Compile Data Set for Download or QSAR
Report error Found 15 Enz. Inhib. hit(s) with all data for entry = 50031220
TargetSodium-dependent serotonin transporter(Rat)
Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50309172((1R,2S)-2-(4-benzylpiperazin-1-yl)-1-(5-chloro-6-m...)
Affinity DataIC50: 12nMAssay Description:Inhibition of [3H]5HT reuptake at rat brain frontal cortex serotonin transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetTransporter(Rat)
Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50309172((1R,2S)-2-(4-benzylpiperazin-1-yl)-1-(5-chloro-6-m...)
Affinity DataIC50: 185nMAssay Description:Inhibition of [3H]norepinephrine reuptake at rat brain frontal cortex norepinephrine transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM82071(NSC_62923 | WY-45030 | VENLAFAXINE | CAS_93413-69-...)
Affinity DataIC50: 350nMAssay Description:Inhibition of [3H]5HT reuptake at rat brain frontal cortex serotonin transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50309175((1R,2R)-2-(4-benzylpiperazin-1-yl)-1-(5-chloro-6-m...)
Affinity DataIC50: 375nMAssay Description:Inhibition of [3H]5HT reuptake at rat brain frontal cortex serotonin transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetTransporter(Rat)
Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50309173(rac-erythro-2-(4-benzylpiperazin-1-yl)-1-(5-chloro...)
Affinity DataIC50: 425nMAssay Description:Inhibition of [3H]norepinephrine reuptake at rat brain frontal cortex norepinephrine transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50309174((1S,2R)-2-(4-benzylpiperazin-1-yl)-1-(5-chloro-6-m...)
Affinity DataIC50: 548nMAssay Description:Inhibition of [3H]5HT reuptake at rat brain frontal cortex serotonin transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50309173(rac-erythro-2-(4-benzylpiperazin-1-yl)-1-(5-chloro...)
Affinity DataIC50: 825nMAssay Description:Inhibition of [3H]5HT reuptake at rat brain frontal cortex serotonin transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50309172((1R,2S)-2-(4-benzylpiperazin-1-yl)-1-(5-chloro-6-m...)
Affinity DataIC50: 1.15E+3nMAssay Description:Inhibition of [3H]dopamine reuptake at rat brain frontal cortex dopamine transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetTransporter(Rat)
Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50309175((1R,2R)-2-(4-benzylpiperazin-1-yl)-1-(5-chloro-6-m...)
Affinity DataIC50: 1.25E+3nMAssay Description:Inhibition of [3H]norepinephrine reuptake at rat brain frontal cortex norepinephrine transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetTransporter(Rat)
Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM82071(NSC_62923 | WY-45030 | VENLAFAXINE | CAS_93413-69-...)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of [3H]norepinephrine reuptake at rat brain frontal cortex norepinephrine transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetTransporter(Rat)
Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50309174((1S,2R)-2-(4-benzylpiperazin-1-yl)-1-(5-chloro-6-m...)
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibition of [3H]norepinephrine reuptake at rat brain frontal cortex norepinephrine transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50309174((1S,2R)-2-(4-benzylpiperazin-1-yl)-1-(5-chloro-6-m...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of [3H]dopamine reuptake at rat brain frontal cortex dopamine transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50309173(rac-erythro-2-(4-benzylpiperazin-1-yl)-1-(5-chloro...)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of [3H]dopamine reuptake at rat brain frontal cortex dopamine transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM50309175((1R,2R)-2-(4-benzylpiperazin-1-yl)-1-(5-chloro-6-m...)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of [3H]dopamine reuptake at rat brain frontal cortex dopamine transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Institute of Pharmaceutical Industry

Curated by ChEMBL
LigandPNGBDBM82071(NSC_62923 | WY-45030 | VENLAFAXINE | CAS_93413-69-...)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of [3H]dopamine reuptake at rat brain frontal cortex dopamine transporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed