Compile Data Set for Download or QSAR
Report error Found 12 Enz. Inhib. hit(s) with all data for entry = 50030982
TargetThyroid hormone receptor beta(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50304781(PF-00277343 | 2-(4-(3-(4-fluorobenzyl)-4-hydroxyph...)
Affinity DataKi:  0.400nMAssay Description:Binding affinity to thyroid receptor betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetThyroid hormone receptor beta(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50304777(2-(4-(7-hydroxy-2,3-dihydro-1H-inden-4-yloxy)-3,5-...)
Affinity DataKi:  0.5nMAssay Description:Binding affinity to thyroid receptor betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetThyroid hormone receptor beta(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50304778(3-(3-chloro-4-(3-(cyclobutylmethylsulfonyl)-4-hydr...)
Affinity DataKi:  0.5nMAssay Description:Binding affinity to thyroid receptor betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetThyroid hormone receptor beta(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50304780(2-(3,5-dichloro-4-(3-(4-fluorobenzyl)-4-hydroxyphe...)
Affinity DataKi:  0.510nMAssay Description:Binding affinity to thyroid receptor betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetThyroid hormone receptor alpha(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50304777(2-(4-(7-hydroxy-2,3-dihydro-1H-inden-4-yloxy)-3,5-...)
Affinity DataKi:  0.700nMAssay Description:Binding affinity to thyroid receptor alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetThyroid hormone receptor beta(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50123049(2-{3,5-Dichloro-4-[4-hydroxy-3-(piperidine-1-carbo...)
Affinity DataKi:  1nMAssay Description:Binding affinity to thyroid receptor betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetThyroid hormone receptor beta(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50304779(2-(3,5-dichloro-4-(4-hydroxy-3-(1,2,3,4-tetrahydro...)
Affinity DataKi:  2nMAssay Description:Binding affinity to thyroid receptor betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetThyroid hormone receptor alpha(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50304778(3-(3-chloro-4-(3-(cyclobutylmethylsulfonyl)-4-hydr...)
Affinity DataKi:  2.10nMAssay Description:Binding affinity to thyroid receptor alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetThyroid hormone receptor alpha(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50304781(PF-00277343 | 2-(4-(3-(4-fluorobenzyl)-4-hydroxyph...)
Affinity DataKi:  3nMAssay Description:Binding affinity to thyroid receptor alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetThyroid hormone receptor alpha(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50304780(2-(3,5-dichloro-4-(3-(4-fluorobenzyl)-4-hydroxyphe...)
Affinity DataKi:  8nMAssay Description:Binding affinity to thyroid receptor alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetThyroid hormone receptor alpha(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50123049(2-{3,5-Dichloro-4-[4-hydroxy-3-(piperidine-1-carbo...)
Affinity DataKi:  20nMAssay Description:Binding affinity to thyroid receptor alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetThyroid hormone receptor alpha(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50304779(2-(3,5-dichloro-4-(4-hydroxy-3-(1,2,3,4-tetrahydro...)
Affinity DataKi:  126nMAssay Description:Binding affinity to thyroid receptor alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed