Compile Data Set for Download or QSAR
Report error Found 30 Enz. Inhib. hit(s) with all data for entry = 50030909
TargetCannabinoid receptor 1(Human)
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50303835(3-(4-Chlorophenyl)-N'-((4-chlorophenyl)sulfonyl)-N...)
Affinity DataKi:  3.10nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50303837([3-(4-Chlorophenyl)-4-phenyl-4,5-dihydro-1H-pyrazo...)
Affinity DataKi:  9.60nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50303844(1-(4-Chlorophenyl)-2-(2-chlorophenyl)-5-ethyl-N-(p...)
Affinity DataKi:  14nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50303836(3-(4-Chlorophenyl)-N'-((4-chlorophenyl)sulfonyl)-N...)
Affinity DataKi:  19nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM21278(SR141716 | 5-(4-chlorophenyl)-1-(2,4-dichloropheny...)
Affinity DataKi:  25nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM29094(3-(4-chlorophenyl)-N''''-(4-chlorophenylsulfonyl)-...)
Affinity DataKi:  25nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50303838(3-(4-Chlorophenyl)-N'-((4-chlorophenyl)sulfonyl)-N...)
Affinity DataKi:  27nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50303846([3-(4-Chlorophenyl)-4-phenyl-4,5-dihydro-1H-pyrazo...)
Affinity DataKi:  31nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50303839(4-Chloro-N-{[3-(4-chlorophenyl)-4-phenyl-4,5-dihyd...)
Affinity DataKi:  42nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50303845(3-(4-Chlorophenyl)-N'-((4-chlorophenyl)sulfonyl)-N...)
Affinity DataKi:  43nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50303841(N-[4-(1,2,3,4-Tetrahydroacridin-9-ylamino)butyl]-2...)
Affinity DataKi:  48nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50303840(4-Chloro-N-{[3-(4-chlorophenyl)-4-phenyl-4,5-dihyd...)
Affinity DataKi:  54nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50303842(N-[7-(1,2,3,4-Tetrahydroacridin-9-ylamino)heptyl]-...)
Affinity DataKi:  88nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50303846([3-(4-Chlorophenyl)-4-phenyl-4,5-dihydro-1H-pyrazo...)
Affinity DataKi:  571nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50303843(5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl...)
Affinity DataKi:  701nMAssay Description:Binding affinity to CB1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM8961(CHEMBL95 | Cognex | cid_1935 | CHEMBL1337960 | 1,2...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]CP-55940 from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM8961(CHEMBL95 | Cognex | cid_1935 | CHEMBL1337960 | 1,2...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM29094(3-(4-chlorophenyl)-N''''-(4-chlorophenylsulfonyl)-...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50303844(1-(4-Chlorophenyl)-2-(2-chlorophenyl)-5-ethyl-N-(p...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50303835(3-(4-Chlorophenyl)-N'-((4-chlorophenyl)sulfonyl)-N...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50303845(3-(4-Chlorophenyl)-N'-((4-chlorophenyl)sulfonyl)-N...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50303842(N-[7-(1,2,3,4-Tetrahydroacridin-9-ylamino)heptyl]-...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50303841(N-[4-(1,2,3,4-Tetrahydroacridin-9-ylamino)butyl]-2...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50303840(4-Chloro-N-{[3-(4-chlorophenyl)-4-phenyl-4,5-dihyd...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50303839(4-Chloro-N-{[3-(4-chlorophenyl)-4-phenyl-4,5-dihyd...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50303838(3-(4-Chlorophenyl)-N'-((4-chlorophenyl)sulfonyl)-N...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50303837([3-(4-Chlorophenyl)-4-phenyl-4,5-dihydro-1H-pyrazo...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50303836(3-(4-Chlorophenyl)-N'-((4-chlorophenyl)sulfonyl)-N...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM21278(SR141716 | 5-(4-chlorophenyl)-1-(2,4-dichloropheny...)
Affinity DataKi:  1.58E+3nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50303843(5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl...)
Affinity DataKi:  6.54E+3nMAssay Description:Binding affinity to mu opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed