Compile Data Set for Download or QSAR
Report error Found 16 Enz. Inhib. hit(s) with all data for entry = 50030741
TargetCannabinoid receptor 1(Rat)
Instituto De Qu£Mica M£Dica

Curated by ChEMBL
LigandPNGBDBM22988(Arachidonoyl ethanolamide | Arachidonoylethanolami...)
Affinity DataKi:  132nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellar membrane after 90 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Instituto De Qu£Mica M£Dica

Curated by ChEMBL
LigandPNGBDBM50300767({[(9Z)-octadec-9-en-1-yl]sulfamoyl}amine | CHEMBL5...)
Affinity DataKi:  1.89E+3nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellar membrane after 90 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Instituto De Qu£Mica M£Dica

Curated by ChEMBL
LigandPNGBDBM50300765(N-(cis-5-cis-8-cis-11-cis-14-eicosatetraenyl)-N'-p...)
Affinity DataKi:  2.34E+3nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellar membrane after 90 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Instituto De Qu£Mica M£Dica

Curated by ChEMBL
LigandPNGBDBM50300770(N-(cis-5-cis-8-cis-11-cis-14-eicosatetraenyl)sulfa...)
Affinity DataKi:  4.01E+3nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellar membrane after 90 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Instituto De Qu£Mica M£Dica

Curated by ChEMBL
LigandPNGBDBM50300769(N-(1-adamantyl)-N'-propylsulfamide | CHEMBL374746)
Affinity DataKi:  4.23E+3nMAssay Description:Displacement of [3H]WIN-55212-2 from CB1 receptor in rat cerebellar membrane after 90 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Instituto De Qu£Mica M£Dica

Curated by ChEMBL
LigandPNGBDBM50300771(N-(cis-9-cis-12-octadecadienyl)sulfamide | CHEMBL5...)
Affinity DataKi:  6.41E+3nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellar membrane after 90 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Instituto De Qu£Mica M£Dica

Curated by ChEMBL
LigandPNGBDBM50202584(N-(2-adamantyl)-N'-propylsulfamide | CHEMBL218643)
Affinity DataKi:  6.67E+3nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellar membrane after 90 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Instituto De Qu£Mica M£Dica

Curated by ChEMBL
LigandPNGBDBM50300766(N-(cis-9-cis-12-octadecadienyl)-N'-propylsulfamide...)
Affinity DataKi:  7.19E+3nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellar membrane after 90 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Instituto De Qu£Mica M£Dica

Curated by ChEMBL
LigandPNGBDBM50300769(N-(1-adamantyl)-N'-propylsulfamide | CHEMBL374746)
Affinity DataKi:  8.58E+3nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellar membrane after 90 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Instituto De Qu£Mica M£Dica

Curated by ChEMBL
LigandPNGBDBM50202583(N-octadecyl-N'-propylsulfamide | CHEMBL219156)
Affinity DataKi:  9.10E+3nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellar membrane after 90 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Instituto De Qu£Mica M£Dica

Curated by ChEMBL
LigandPNGBDBM50300764(N-oleyl-N'-propylsulfamide | CHEMBL571044)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellar membrane after 90 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Instituto De Qu£Mica M£Dica

Curated by ChEMBL
LigandPNGBDBM50202579(N-octadecylsulfamide | CHEMBL218794)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellar membrane after 90 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Instituto De Qu£Mica M£Dica

Curated by ChEMBL
LigandPNGBDBM50300768(N-(1-(1-adamantyl)ethyl)-N'-propylsulfamide | CHEM...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellar membrane after 90 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Instituto De Qu£Mica M£Dica

Curated by ChEMBL
LigandPNGBDBM50202583(N-octadecyl-N'-propylsulfamide | CHEMBL219156)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]WIN-55212-2 from CB1 receptor in rat cerebellar membrane after 90 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Instituto De Qu£Mica M£Dica

Curated by ChEMBL
LigandPNGBDBM50202584(N-(2-adamantyl)-N'-propylsulfamide | CHEMBL218643)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]WIN-55212-2 from CB1 receptor in rat cerebellar membrane after 90 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
Instituto De Qu£Mica M£Dica

Curated by ChEMBL
LigandPNGBDBM50300768(N-(1-(1-adamantyl)ethyl)-N'-propylsulfamide | CHEM...)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]WIN-55212-2 from CB1 receptor in rat cerebellar membrane after 90 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed