Compile Data Set for Download or QSAR
Report error Found 58 Enz. Inhib. hit(s) with all data for entry = 50030842
TargetProtein kinase C theta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50302529(4-(4-methyl-1H-indol-5-ylamino)-5-(4-(2-(4-methylp...)
Affinity DataIC50: 3.60nMAssay Description:Inhibition of human PKCtheta by IMAP kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50302507(4-(4-methyl-1H-indol-5-ylamino)-5-(3-(2-(4-methylp...)
Affinity DataIC50: 4.70nMAssay Description:Inhibition of human PKCtheta by IMAP kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50302531(4-(4-methyl-1H-indol-5-ylamino)-5-(3-(2-(pyrrolidi...)
Affinity DataIC50: 4.70nMAssay Description:Inhibition of human PKCtheta by IMAP kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50302526(5-(3-methoxystyryl)-4-(4-methyl-1H-indol-5-ylamino...)
Affinity DataIC50: 7nMAssay Description:Inhibition of human PKCtheta by IMAP kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetProtein kinase C epsilon type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50302507(4-(4-methyl-1H-indol-5-ylamino)-5-(3-(2-(4-methylp...)
Affinity DataIC50: 7nMAssay Description:Inhibition of PKCepsilon by IMAP kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50302528(4-(4-methyl-1H-indol-5-ylamino)-5-(2-(2-(4-methylp...)
Affinity DataIC50: 7.60nMAssay Description:Inhibition of human PKCtheta by IMAP kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50302525(5-(2-methoxystyryl)-4-(4-methyl-1H-indol-5-ylamino...)
Affinity DataIC50: 8.20nMAssay Description:Inhibition of human PKCtheta by IMAP kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50302509(4-(4-methyl-1H-indol-5-ylamino)-5-styrylnicotinoni...)
Affinity DataIC50: 8.30nMAssay Description:Inhibition of human PKCtheta by IMAP kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50302532(4-(4-methyl-1H-indol-5-ylamino)-5-(4-(2-(pyrrolidi...)
Affinity DataIC50: 9.10nMAssay Description:Inhibition of human PKCtheta by IMAP kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50302511(4-(3H-indol-4-ylamino)-5-styrylnicotinonitrile | C...)
Affinity DataIC50: 13nMAssay Description:Inhibition of human PKCtheta by IMAP kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50302530(4-(4-methyl-1H-indol-5-ylamino)-5-(2-(2-(pyrrolidi...)
Affinity DataIC50: 13nMAssay Description:Inhibition of human PKCtheta by IMAP kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50302527(5-(4-methoxystyryl)-4-(4-methyl-1H-indol-5-ylamino...)
Affinity DataIC50: 13nMAssay Description:Inhibition of human PKCtheta by IMAP kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50302510(4-(1H-indol-5-ylamino)-5-styrylnicotinonitrile | C...)
Affinity DataIC50: 24nMAssay Description:Inhibition of human PKCtheta by IMAP kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50302531(4-(4-methyl-1H-indol-5-ylamino)-5-(3-(2-(pyrrolidi...)
Affinity DataIC50: 25nMAssay Description:Inhibition of PKCdelta by IMAP kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50302524(5-(2-cyclohexylvinyl)-4-(4-methyl-1H-indol-5-ylami...)
Affinity DataIC50: 26nMAssay Description:Inhibition of human PKCtheta by IMAP kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50302528(4-(4-methyl-1H-indol-5-ylamino)-5-(2-(2-(4-methylp...)
Affinity DataIC50: 34nMAssay Description:Inhibition of PKCdelta by IMAP kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50302516(4-(4,7-dimethyl-1H-indol-5-ylamino)-5-styrylnicoti...)
Affinity DataIC50: 34nMAssay Description:Inhibition of human PKCtheta by IMAP kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50302523(4-(4-methyl-1H-indol-5-ylamino)-5-phenethylnicotin...)
Affinity DataIC50: 34nMAssay Description:Inhibition of human PKCtheta by IMAP kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50302529(4-(4-methyl-1H-indol-5-ylamino)-5-(4-(2-(4-methylp...)
Affinity DataIC50: 41nMAssay Description:Inhibition of PKCdelta by IMAP kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50302507(4-(4-methyl-1H-indol-5-ylamino)-5-(3-(2-(4-methylp...)
Affinity DataIC50: 53nMAssay Description:Inhibition of PKCdelta by IMAP kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50302526(5-(3-methoxystyryl)-4-(4-methyl-1H-indol-5-ylamino...)
Affinity DataIC50: 62nMAssay Description:Inhibition of PKCdelta by IMAP kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50302518(4-(6-chloro-1H-indol-5-ylamino)-5-styrylnicotinoni...)
Affinity DataIC50: 65nMAssay Description:Inhibition of human PKCtheta by IMAP kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50302515(4-(2,4-dimethyl-1H-indol-5-ylamino)-5-styrylnicoti...)
Affinity DataIC50: 70nMAssay Description:Inhibition of human PKCtheta by IMAP kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50302509(4-(4-methyl-1H-indol-5-ylamino)-5-styrylnicotinoni...)
Affinity DataIC50: 72nMAssay Description:Inhibition of PKCdelta by IMAP kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50302519(4-(7-chloro-4-methyl-1H-indol-5-ylamino)-5-styryln...)
Affinity DataIC50: 77nMAssay Description:Inhibition of human PKCtheta by IMAP kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50302508((Z)-4-(4-methyl-1H-indol-5-ylamino)-5-styrylnicoti...)
Affinity DataIC50: 79nMAssay Description:Inhibition of human PKCtheta by IMAP kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50302532(4-(4-methyl-1H-indol-5-ylamino)-5-(4-(2-(pyrrolidi...)
Affinity DataIC50: 81nMAssay Description:Inhibition of PKCdelta by IMAP kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50302521(4-(4-methyl-1H-indol-5-yloxy)-5-styrylnicotinonitr...)
Affinity DataIC50: 90nMAssay Description:Inhibition of human PKCtheta by IMAP kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50302511(4-(3H-indol-4-ylamino)-5-styrylnicotinonitrile | C...)
Affinity DataIC50: 96nMAssay Description:Inhibition of PKCdelta by IMAP kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50302525(5-(2-methoxystyryl)-4-(4-methyl-1H-indol-5-ylamino...)
Affinity DataIC50: 110nMAssay Description:Inhibition of PKCdelta by IMAP kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50302530(4-(4-methyl-1H-indol-5-ylamino)-5-(2-(2-(pyrrolidi...)
Affinity DataIC50: 140nMAssay Description:Inhibition of PKCdelta by IMAP kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50302527(5-(4-methoxystyryl)-4-(4-methyl-1H-indol-5-ylamino...)
Affinity DataIC50: 150nMAssay Description:Inhibition of PKCdelta by IMAP kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50302517(4-(1,4-dimethyl-1H-indol-5-ylamino)-5-styrylnicoti...)
Affinity DataIC50: 190nMAssay Description:Inhibition of human PKCtheta by IMAP kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50302510(4-(1H-indol-5-ylamino)-5-styrylnicotinonitrile | C...)
Affinity DataIC50: 240nMAssay Description:Inhibition of PKCdelta by IMAP kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetProtein kinase C eta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50302507(4-(4-methyl-1H-indol-5-ylamino)-5-(3-(2-(4-methylp...)
Affinity DataIC50: 330nMAssay Description:Inhibition of PKCeta by IMAP kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50302508((Z)-4-(4-methyl-1H-indol-5-ylamino)-5-styrylnicoti...)
Affinity DataIC50: 350nMAssay Description:Inhibition of PKCdelta by IMAP kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50302514(4-(2-methyl-1H-indol-5-ylamino)-5-styrylnicotinoni...)
Affinity DataIC50: 360nMAssay Description:Inhibition of human PKCtheta by IMAP kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50302524(5-(2-cyclohexylvinyl)-4-(4-methyl-1H-indol-5-ylami...)
Affinity DataIC50: 420nMAssay Description:Inhibition of PKCdelta by IMAP kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50302522(4-((1H-indol-5-yl)(methyl)amino)-5-styrylnicotinon...)
Affinity DataIC50: 440nMAssay Description:Inhibition of human PKCtheta by IMAP kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lck(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50302507(4-(4-methyl-1H-indol-5-ylamino)-5-(3-(2-(4-methylp...)
Affinity DataIC50: 520nMAssay Description:Inhibition of LckMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lyn(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50302507(4-(4-methyl-1H-indol-5-ylamino)-5-(3-(2-(4-methylp...)
Affinity DataIC50: 520nMAssay Description:Inhibition of LynMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50302515(4-(2,4-dimethyl-1H-indol-5-ylamino)-5-styrylnicoti...)
Affinity DataIC50: 620nMAssay Description:Inhibition of PKCdelta by IMAP kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50302523(4-(4-methyl-1H-indol-5-ylamino)-5-phenethylnicotin...)
Affinity DataIC50: 670nMAssay Description:Inhibition of PKCdelta by IMAP kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50302520(4-(1H-indol-5-yloxy)-5-styrylnicotinonitrile | CHE...)
Affinity DataIC50: 690nMAssay Description:Inhibition of human PKCtheta by IMAP kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50302514(4-(2-methyl-1H-indol-5-ylamino)-5-styrylnicotinoni...)
Affinity DataIC50: 800nMAssay Description:Inhibition of PKCdelta by IMAP kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50302519(4-(7-chloro-4-methyl-1H-indol-5-ylamino)-5-styryln...)
Affinity DataIC50: 880nMAssay Description:Inhibition of PKCdelta by IMAP kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50302518(4-(6-chloro-1H-indol-5-ylamino)-5-styrylnicotinoni...)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of PKCdelta by IMAP kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetProtein kinase C beta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50302507(4-(4-methyl-1H-indol-5-ylamino)-5-(3-(2-(4-methylp...)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of PKCbeta by IMAP kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50302516(4-(4,7-dimethyl-1H-indol-5-ylamino)-5-styrylnicoti...)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of PKCdelta by IMAP kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50302512(4-(1H-indol-6-ylamino)-5-styrylnicotinonitrile | C...)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of human PKCtheta by IMAP kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
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