Compile Data Set for Download or QSAR
Report error Found 43 Enz. Inhib. hit(s) with all data for entry = 50031366
TargetNeuropeptide Y receptor type 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50312042BDBM50312042((S)-N-(4-(4-phenyl-5,6-dihydro-4H-1,3-thiazin-2-yl...)
Affinity DataKi:  30nMAssay Description:Displacement of [125I]pig PPY from human NPY1 receptor expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50312032BDBM50312032((+/-)-N-(4-(4-methyl-5,6-dihydro-4H-1,3-thiazin-2-...)
Affinity DataKi:  50nMAssay Description:Displacement of [125I]pig PPY from human NPY1 receptor expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50312033BDBM50312033((+/-)-N-(4-(4-isopropyl-5,6-dihydro-4H-1,3-thiazin...)
Affinity DataKi:  53nMAssay Description:Displacement of [125I]pig PPY from human NPY1 receptor expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50312038BDBM50312038((+/-)-N-(4-(4-(4-methoxyphenyl)-5,6-dihydro-4H-1,3...)
Affinity DataKi:  55nMAssay Description:Displacement of [125I]pig PPY from human NPY1 receptor expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50312037BDBM50312037((+/-)-N-(4-(4-phenyl-5,6-dihydro-4H-1,3-thiazin-2-...)
Affinity DataKi:  55nMAssay Description:Displacement of [125I]pig PPY from human NPY1 receptor expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50312034BDBM50312034((+/-)-N-(4-(4-isobutyl-5,6-dihydro-4H-1,3-thiazin-...)
Affinity DataKi:  62nMAssay Description:Displacement of [125I]pig PPY from human NPY1 receptor expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50312028BDBM50312028((+/-)-N-(4-(4-butyl-4,5-dihydrothiazol-2-ylamino)p...)
Affinity DataKi:  69nMAssay Description:Displacement of [125I]pig PPY from human NPY1 receptor expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50312040BDBM50312040((+/-)-N-(4-(4-(3-chlorophenyl)-5,6-dihydro-4H-1,3-...)
Affinity DataKi:  107nMAssay Description:Displacement of [125I]pig PPY from human NPY1 receptor expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50312039BDBM50312039((+/-)-N-(4-(4-(4-chlorophenyl)-5,6-dihydro-4H-1,3-...)
Affinity DataKi:  122nMAssay Description:Displacement of [125I]pig PPY from human NPY1 receptor expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50312026BDBM50312026((R)-N-(4-(4-ethyl-4,5-dihydrothiazol-2-ylamino)phe...)
Affinity DataKi:  153nMAssay Description:Displacement of [125I]pig PPY from human NPY1 receptor expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50312030BDBM50312030((R)-N-(4-(4-phenyl-4,5-dihydrothiazol-2-ylamino)ph...)
Affinity DataKi:  175nMAssay Description:Displacement of [125I]pig PPY from human NPY1 receptor expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50312035BDBM50312035((+/-)-N-(4-(4-phenethyl-5,6-dihydro-4H-1,3-thiazin...)
Affinity DataKi:  195nMAssay Description:Displacement of [125I]pig PPY from human NPY1 receptor expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50312017BDBM50312017(N-(4-(5,6-dihydro-4H-1,3-thiazin-2-ylamino)pheneth...)
Affinity DataKi:  221nMAssay Description:Displacement of [125I]pig PPY from human NPY1 receptor expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50312007BDBM50312007(N-(4-(4,5-dihydrothiazol-2-ylamino)phenethyl)benzo...)
Affinity DataKi:  248nMAssay Description:Displacement of [125I]pig PPY from human NPY1 receptor expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50312024BDBM50312024(5,6-dichloro-N-(4-(5,6-dihydro-4H-1,3-thiazin-2-yl...)
Affinity DataKi:  316nMAssay Description:Displacement of [125I]pig PPY from human NPY1 receptor expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50312020BDBM50312020(N-(4-(5,6-dihydro-4H-1,3-thiazin-2-ylamino)pheneth...)
Affinity DataKi:  318nMAssay Description:Displacement of [125I]pig PPY from human NPY1 receptor expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50312036BDBM50312036((+/-)-N-(4-(4-cyclohexyl-5,6-dihydro-4H-1,3-thiazi...)
Affinity DataKi:  332nMAssay Description:Displacement of [125I]pig PPY from human NPY1 receptor expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50312021BDBM50312021(6-chloro-N-(4-(5,6-dihydro-4H-1,3-thiazin-2-ylamin...)
Affinity DataKi:  342nMAssay Description:Displacement of [125I]pig PPY from human NPY1 receptor expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50312025BDBM50312025((R)-N-(4-(4-methyl-4,5-dihydrothiazol-2-ylamino)ph...)
Affinity DataKi:  379nMAssay Description:Displacement of [125I]pig PPY from human NPY1 receptor expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50312043BDBM50312043((R)-N-(4-(4-phenyl-5,6-dihydro-4H-1,3-thiazin-2-yl...)
Affinity DataKi:  464nMAssay Description:Displacement of [125I]pig PPY from human NPY1 receptor expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50312027BDBM50312027((+/-)-N-(4-(4-propyl-4,5-dihydrothiazol-2-ylamino)...)
Affinity DataKi:  482nMAssay Description:Displacement of [125I]pig PPY from human NPY1 receptor expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50312018BDBM50312018(N-(4-(5,6-dihydro-4H-1,3-thiazin-2-ylamino)pheneth...)
Affinity DataKi:  616nMAssay Description:Displacement of [125I]pig PPY from human NPY1 receptor expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50312029BDBM50312029((R)-N-(4-(4-isobutyl-4,5-dihydrothiazol-2-ylamino)...)
Affinity DataKi:  712nMAssay Description:Displacement of [125I]pig PPY from human NPY1 receptor expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50312041BDBM50312041((+/-)-N-(4-(4-(2-chlorophenyl)-5,6-dihydro-4H-1,3-...)
Affinity DataKi:  956nMAssay Description:Displacement of [125I]pig PPY from human NPY1 receptor expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50312010BDBM50312010(N-(4-(4,5-dihydrothiazol-2-ylamino)phenethyl)-6-me...)
Affinity DataKi:  1.06E+3nMAssay Description:Displacement of [125I]pig PPY from human NPY1 receptor expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50312012BDBM50312012(N-(4-(4,5-dihydrothiazol-2-ylamino)phenethyl)-6-fl...)
Affinity DataKi:  1.12E+3nMAssay Description:Displacement of [125I]pig PPY from human NPY1 receptor expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50312013BDBM50312013(6-chloro-N-(4-(4,5-dihydrothiazol-2-ylamino)phenet...)
Affinity DataKi:  1.24E+3nMAssay Description:Displacement of [125I]pig PPY from human NPY1 receptor expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50312019BDBM50312019(N-(4-(5,6-dihydro-4H-1,3-thiazin-2-ylamino)pheneth...)
Affinity DataKi:  1.25E+3nMAssay Description:Displacement of [125I]pig PPY from human NPY1 receptor expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50312011BDBM50312011(N-(4-(4,5-dihydrothiazol-2-ylamino)phenethyl)-6-me...)
Affinity DataKi:  1.67E+3nMAssay Description:Displacement of [125I]pig PPY from human NPY1 receptor expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50312031BDBM50312031(N-(4-(5-methoxy-4,5-dihydrothiazol-2-ylamino)phene...)
Affinity DataKi:  2.55E+3nMAssay Description:Displacement of [125I]pig PPY from human NPY1 receptor expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50312022BDBM50312022(N-(4-(5,6-dihydro-4H-1,3-thiazin-2-ylamino)pheneth...)
Affinity DataKi:  3.30E+3nMAssay Description:Displacement of [125I]pig PPY from human NPY1 receptor expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50312008BDBM50312008(N-(4-(4,5-dihydrothiazol-2-ylamino)phenethyl)-4-me...)
Affinity DataKi:  3.46E+3nMAssay Description:Displacement of [125I]pig PPY from human NPY1 receptor expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50312016BDBM50312016(5,6-dichloro-N-(4-(4,5-dihydrothiazol-2-ylamino)ph...)
Affinity DataKi:  3.64E+3nMAssay Description:Displacement of [125I]pig PPY from human NPY1 receptor expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50312009BDBM50312009(N-(4-(4,5-dihydrothiazol-2-ylamino)phenethyl)-4-me...)
Affinity DataKi:  3.99E+3nMAssay Description:Displacement of [125I]pig PPY from human NPY1 receptor expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50312023BDBM50312023(N-(4-(5,6-dihydro-4H-1,3-thiazin-2-ylamino)pheneth...)
Affinity DataKi:  5.20E+3nMAssay Description:Displacement of [125I]pig PPY from human NPY1 receptor expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50312014BDBM50312014(N-(4-(4,5-dihydrothiazol-2-ylamino)phenethyl)-6-ni...)
Affinity DataKi:  5.25E+3nMAssay Description:Displacement of [125I]pig PPY from human NPY1 receptor expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50312015BDBM50312015(N-(4-(4,5-dihydrothiazol-2-ylamino)phenethyl)-6-(m...)
Affinity DataKi:  5.92E+3nMAssay Description:Displacement of [125I]pig PPY from human NPY1 receptor expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50312042BDBM50312042((S)-N-(4-(4-phenyl-5,6-dihydro-4H-1,3-thiazin-2-yl...)
Affinity DataKi:  5.98E+3nMAssay Description:Displacement of [125I]pig PPY from human NPY5 receptor expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50312042BDBM50312042((S)-N-(4-(4-phenyl-5,6-dihydro-4H-1,3-thiazin-2-yl...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I]human PP from human NPY4 receptor expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 4(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50312007BDBM50312007(N-(4-(4,5-dihydrothiazol-2-ylamino)phenethyl)benzo...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I]human PP from human NPY4 receptor expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 2(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50312042BDBM50312042((S)-N-(4-(4-phenyl-5,6-dihydro-4H-1,3-thiazin-2-yl...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I]pig PPY from human NPY2 receptor expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 2(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50312007BDBM50312007(N-(4-(4,5-dihydrothiazol-2-ylamino)phenethyl)benzo...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I]pig PPY from human NPY2 receptor expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50312007BDBM50312007(N-(4-(4,5-dihydrothiazol-2-ylamino)phenethyl)benzo...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I]pig PPY from human NPY5 receptor expressed in CHOK1 cells by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed