Compile Data Set for Download or QSAR
Report error Found 60 Enz. Inhib. hit(s) with all data for entry = 50031216
TargetRho-associated protein kinase 2(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50309123(4-(6-(piperazin-1-yl)-5-(pyrrolidin-1-yl)pyrazin-2...)
Affinity DataIC50: 17nMAssay Description:Inhibition of human recombinant ROCK2More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetRho-associated protein kinase 2(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50309122(4-(6-(1,4-diazepan-1-yl)-5-(pyrrolidin-1-yl)pyrazi...)
Affinity DataIC50: 21nMAssay Description:Inhibition of human recombinant ROCK2More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetRho-associated protein kinase 2(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50309120((1-(6-(pyridin-4-yl)-3-(pyrrolidin-1-yl)pyrazin-2-...)
Affinity DataIC50: 28nMAssay Description:Inhibition of human recombinant ROCK2More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetRho-associated protein kinase 1(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50309123(4-(6-(piperazin-1-yl)-5-(pyrrolidin-1-yl)pyrazin-2...)
Affinity DataIC50: 34nMAssay Description:Inhibition of human recombinant ROCK1More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetRho-associated protein kinase 2(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50309116(1-(6-(pyridin-4-yl)-3-(pyrrolidin-1-yl)pyrazin-2-y...)
Affinity DataIC50: 39nMAssay Description:Inhibition of human recombinant ROCK2More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetRho-associated protein kinase 2(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50309121(N-methyl-1-(1-(6-(pyridin-4-yl)-3-(pyrrolidin-1-yl...)
Affinity DataIC50: 49nMAssay Description:Inhibition of human recombinant ROCK2More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetRho-associated protein kinase 2(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50309118(1-(6-(pyridin-4-yl)-3-(pyrrolidin-1-yl)pyrazin-2-y...)
Affinity DataIC50: 62nMAssay Description:Inhibition of human recombinant ROCK2More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetRho-associated protein kinase 2(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50309117(3-(piperazin-1-yl)-5-(pyridin-4-yl)-2-(pyrrolidin-...)
Affinity DataIC50: 62nMAssay Description:Inhibition of human recombinant ROCK2More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetRho-associated protein kinase 2(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50309126(2-(4-(6-(pyridin-4-yl)-3-(pyrrolidin-1-yl)pyrazin-...)
Affinity DataIC50: 78nMAssay Description:Inhibition of human recombinant ROCK2More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetRho-associated protein kinase 2(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50309124(1-(3-(pyrrolidin-1-yl)-6-(1H-pyrrolo[2,3-b]pyridin...)
Affinity DataIC50: 89nMAssay Description:Inhibition of human recombinant ROCK2More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetRho-associated protein kinase 1(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50309120((1-(6-(pyridin-4-yl)-3-(pyrrolidin-1-yl)pyrazin-2-...)
Affinity DataIC50: 130nMAssay Description:Inhibition of human recombinant ROCK1More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetRho-associated protein kinase 1(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50309121(N-methyl-1-(1-(6-(pyridin-4-yl)-3-(pyrrolidin-1-yl...)
Affinity DataIC50: 150nMAssay Description:Inhibition of human recombinant ROCK1More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetRho-associated protein kinase 1(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50309122(4-(6-(1,4-diazepan-1-yl)-5-(pyrrolidin-1-yl)pyrazi...)
Affinity DataIC50: 170nMAssay Description:Inhibition of human recombinant ROCK1More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetRho-associated protein kinase 2(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50309119(N-methyl-1-(6-(pyridin-4-yl)-3-(pyrrolidin-1-yl)py...)
Affinity DataIC50: 250nMAssay Description:Inhibition of human recombinant ROCK2More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetRho-associated protein kinase 1(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50309118(1-(6-(pyridin-4-yl)-3-(pyrrolidin-1-yl)pyrazin-2-y...)
Affinity DataIC50: 290nMAssay Description:Inhibition of human recombinant ROCK1More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetRho-associated protein kinase 1(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50309126(2-(4-(6-(pyridin-4-yl)-3-(pyrrolidin-1-yl)pyrazin-...)
Affinity DataIC50: 300nMAssay Description:Inhibition of human recombinant ROCK1More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetRho-associated protein kinase 2(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50309125(2-(4-(3-(dimethylamino)-6-(pyridin-4-yl)pyrazin-2-...)
Affinity DataIC50: 300nMAssay Description:Inhibition of human recombinant ROCK2More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetRho-associated protein kinase 1(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50309124(1-(3-(pyrrolidin-1-yl)-6-(1H-pyrrolo[2,3-b]pyridin...)
Affinity DataIC50: 300nMAssay Description:Inhibition of human recombinant ROCK1More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetRho-associated protein kinase 1(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50309116(1-(6-(pyridin-4-yl)-3-(pyrrolidin-1-yl)pyrazin-2-y...)
Affinity DataIC50: 320nMAssay Description:Inhibition of human recombinant ROCK1More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetRho-associated protein kinase 2(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50309113(1-methyl-4-(6-(pyridin-4-yl)-3-(pyrrolidin-1-yl)py...)
Affinity DataIC50: 330nMAssay Description:Inhibition of human recombinant ROCK2More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetRho-associated protein kinase 2(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50309103(3-(4-methyl-1,4-diazepan-1-yl)-5-(1H-pyrrolo[2,3-b...)
Affinity DataIC50: 530nMAssay Description:Inhibition of human recombinant ROCK2More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetRho-associated protein kinase 2(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50309114(1-methyl-4-(3-(piperidin-1-yl)-6-(pyridin-4-yl)pyr...)
Affinity DataIC50: 560nMAssay Description:Inhibition of human recombinant ROCK2More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetRho-associated protein kinase 1(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50309117(3-(piperazin-1-yl)-5-(pyridin-4-yl)-2-(pyrrolidin-...)
Affinity DataIC50: 610nMAssay Description:Inhibition of human recombinant ROCK1More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetRho-associated protein kinase 2(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50309105(5-(1H-indazol-5-yl)-3-(4-methyl-1,4-diazepan-1-yl)...)
Affinity DataIC50: 950nMAssay Description:Inhibition of human recombinant ROCK2More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetRho-associated protein kinase 1(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50309125(2-(4-(3-(dimethylamino)-6-(pyridin-4-yl)pyrazin-2-...)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of human recombinant ROCK1More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetRho-associated protein kinase 1(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50309103(3-(4-methyl-1,4-diazepan-1-yl)-5-(1H-pyrrolo[2,3-b...)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of human recombinant ROCK1More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetRho-associated protein kinase 2(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50309108(N,N-dimethyl-3-(4-methyl-1,4-diazepan-1-yl)-5-(pyr...)
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of human recombinant ROCK2More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetRho-associated protein kinase 1(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50309119(N-methyl-1-(6-(pyridin-4-yl)-3-(pyrrolidin-1-yl)py...)
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of human recombinant ROCK1More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetRho-associated protein kinase 1(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50309105(5-(1H-indazol-5-yl)-3-(4-methyl-1,4-diazepan-1-yl)...)
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of human recombinant ROCK1More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetRho-associated protein kinase 2(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50309107(N-methyl-3-(4-methyl-1,4-diazepan-1-yl)-5-(pyridin...)
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of human recombinant ROCK2More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetRho-associated protein kinase 2(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50309098(3-(4-methyl-1,4-diazepan-1-yl)-5-(pyridin-4-yl)pyr...)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of human recombinant ROCK2More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetRho-associated protein kinase 2(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50309104(5-(1H-indazol-4-yl)-3-(4-methyl-1,4-diazepan-1-yl)...)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of human recombinant ROCK2More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetRho-associated protein kinase 2(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50309097(2-(4-(3-amino-6-(pyridin-4-yl)pyrazin-2-yl)piperaz...)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of human recombinant ROCK2More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetRho-associated protein kinase 1(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50309109(N,N-diethyl-3-(4-methyl-1,4-diazepan-1-yl)-5-(pyri...)
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of human recombinant ROCK1More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetRho-associated protein kinase 2(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50309102(3-(4-methyl-1,4-diazepan-1-yl)-5-(1H-pyrazol-3-yl)...)
Affinity DataIC50: 2.90E+3nMAssay Description:Inhibition of human recombinant ROCK2More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetRho-associated protein kinase 2(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50309110(2-(3-(4-methyl-1,4-diazepan-1-yl)-5-(pyridin-4-yl)...)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of human recombinant ROCK2More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetRho-associated protein kinase 1(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50309097(2-(4-(3-amino-6-(pyridin-4-yl)pyrazin-2-yl)piperaz...)
Affinity DataIC50: 4.60E+3nMAssay Description:Inhibition of human recombinant ROCK1More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetRho-associated protein kinase 1(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50309098(3-(4-methyl-1,4-diazepan-1-yl)-5-(pyridin-4-yl)pyr...)
Affinity DataIC50: 4.60E+3nMAssay Description:Inhibition of human recombinant ROCK1More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetRho-associated protein kinase 1(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50309113(1-methyl-4-(6-(pyridin-4-yl)-3-(pyrrolidin-1-yl)py...)
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of human recombinant ROCK1More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetRho-associated protein kinase 2(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50309115(4-(3-(4-methyl-1,4-diazepan-1-yl)-5-(pyridin-4-yl)...)
Affinity DataIC50: 6.30E+3nMAssay Description:Inhibition of human recombinant ROCK2More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetRho-associated protein kinase 1(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50309108(N,N-dimethyl-3-(4-methyl-1,4-diazepan-1-yl)-5-(pyr...)
Affinity DataIC50: 6.50E+3nMAssay Description:Inhibition of human recombinant ROCK1More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetRho-associated protein kinase 2(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50309109(N,N-diethyl-3-(4-methyl-1,4-diazepan-1-yl)-5-(pyri...)
Affinity DataIC50: 6.70E+3nMAssay Description:Inhibition of human recombinant ROCK2More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetRho-associated protein kinase 1(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50309107(N-methyl-3-(4-methyl-1,4-diazepan-1-yl)-5-(pyridin...)
Affinity DataIC50: 6.90E+3nMAssay Description:Inhibition of human recombinant ROCK1More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetRho-associated protein kinase 1(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50309104(5-(1H-indazol-4-yl)-3-(4-methyl-1,4-diazepan-1-yl)...)
Affinity DataIC50: 9.60E+3nMAssay Description:Inhibition of human recombinant ROCK1More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetRho-associated protein kinase 1(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50309111(N-(2-methoxyethyl)-3-(4-methyl-1,4-diazepan-1-yl)-...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant ROCK1More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetRho-associated protein kinase 2(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50309106(5-(1H-indazol-6-yl)-3-(4-methyl-1,4-diazepan-1-yl)...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant ROCK2More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetRho-associated protein kinase 1(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50309106(5-(1H-indazol-6-yl)-3-(4-methyl-1,4-diazepan-1-yl)...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant ROCK1More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetRho-associated protein kinase 1(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50309114(1-methyl-4-(3-(piperidin-1-yl)-6-(pyridin-4-yl)pyr...)
Affinity DataIC50: 1.80E+4nMAssay Description:Inhibition of human recombinant ROCK1More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetRho-associated protein kinase 1(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50309101(5-(2-aminopyridin-4-yl)-3-(4-methyl-1,4-diazepan-1...)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of human recombinant ROCK1More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetRho-associated protein kinase 1(Human)
Amri

Curated by ChEMBL
LigandPNGBDBM50309102(3-(4-methyl-1,4-diazepan-1-yl)-5-(1H-pyrazol-3-yl)...)
Affinity DataIC50: 3.70E+4nMAssay Description:Inhibition of human recombinant ROCK1More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
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