Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) with all data for entry = 50031218
Target2-5A-dependent ribonuclease(Human)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50152834([(2R,3R,4R,5R)-5-(6-amino-9H-purin-9-yl)-4-[({[(2R...)
Affinity DataEC50:  9.70nMAssay Description:Inhibition of human RNaseL ANK domain expressed in Escherichia coli assessed as 5' flurescein-r(C11U2C7)-3' RNA cleavageMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
Target2-5A-dependent ribonuclease(Human)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50309127({[(2R,3R,4R,5R)-4-[({[(2R,3R,4R,5R)-5-(6-amino-8-m...)
Affinity DataEC50: >50nMAssay Description:Inhibition of human RNaseL ANK domain expressed in Escherichia coli assessed as 5' flurescein-r(C11U2C7)-3' RNA cleavageMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
Target2-5A-dependent ribonuclease(Human)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50309128({[(2R,3R,4R,5R)-4-[({[(2R,3S,4R,5R)-5-(6-amino-8-m...)
Affinity DataEC50: >50nMAssay Description:Inhibition of human RNaseL ANK domain expressed in Escherichia coli assessed as 5' flurescein-r(C11U2C7)-3' RNA cleavageMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
Target2-5A-dependent ribonuclease(Human)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50309129({[(2R,3R,4R,5R)-4-[({[(2R,3R,4R,5R)-4-[({[(2R,3S,4...)
Affinity DataEC50:  2.5nMAssay Description:Inhibition of human RNaseL ANK domain expressed in Escherichia coli assessed as 5' flurescein-r(C11U2C7)-3' RNA cleavageMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
Target2-5A-dependent ribonuclease(Human)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50309130({[(2R,3R,4R,5R)-4-[({[(2R,3R,4R,5R)-4-[({[(2R,3R,4...)
Affinity DataEC50:  2.5nMAssay Description:Inhibition of human RNaseL ANK domain expressed in Escherichia coli assessed as 5' flurescein-r(C11U2C7)-3' RNA cleavageMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed