Compile Data Set for Download or QSAR
Report error Found 109 Enz. Inhib. hit(s) with all data for entry = 50038951
TargetGlycogen synthase kinase-3 beta(Human)
Technische Universit£T Braunschweig

Curated by ChEMBL
LigandPNGBDBM7262(NSC 705701 | BDBM84528 | alsterpaullone | 9-Nitrop...)
Affinity DataIC50: 4nMAssay Description:Inhibition of GSK3-beta expressed in insect Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Technische Universit£T Braunschweig

Curated by ChEMBL
LigandPNGBDBM7263(CHEMBL299756 | 9-oxo-8,18-diazatetracyclo[9.7.0.0^...)
Affinity DataIC50: 10nMAssay Description:Inhibition of GSK3-beta expressed in insect Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Technische Universit£T Braunschweig

Curated by ChEMBL
LigandPNGBDBM50300062(9-Bromo-2-methoxy-5,12-dihydro-7H-benzo[2,3]azepin...)
Affinity DataIC50: 15nMAssay Description:Inhibition of GSK3-betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Technische Universit£T Braunschweig

Curated by ChEMBL
LigandPNGBDBM7265(NSC 708244 | 4,5-dimethoxy-9-oxo-8,18-diazatetracy...)
Affinity DataIC50: 18nMAssay Description:Inhibition of GSK3-beta expressed in insect Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Technische Universit£T Braunschweig

Curated by ChEMBL
LigandPNGBDBM7322(14-bromo-5-hydroxy-8,18-diazatetracyclo[9.7.0.0^{2...)
Affinity DataIC50: 18nMAssay Description:Inhibition of GSK3-betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Technische Universit£T Braunschweig

Curated by ChEMBL
LigandPNGBDBM7266(cid_3820 | NSC 664704 | 9-bromopaullone | 14-bromo...)
Affinity DataIC50: 23nMAssay Description:Inhibition of GSK3-beta expressed in insect Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
LigandPNGBDBM7263(CHEMBL299756 | 9-oxo-8,18-diazatetracyclo[9.7.0.0^...)
Affinity DataIC50: 24nMAssay Description:Inhibition of CDK1/cyclin B expressed in M phase starfish oocyteMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Technische Universit£T Braunschweig

Curated by ChEMBL
LigandPNGBDBM7267(CHEMBL98153 | 14-chloro-8,18-diazatetracyclo[9.7.0...)
Affinity DataIC50: 24nMAssay Description:Inhibition of GSK3-beta expressed in insect Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Technische Universit£T Braunschweig

Curated by ChEMBL
LigandPNGBDBM7268(NSC 701590 | 9-trifluoromethylpaullone | 14-(trifl...)
Affinity DataIC50: 30nMAssay Description:Inhibition of GSK3-beta expressed in insect Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
LigandPNGBDBM7262(NSC 705701 | BDBM84528 | alsterpaullone | 9-Nitrop...)
Affinity DataIC50: 35nMAssay Description:Inhibition of CDK1/cyclin B expressed in M phase starfish oocyteMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
LigandPNGBDBM7265(NSC 708244 | 4,5-dimethoxy-9-oxo-8,18-diazatetracy...)
Affinity DataIC50: 44nMAssay Description:Inhibition of CDK1/cyclin B expressed in M phase starfish oocyteMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Technische Universit£T Braunschweig

Curated by ChEMBL
LigandPNGBDBM7270(4,5-dimethoxy-14-(trifluoromethyl)-8,18-diazatetra...)
Affinity DataIC50: 75nMAssay Description:Inhibition of GSK3-betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Technische Universit£T Braunschweig

Curated by ChEMBL
LigandPNGBDBM7272(14-fluoro-8,18-diazatetracyclo[9.7.0.0^{2,7}.0^{12...)
Affinity DataIC50: 80nMAssay Description:Inhibition of GSK3-beta expressed in insect Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Technische Universit£T Braunschweig

Curated by ChEMBL
LigandPNGBDBM7273(CHEMBL319373 | 14-bromo-4,5-dimethoxy-8,18-diazate...)
Affinity DataIC50: 100nMAssay Description:Inhibition of GSK3-beta expressed in insect Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Technische Universit£T Braunschweig

Curated by ChEMBL
LigandPNGBDBM7275(NSC 675995 | CHEMBL317964 | 9-methylpaullone | 14-...)
Affinity DataIC50: 130nMAssay Description:Inhibition of GSK3-beta expressed in insect Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
LigandPNGBDBM7273(CHEMBL319373 | 14-bromo-4,5-dimethoxy-8,18-diazate...)
Affinity DataIC50: 200nMAssay Description:Inhibition of CDK1/cyclin B expressed in M phase starfish oocyteMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Technische Universit£T Braunschweig

Curated by ChEMBL
LigandPNGBDBM7278(11-chloropaullone | CHEMBL318471 | 16-chloro-8,18-...)
Affinity DataIC50: 200nMAssay Description:Inhibition of GSK3-beta expressed in insect Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Technische Universit£T Braunschweig

Curated by ChEMBL
LigandPNGBDBM7320(5-methoxy-14-(trifluoromethyl)-8,18-diazatetracycl...)
Affinity DataIC50: 240nMAssay Description:Inhibition of GSK3-betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
LigandPNGBDBM7270(4,5-dimethoxy-14-(trifluoromethyl)-8,18-diazatetra...)
Affinity DataIC50: 280nMAssay Description:Inhibition of CDK1/cyclin BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
LigandPNGBDBM50300063(9-(Methylsulfinyl)-7,12-dihydroindolo[3,2-d][1]ben...)
Affinity DataIC50: 280nMAssay Description:Inhibition of CDK1/cyclin BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
LigandPNGBDBM7268(NSC 701590 | 9-trifluoromethylpaullone | 14-(trifl...)
Affinity DataIC50: 400nMAssay Description:Inhibition of CDK1/cyclin B expressed in M phase starfish oocyteMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
LigandPNGBDBM7266(cid_3820 | NSC 664704 | 9-bromopaullone | 14-bromo...)
Affinity DataIC50: 400nMAssay Description:Inhibition of CDK1/cyclin B expressed in M phase starfish oocyteMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Technische Universit£T Braunschweig

Curated by ChEMBL
LigandPNGBDBM7283(NSC 704071 | CHEMBL318208 | 14-bromo-18-methyl-8,1...)
Affinity DataIC50: 400nMAssay Description:Inhibition of GSK3-beta expressed in insect Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
LigandPNGBDBM50300062(9-Bromo-2-methoxy-5,12-dihydro-7H-benzo[2,3]azepin...)
Affinity DataIC50: 400nMAssay Description:Inhibition of CDK1/cyclin BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
LigandPNGBDBM50300064(9-(methylthio)-7,12-dihydroindolo[3,2-d][1]benzaze...)
Affinity DataIC50: 400nMAssay Description:Inhibition of CDK1/cyclin BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
LigandPNGBDBM7267(CHEMBL98153 | 14-chloro-8,18-diazatetracyclo[9.7.0...)
Affinity DataIC50: 600nMAssay Description:Inhibition of CDK1/cyclin B expressed in M phase starfish oocyteMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
LigandPNGBDBM7322(14-bromo-5-hydroxy-8,18-diazatetracyclo[9.7.0.0^{2...)
Affinity DataIC50: 600nMAssay Description:Inhibition of CDK1/cyclin BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Technische Universit£T Braunschweig

Curated by ChEMBL
LigandPNGBDBM7287(8,18-diazatetracyclo[9.7.0.0^{2,7}.0^{12,17}]octad...)
Affinity DataIC50: 620nMAssay Description:Inhibition of GSK3-beta expressed in insect Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
LigandPNGBDBM7320(5-methoxy-14-(trifluoromethyl)-8,18-diazatetracycl...)
Affinity DataIC50: 700nMAssay Description:Inhibition of CDK1/cyclin BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
TargetMalate dehydrogenase, mitochondrial(Human)
Technische Universit£T Braunschweig

Curated by ChEMBL
LigandPNGBDBM50300050(9-tert-Butyl-5-(3,4-dichlorobenzyl)-7,12-dihydroin...)
Affinity DataIC50: 770nMAssay Description:Inhibition of mitochondrial malate dehydrogenase by spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
TargetMalate dehydrogenase, mitochondrial(Human)
Technische Universit£T Braunschweig

Curated by ChEMBL
LigandPNGBDBM50300053(9-Bromo-5-(3,4-dichlorobenzyl)-7,12-dihydroindolo[...)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of mitochondrial malate dehydrogenase by spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Technische Universit£T Braunschweig

Curated by ChEMBL
LigandPNGBDBM50300064(9-(methylthio)-7,12-dihydroindolo[3,2-d][1]benzaze...)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of GSK3-betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
LigandPNGBDBM7278(11-chloropaullone | CHEMBL318471 | 16-chloro-8,18-...)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of CDK1/cyclin B expressed in M phase starfish oocyteMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
LigandPNGBDBM7272(14-fluoro-8,18-diazatetracyclo[9.7.0.0^{2,7}.0^{12...)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of CDK1/cyclin B expressed in M phase starfish oocyteMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
TargetMalate dehydrogenase, mitochondrial(Human)
Technische Universit£T Braunschweig

Curated by ChEMBL
LigandPNGBDBM50300055(9-Bromo-5-(4-methylbenzyl)-7,12-dihydroindolo[3,2-...)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of mitochondrial malate dehydrogenase by spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
TargetMalate dehydrogenase, mitochondrial(Human)
Technische Universit£T Braunschweig

Curated by ChEMBL
LigandPNGBDBM50300059(5-Benzyl-9-tert-butyl-7,12-dihydroindolo[3,2-d][1]...)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of mitochondrial malate dehydrogenase by spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
TargetMalate dehydrogenase, mitochondrial(Human)
Technische Universit£T Braunschweig

Curated by ChEMBL
LigandPNGBDBM50300054(9-Bromo-5-(4-methoxybenzyl)-7,12-dihydroindolo[3,2...)
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of mitochondrial malate dehydrogenase by spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
LigandPNGBDBM7275(NSC 675995 | CHEMBL317964 | 9-methylpaullone | 14-...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of CDK1/cyclin B expressed in M phase starfish oocyteMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Technische Universit£T Braunschweig

Curated by ChEMBL
LigandPNGBDBM7300(NSC 702376 | 9-bromo-5-methylpaullone | 14-bromo-8...)
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of GSK3-beta expressed in insect Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
TargetMalate dehydrogenase, mitochondrial(Human)
Technische Universit£T Braunschweig

Curated by ChEMBL
LigandPNGBDBM7307(CHEMBL99779 | NSC 702377 | 8-benzyl-14-bromo-8,18-...)
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of mitochondrial malate dehydrogenase by spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
LigandPNGBDBM7306(8,10-dichloropaullone | CHEMBL316512 | NSC 703056 ...)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of CDK1/cyclin B expressed in M phase starfish oocyteMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
TargetMalate dehydrogenase, mitochondrial(Human)
Technische Universit£T Braunschweig

Curated by ChEMBL
LigandPNGBDBM50300044(Octyl 6-oxo-5,6,7,12-tetrahydroindolo[3,2-d][1]ben...)
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of mitochondrial malate dehydrogenase by spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
TargetMalate dehydrogenase, mitochondrial(Human)
Technische Universit£T Braunschweig

Curated by ChEMBL
LigandPNGBDBM50300060(5-Benzyl-9-chloro-7,12-dihydroindolo[3,2-d][1]benz...)
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of mitochondrial malate dehydrogenase by spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Technische Universit£T Braunschweig

Curated by ChEMBL
LigandPNGBDBM7304(9-bromo-12-(2-propenyl)-paullone | NSC 704072 | CH...)
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of GSK3-beta expressed in insect Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
TargetMalate dehydrogenase, mitochondrial(Human)
Technische Universit£T Braunschweig

Curated by ChEMBL
LigandPNGBDBM50300058(5-Benzyl-9-trifluoromethyl-7,12-dihydroindolo[3,2-...)
Affinity DataIC50: 4.20E+3nMAssay Description:Inhibition of mitochondrial malate dehydrogenase by spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
LigandPNGBDBM50300061(Methyl 6-oxo-5,6,7,12-tetrahydroindolo[3,2-d][1]be...)
Affinity DataIC50: 4.20E+3nMAssay Description:Inhibition of CDK1/cyclin BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Technische Universit£T Braunschweig

Curated by ChEMBL
LigandPNGBDBM7305(NSC 699471 | 9-bromo-4-hydroxypaullone | CHEMBL954...)
Affinity DataIC50: 4.30E+3nMAssay Description:Inhibition of GSK3-beta expressed in insect Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
TargetMalate dehydrogenase, mitochondrial(Human)
Technische Universit£T Braunschweig

Curated by ChEMBL
LigandPNGBDBM50300045(Hexyl 6-oxo-5,6,7,12-tetrahydroindolo[3,2-d][1]ben...)
Affinity DataIC50: 4.30E+3nMAssay Description:Inhibition of mitochondrial malate dehydrogenase by spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
TargetMalate dehydrogenase, mitochondrial(Human)
Technische Universit£T Braunschweig

Curated by ChEMBL
LigandPNGBDBM50300046(Pentyl 6-oxo-5,6,7,12-tetrahydroindolo[3,2-d][1]be...)
Affinity DataIC50: 4.40E+3nMAssay Description:Inhibition of mitochondrial malate dehydrogenase by spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Technische Universit£T Braunschweig

Curated by ChEMBL
LigandPNGBDBM7306(8,10-dichloropaullone | CHEMBL316512 | NSC 703056 ...)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of GSK3-beta expressed in insect Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
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