Compile Data Set for Download or QSAR
Report error Found 24 Enz. Inhib. hit(s) with all data for entry = 50041754
Target5-hydroxytryptamine receptor 1A(Human)
University of Porto

Curated by ChEMBL
LigandPNGBDBM50414860(CHEMBL574604)
Affinity DataKi:  11.0nMAssay Description:Displacement of [3H]8-OH-DPAT from human recombinant 5-HT1A receptor expressed in HEK293 cells after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
University of Porto

Curated by ChEMBL
LigandPNGBDBM50414857(CHEMBL576586)
Affinity DataKi:  15.8nMAssay Description:Displacement of [3H]ketanserin from 5-HT2A receptor in Wistar Hannover rat brain cortex membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
University of Porto

Curated by ChEMBL
LigandPNGBDBM50414865(CHEMBL573482)
Affinity DataKi:  30.2nMAssay Description:Displacement of [3H]8-OH-DPAT from human recombinant 5-HT1A receptor expressed in HEK293 cells after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
University of Porto

Curated by ChEMBL
LigandPNGBDBM50216040(3-(4-(4-phenyl-1-piperazinyl)butyl)quinazolin-4(3H...)
Affinity DataKi:  36.3nMAssay Description:Displacement of [3H]8-OH-DPAT from human recombinant 5-HT1A receptor expressed in HEK293 cells after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
University of Porto

Curated by ChEMBL
LigandPNGBDBM50414866(CHEMBL573264)
Affinity DataKi:  42.7nMAssay Description:Displacement of [3H]8-OH-DPAT from human recombinant 5-HT1A receptor expressed in HEK293 cells after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
University of Porto

Curated by ChEMBL
LigandPNGBDBM50414858(CHEMBL573256)
Affinity DataKi:  50.1nMAssay Description:Displacement of [3H]8-OH-DPAT from human recombinant 5-HT1A receptor expressed in HEK293 cells after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
University of Porto

Curated by ChEMBL
LigandPNGBDBM50414861(CHEMBL574827)
Affinity DataKi:  50.1nMAssay Description:Displacement of [3H]8-OH-DPAT from human recombinant 5-HT1A receptor expressed in HEK293 cells after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
University of Porto

Curated by ChEMBL
LigandPNGBDBM50414859(CHEMBL574822)
Affinity DataKi:  53.7nMAssay Description:Displacement of [3H]8-OH-DPAT from human recombinant 5-HT1A receptor expressed in HEK293 cells after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
University of Porto

Curated by ChEMBL
LigandPNGBDBM50414861(CHEMBL574827)
Affinity DataKi:  67.6nMAssay Description:Displacement of [3H]ketanserin from 5-HT2A receptor in Wistar Hannover rat brain cortex membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
University of Porto

Curated by ChEMBL
LigandPNGBDBM50414862(CHEMBL583583)
Affinity DataKi:  100nMAssay Description:Displacement of [3H]8-OH-DPAT from human recombinant 5-HT1A receptor expressed in HEK293 cells after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
University of Porto

Curated by ChEMBL
LigandPNGBDBM50414867(CHEMBL575032)
Affinity DataKi:  204nMAssay Description:Displacement of [3H]8-OH-DPAT from human recombinant 5-HT1A receptor expressed in HEK293 cells after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
University of Porto

Curated by ChEMBL
LigandPNGBDBM50414857(CHEMBL576586)
Affinity DataKi:  234nMAssay Description:Displacement of [3H]8-OH-DPAT from human recombinant 5-HT1A receptor expressed in HEK293 cells after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
University of Porto

Curated by ChEMBL
LigandPNGBDBM50414867(CHEMBL575032)
Affinity DataKi:  269nMAssay Description:Displacement of [3H]ketanserin from 5-HT2A receptor in Wistar Hannover rat brain cortex membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
University of Porto

Curated by ChEMBL
LigandPNGBDBM50414865(CHEMBL573482)
Affinity DataKi:  302nMAssay Description:Displacement of [3H]ketanserin from 5-HT2A receptor in Wistar Hannover rat brain cortex membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
University of Porto

Curated by ChEMBL
LigandPNGBDBM50414866(CHEMBL573264)
Affinity DataKi:  372nMAssay Description:Displacement of [3H]ketanserin from 5-HT2A receptor in Wistar Hannover rat brain cortex membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
University of Porto

Curated by ChEMBL
LigandPNGBDBM50414864(CHEMBL574828)
Affinity DataKi:  398nMAssay Description:Displacement of [3H]8-OH-DPAT from human recombinant 5-HT1A receptor expressed in HEK293 cells after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
University of Porto

Curated by ChEMBL
LigandPNGBDBM50414863(CHEMBL573237)
Affinity DataKi:  417nMAssay Description:Displacement of [3H]8-OH-DPAT from human recombinant 5-HT1A receptor expressed in HEK293 cells after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
University of Porto

Curated by ChEMBL
LigandPNGBDBM50414862(CHEMBL583583)
Affinity DataKi:  457nMAssay Description:Displacement of [3H]ketanserin from 5-HT2A receptor in Wistar Hannover rat brain cortex membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
University of Porto

Curated by ChEMBL
LigandPNGBDBM50216040(3-(4-(4-phenyl-1-piperazinyl)butyl)quinazolin-4(3H...)
Affinity DataKi:  562nMAssay Description:Displacement of [3H]ketanserin from 5-HT2A receptor in Wistar Hannover rat brain cortex membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
University of Porto

Curated by ChEMBL
LigandPNGBDBM50414864(CHEMBL574828)
Affinity DataKi:  575nMAssay Description:Displacement of [3H]ketanserin from 5-HT2A receptor in Wistar Hannover rat brain cortex membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
University of Porto

Curated by ChEMBL
LigandPNGBDBM50414863(CHEMBL573237)
Affinity DataKi:  661nMAssay Description:Displacement of [3H]ketanserin from 5-HT2A receptor in Wistar Hannover rat brain cortex membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
University of Porto

Curated by ChEMBL
LigandPNGBDBM50414860(CHEMBL574604)
Affinity DataKi:  1.45E+3nMAssay Description:Displacement of [3H]ketanserin from 5-HT2A receptor in Wistar Hannover rat brain cortex membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
University of Porto

Curated by ChEMBL
LigandPNGBDBM50414858(CHEMBL573256)
Affinity DataKi:  1.82E+3nMAssay Description:Displacement of [3H]ketanserin from 5-HT2A receptor in Wistar Hannover rat brain cortex membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
University of Porto

Curated by ChEMBL
LigandPNGBDBM50414859(CHEMBL574822)
Affinity DataKi:  2.14E+3nMAssay Description:Displacement of [3H]ketanserin from 5-HT2A receptor in Wistar Hannover rat brain cortex membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2013
Entry Details Article
PubMed