Compile Data Set for Download or QSAR
Report error Found 52 Enz. Inhib. hit(s) with all data for entry = 50030978
TargetSerine/threonine-protein kinase mTOR(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50304675(1-(4-(4-(8-oxa-3-azabicyclo[3.2.1]octan-3-yl)thien...)
Affinity DataIC50: 0.290nMAssay Description:Inhibition of mTORMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50304672(1-(4-(4-(8-oxa-3-azabicyclo[3.2.1]octan-3-yl)thien...)
Affinity DataIC50: 0.340nMAssay Description:Inhibition of mTORMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50304676(1-(4-(4-(8-oxa-3-azabicyclo[3.2.1]octan-3-yl)thien...)
Affinity DataIC50: 0.440nMAssay Description:Inhibition of mTORMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50304667(1-(4-(4-(8-oxa-3-azabicyclo[3.2.1]octan-3-yl)-6-((...)
Affinity DataIC50: 0.450nMAssay Description:Inhibition of mTORMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50304665(1-(4-(4-(8-oxa-3-azabicyclo[3.2.1]octan-3-yl)-6-((...)
Affinity DataIC50: 0.600nMAssay Description:Inhibition of mTORMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50304673(1-(4-(4-(8-oxa-3-azabicyclo[3.2.1]octan-3-yl)thien...)
Affinity DataIC50: 0.680nMAssay Description:Inhibition of mTORMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50304670(1-(4-(4-(8-oxa-3-azabicyclo[3.2.1]octan-3-yl)thien...)
Affinity DataIC50: 0.700nMAssay Description:Inhibition of mTORMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50304671(1-(4-(4-(8-oxa-3-azabicyclo[3.2.1]octan-3-yl)thien...)
Affinity DataIC50: 0.700nMAssay Description:Inhibition of mTORMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50304669(1-(4-(4-(8-oxa-3-azabicyclo[3.2.1]octan-3-yl)thien...)
Affinity DataIC50: 0.900nMAssay Description:Inhibition of mTORMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50304680(1-(4-(4-(8-oxa-3-azabicyclo[3.2.1]octan-3-yl)-6-((...)
Affinity DataIC50: 1nMAssay Description:Inhibition of mTORMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50304674(1-(4-(4-(8-oxa-3-azabicyclo[3.2.1]octan-3-yl)thien...)
Affinity DataIC50: 1.25nMAssay Description:Inhibition of mTORMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50304678(1-(4-(4-(8-oxa-3-azabicyclo[3.2.1]octan-3-yl)-6-((...)
Affinity DataIC50: 1.40nMAssay Description:Inhibition of mTORMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50304666(1-(4-(4-(8-oxa-3-azabicyclo[3.2.1]octan-3-yl)-6-((...)
Affinity DataIC50: 3.70nMAssay Description:Inhibition of mTORMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50304681(1-(4-(4-(8-oxa-3-azabicyclo[3.2.1]octan-3-yl)-6-((...)
Affinity DataIC50: 4.70nMAssay Description:Inhibition of mTORMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
LigandPNGBDBM50304667(1-(4-(4-(8-oxa-3-azabicyclo[3.2.1]octan-3-yl)-6-((...)
Affinity DataIC50: 8.30nMAssay Description:Inhibition of PI3KalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
LigandPNGBDBM50304689(5-(4-morpholinothieno[3,2-d]pyrimidin-2-yl)pyrimid...)
Affinity DataIC50: 8.5nMAssay Description:Inhibition of PI3KalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50304668(methyl 4-(4-(8-oxa-3-azabicyclo[3.2.1]octan-3-yl)t...)
Affinity DataIC50: 11nMAssay Description:Inhibition of mTORMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
LigandPNGBDBM50304665(1-(4-(4-(8-oxa-3-azabicyclo[3.2.1]octan-3-yl)-6-((...)
Affinity DataIC50: 12nMAssay Description:Inhibition of PI3KalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50304679(1-(4-(4-(8-oxa-3-azabicyclo[3.2.1]octan-3-yl)-6-((...)
Affinity DataIC50: 16nMAssay Description:Inhibition of mTORMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50304677(1-(4-(4-(8-oxa-3-azabicyclo[3.2.1]octan-3-yl)-6-((...)
Affinity DataIC50: 20nMAssay Description:Inhibition of mTORMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50304687(3-(2-(1H-indol-5-yl)thieno[3,2-d]pyrimidin-4-yl)-8...)
Affinity DataIC50: 22nMAssay Description:Inhibition of mTORMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50304688(N-(4-(4-(8-oxa-3-azabicyclo[3.2.1]octan-3-yl)thien...)
Affinity DataIC50: 26.5nMAssay Description:Inhibition of mTORMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50304684(4-(4-(8-oxa-3-azabicyclo[3.2.1]octan-3-yl)thieno[3...)
Affinity DataIC50: 32nMAssay Description:Inhibition of mTORMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50304685(5-(4-(8-oxa-3-azabicyclo[3.2.1]octan-3-yl)thieno[3...)
Affinity DataIC50: 35nMAssay Description:Inhibition of mTORMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
LigandPNGBDBM25018(thienopyrimidine derivative, 1 | CHEMBL541643 | 3-...)
Affinity DataIC50: 41nMAssay Description:Inhibition of PI3KalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
LigandPNGBDBM50304678(1-(4-(4-(8-oxa-3-azabicyclo[3.2.1]octan-3-yl)-6-((...)
Affinity DataIC50: 46nMAssay Description:Inhibition of PI3KalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM25018(thienopyrimidine derivative, 1 | CHEMBL541643 | 3-...)
Affinity DataIC50: 49nMAssay Description:Inhibition of mTORMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50304683(5-(4-(8-oxa-3-azabicyclo[3.2.1]octan-3-yl)thieno[3...)
Affinity DataIC50: 57nMAssay Description:Inhibition of mTORMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50304682(3-(4-(8-oxa-3-azabicyclo[3.2.1]octan-3-yl)thieno[3...)
Affinity DataIC50: 58nMAssay Description:Inhibition of mTORMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50304689(5-(4-morpholinothieno[3,2-d]pyrimidin-2-yl)pyrimid...)
Affinity DataIC50: 61nMAssay Description:Inhibition of mTORMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
LigandPNGBDBM50304676(1-(4-(4-(8-oxa-3-azabicyclo[3.2.1]octan-3-yl)thien...)
Affinity DataIC50: 80nMAssay Description:Inhibition of PI3KalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
LigandPNGBDBM50304674(1-(4-(4-(8-oxa-3-azabicyclo[3.2.1]octan-3-yl)thien...)
Affinity DataIC50: 82nMAssay Description:Inhibition of PI3KalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
LigandPNGBDBM50304666(1-(4-(4-(8-oxa-3-azabicyclo[3.2.1]octan-3-yl)-6-((...)
Affinity DataIC50: 86nMAssay Description:Inhibition of PI3KalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50304686(4-(4-(8-oxa-3-azabicyclo[3.2.1]octan-3-yl)thieno[3...)
Affinity DataIC50: 100nMAssay Description:Inhibition of mTORMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
LigandPNGBDBM50304675(1-(4-(4-(8-oxa-3-azabicyclo[3.2.1]octan-3-yl)thien...)
Affinity DataIC50: 119nMAssay Description:Inhibition of PI3KalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
LigandPNGBDBM50304681(1-(4-(4-(8-oxa-3-azabicyclo[3.2.1]octan-3-yl)-6-((...)
Affinity DataIC50: 148nMAssay Description:Inhibition of PI3KalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
LigandPNGBDBM50304680(1-(4-(4-(8-oxa-3-azabicyclo[3.2.1]octan-3-yl)-6-((...)
Affinity DataIC50: 179nMAssay Description:Inhibition of PI3KalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
LigandPNGBDBM50304683(5-(4-(8-oxa-3-azabicyclo[3.2.1]octan-3-yl)thieno[3...)
Affinity DataIC50: 246nMAssay Description:Inhibition of PI3KalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
LigandPNGBDBM50304677(1-(4-(4-(8-oxa-3-azabicyclo[3.2.1]octan-3-yl)-6-((...)
Affinity DataIC50: 322nMAssay Description:Inhibition of PI3KalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
LigandPNGBDBM50304672(1-(4-(4-(8-oxa-3-azabicyclo[3.2.1]octan-3-yl)thien...)
Affinity DataIC50: 324nMAssay Description:Inhibition of PI3KalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
LigandPNGBDBM50304682(3-(4-(8-oxa-3-azabicyclo[3.2.1]octan-3-yl)thieno[3...)
Affinity DataIC50: 399nMAssay Description:Inhibition of PI3KalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
LigandPNGBDBM50304669(1-(4-(4-(8-oxa-3-azabicyclo[3.2.1]octan-3-yl)thien...)
Affinity DataIC50: 423nMAssay Description:Inhibition of PI3KalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
LigandPNGBDBM50304671(1-(4-(4-(8-oxa-3-azabicyclo[3.2.1]octan-3-yl)thien...)
Affinity DataIC50: 825nMAssay Description:Inhibition of PI3KalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
LigandPNGBDBM50304679(1-(4-(4-(8-oxa-3-azabicyclo[3.2.1]octan-3-yl)-6-((...)
Affinity DataIC50: 874nMAssay Description:Inhibition of PI3KalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
LigandPNGBDBM50304670(1-(4-(4-(8-oxa-3-azabicyclo[3.2.1]octan-3-yl)thien...)
Affinity DataIC50: 1.26E+3nMAssay Description:Inhibition of PI3KalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
LigandPNGBDBM50304673(1-(4-(4-(8-oxa-3-azabicyclo[3.2.1]octan-3-yl)thien...)
Affinity DataIC50: 1.36E+3nMAssay Description:Inhibition of PI3KalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
LigandPNGBDBM50304685(5-(4-(8-oxa-3-azabicyclo[3.2.1]octan-3-yl)thieno[3...)
Affinity DataIC50: 1.77E+3nMAssay Description:Inhibition of PI3KalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
LigandPNGBDBM50304688(N-(4-(4-(8-oxa-3-azabicyclo[3.2.1]octan-3-yl)thien...)
Affinity DataIC50: 4.37E+3nMAssay Description:Inhibition of PI3KalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
LigandPNGBDBM50304668(methyl 4-(4-(8-oxa-3-azabicyclo[3.2.1]octan-3-yl)t...)
Affinity DataIC50: 6.20E+3nMAssay Description:Inhibition of PI3KalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
LigandPNGBDBM50304684(4-(4-(8-oxa-3-azabicyclo[3.2.1]octan-3-yl)thieno[3...)
Affinity DataIC50: 6.27E+3nMAssay Description:Inhibition of PI3KalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
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