trans-3-(2-Phenylethyl)-2,3,4,4aalpha,5,6,7,7a...)
Affinity DataKi:  15nMAssay Description:Displacement of [125I]OXY from human kappa opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50303852((-)-trans-3-(2-Phenylethyl)-2,3,4,4aalpha,5,6,7,7a...)
Affinity DataKi:  15nMAssay Description:Displacement of [125I]OXY from human kappa opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Rat)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50001033(3-But-2-enyl-6,11-dimethyl-1,2,3,4,5,6-hexahydro-2...)
Affinity DataKi:  16nMAssay Description:Displacement of [3H](+)-pentazocine from sigma1 receptor in rat brain homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50303853((+)-trans-9-Methoxy-3-(2-phenylethyl)-2,3,4,4aalph...)
Affinity DataKi:  24nMAssay Description:Binding affinity to human mu opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50303853((+)-trans-9-Methoxy-3-(2-phenylethyl)-2,3,4,4aalph...)
Affinity DataKi:  24nMAssay Description:Displacement of [125I]OXY from human mu opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50001033(3-But-2-enyl-6,11-dimethyl-1,2,3,4,5,6-hexahydro-2...)
Affinity DataKi:  49nMAssay Description:Displacement of [125I]OXY from human delta opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50000788([17-(2,3-3H-2-propenyl)]-4, 5a -epoxy-3,14-dihydro...)
Affinity DataKi:  51nMAssay Description:Displacement of [125I]OXY from human delta opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Rat)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50303850((-)-trans-3-Cyclopropylmethyl-9-methoxy-2,3,4,4aal...)
Affinity DataKi:  62nMAssay Description:Displacement of [3H](+)-pentazocine from sigma1 receptor in rat brain homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Rat)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50303850((-)-trans-3-Cyclopropylmethyl-9-methoxy-2,3,4,4aal...)
Affinity DataKi:  62nMAssay Description:Displacement of [3H](+)-pentazocine from sigma1 receptor in rat brain homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Rat)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50037134((-)-trans-3-Cyclopropylmethyl-2,3,4,4aalpha,5,6,7,...)
Affinity DataKi:  201nMAssay Description:Displacement of [3H](+)-pentazocine from sigma1 receptor in rat brain homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Rat)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50037134((-)-trans-3-Cyclopropylmethyl-2,3,4,4aalpha,5,6,7,...)
Affinity DataKi:  201nMAssay Description:Displacement of [3H](+)-pentazocine from sigma1 receptor in rat brain homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50303847((-)-trans-9-Methoxy-3-methyl-2,3,4,4aalpha,5,6,7,7...)
Affinity DataKi:  236nMAssay Description:Displacement of [125I]OXY from human mu opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50303847((-)-trans-9-Methoxy-3-methyl-2,3,4,4aalpha,5,6,7,7...)
Affinity DataKi:  236nMAssay Description:Binding affinity to human mu opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Rat)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50303852((-)-trans-3-(2-Phenylethyl)-2,3,4,4aalpha,5,6,7,7a...)
Affinity DataKi:  239nMAssay Description:Displacement of [3H](+)-pentazocine from sigma1 receptor in rat brain homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Rat)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50303852((-)-trans-3-(2-Phenylethyl)-2,3,4,4aalpha,5,6,7,7a...)
Affinity DataKi:  239nMAssay Description:Displacement of [3H](+)-pentazocine from sigma1 receptor in rat brain homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50303853((+)-trans-9-Methoxy-3-(2-phenylethyl)-2,3,4,4aalph...)
Affinity DataKi:  490nMAssay Description:Displacement of [125I]OXY from human delta opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Rat)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50303853((+)-trans-9-Methoxy-3-(2-phenylethyl)-2,3,4,4aalph...)
Affinity DataKi:  560nMAssay Description:Displacement of [3H](+)-pentazocine from sigma1 receptor in rat brain homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Rat)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50303853((+)-trans-9-Methoxy-3-(2-phenylethyl)-2,3,4,4aalph...)
Affinity DataKi:  560nMAssay Description:Displacement of [3H](+)-pentazocine from sigma1 receptor in rat brain homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50303851((+)-cis-3-Methyl-2,3,4,4aalpha,5,6,7,7aalpha-octah...)
Affinity DataKi:  565nMAssay Description:Displacement of [125I]OXY from human kappa opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50303851((+)-cis-3-Methyl-2,3,4,4aalpha,5,6,7,7aalpha-octah...)
Affinity DataKi:  565nMAssay Description:Displacement of [125I]OXY from human kappa opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50303853((+)-trans-9-Methoxy-3-(2-phenylethyl)-2,3,4,4aalph...)
Affinity DataKi:  1.14E+3nMAssay Description:Displacement of [125I]OXY from human kappa opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50303853((+)-trans-9-Methoxy-3-(2-phenylethyl)-2,3,4,4aalph...)
Affinity DataKi:  1.14E+3nMAssay Description:Displacement of [125I]OXY from human kappa opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50303847((-)-trans-9-Methoxy-3-methyl-2,3,4,4aalpha,5,6,7,7...)
Affinity DataKi:  3.47E+3nMAssay Description:Displacement of [125I]OXY from human kappa opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50303847((-)-trans-9-Methoxy-3-methyl-2,3,4,4aalpha,5,6,7,7...)
Affinity DataKi:  3.47E+3nMAssay Description:Displacement of [125I]OXY from human kappa opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50303850((-)-trans-3-Cyclopropylmethyl-9-methoxy-2,3,4,4aal...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I]OXY from human mu opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50303847((-)-trans-9-Methoxy-3-methyl-2,3,4,4aalpha,5,6,7,7...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I]OXY from human delta opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50303849((-)-cis-9-Methoxy-3-methyl-2,3,4,4aalpha,5,6,7,7aa...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I]OXY from human kappa opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50303848((-)-trans-3-Methyl-2,3,4,4aalpha,5,6,7,7aalpha-oct...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I]OXY from human delta opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50303851((+)-cis-3-Methyl-2,3,4,4aalpha,5,6,7,7aalpha-octah...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I]OXY from human mu opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50303851((+)-cis-3-Methyl-2,3,4,4aalpha,5,6,7,7aalpha-octah...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I]OXY from human delta opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Rat)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50303848((-)-trans-3-Methyl-2,3,4,4aalpha,5,6,7,7aalpha-oct...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H](+)-pentazocine from sigma1 receptor in rat brain homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50303850((-)-trans-3-Cyclopropylmethyl-9-methoxy-2,3,4,4aal...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I]OXY from human kappa opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
Displayed 1 to 50 (of 62 total ) | Next | Last >>
Jump to: