Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 50038909
TargetBcl-2-like protein 1(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM21447(4-(4-{[2-(4-chlorophenyl)phenyl]methyl}piperazin-1...)
Affinity DataKi:  188nMAssay Description:Inhibition of recombinant His6-tagged Bcl-XL expressed in Escherichia coli BL21 (DE3) and Flu-Bak peptide interaction by fluorescence polarization as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2012
Entry Details Article
PubMed
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM23223(Tash 1 | Gossypol, 4 | 7-[8-formyl-1,6,7-trihydrox...)
Affinity DataKi:  6.54E+3nMAssay Description:Inhibition of recombinant His6-tagged MCL1 (171-326) expressed in Escherichia coli BL21 (DE3) and Flu-Bak peptide interaction by fluorescence polariz...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2012
Entry Details Article
PubMed
TargetBcl-2-like protein 1(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50297392(ethyl 2-amino-4-(2-ethoxy-2-oxoethyl)-6-phenyl-4H-...)
Affinity DataKi:  3.44E+5nMAssay Description:Inhibition of recombinant His6-tagged Bcl-XL expressed in Escherichia coli BL21 (DE3) and Flu-Bak peptide interaction by fluorescence polarization as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2012
Entry Details Article
PubMed
TargetBcl-2-like protein 1(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50200965(Ethyl-2-amino-6-bromo-4-(1-cyano-2-ethoxy-2-oxoeth...)
Affinity DataKi:  6.60E+5nMAssay Description:Inhibition of recombinant His6-tagged Bcl-XL expressed in Escherichia coli BL21 (DE3) and Flu-Bak peptide interaction by fluorescence polarization as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2012
Entry Details Article
PubMed
TargetBcl-2-like protein 1(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50297393(Ethyl 2-Amino-6-(3',5'-dimethoxyphenyl)-4-(2-ethox...)
Affinity DataKi:  1.24E+6nMAssay Description:Inhibition of recombinant His6-tagged Bcl-XL expressed in Escherichia coli BL21 (DE3) and Flu-Bak peptide interaction by fluorescence polarization as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2012
Entry Details Article
PubMed
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50297393(Ethyl 2-Amino-6-(3',5'-dimethoxyphenyl)-4-(2-ethox...)
Affinity DataKi:  4.20E+7nMAssay Description:Inhibition of recombinant His6-tagged MCL1 (171-326) expressed in Escherichia coli BL21 (DE3) and Flu-Bak peptide interaction by fluorescence polariz...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2012
Entry Details Article
PubMed