Compile Data Set for Download or QSAR
Report error Found 52 Enz. Inhib. hit(s) with all data for entry = 50030935
TargetAcetylcholinesterase(Rat)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50304245(6,7-Dimethoxy-3-[4-(pyrrolidin-1-ylmethyl)-phenyl]...)
Affinity DataIC50: 4nMAssay Description:Inhibition of AChE in rat cortex after 15 mins by modified Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetAcetylcholinesterase(Rat)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM8960(2-[(1-benzylpiperidin-4-yl)methyl]-5,6-dimethoxy-2...)
Affinity DataIC50: 12nMAssay Description:Inhibition of AChE in rat cortex after 15 mins by modified Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetAcetylcholinesterase(Rat)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50304246(6,7-Dimethoxy-2-[4-(piperidin-1-ylmethyl)-phenyl]-...)
Affinity DataIC50: 34nMAssay Description:Inhibition of AChE in rat cortex after 15 mins by modified Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetAcetylcholinesterase(Rat)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50304249((E)-1-(2-Hydroxy-4,5-dimethoxyphenyl)-3-[4-(pyrrol...)
Affinity DataIC50: 37nMAssay Description:Inhibition of AChE in rat cortex after 15 mins by modified Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetAcetylcholinesterase(Rat)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50304247((E)-1-(2-Hydroxy-4,5-dimethoxyphenyl)-3-[3-(pyrrol...)
Affinity DataIC50: 47nMAssay Description:Inhibition of AChE in rat cortex after 15 mins by modified Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetAcetylcholinesterase(Rat)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50304248(6,7-Dimethoxy-2-[4-(pyrrolidin-1-ylmethyl)-phenyl]...)
Affinity DataIC50: 55nMAssay Description:Inhibition of AChE in rat cortex after 15 mins by modified Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetAcetylcholinesterase(Rat)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50304250(6,7-Dimethoxy-3-[4-(piperidin-1-ylmethyl)-phenyl]-...)
Affinity DataIC50: 68nMAssay Description:Inhibition of AChE in rat cortex after 15 mins by modified Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetAcetylcholinesterase(Rat)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50304227(6,7-Dimethoxy-3-[3-(pyrrolidin-1-ylmethyl)-phenyl]...)
Affinity DataIC50: 70nMAssay Description:Inhibition of AChE in rat cortex after 15 mins by modified Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetAcetylcholinesterase(Rat)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50304228((E)-3-{4-[(Diethylamino)-methyl]-phenyl}-1-(2-hydr...)
Affinity DataIC50: 103nMAssay Description:Inhibition of AChE in rat cortex after 15 mins by modified Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetAcetylcholinesterase(Rat)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50304229((E)-1-(2-Hydroxy-4,5-dimethoxyphenyl)-3-[4-(piperi...)
Affinity DataIC50: 122nMAssay Description:Inhibition of AChE in rat cortex after 15 mins by modified Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetAcetylcholinesterase(Rat)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50304230((E)-3-{4-[(Ethylmethylamino)-methyl]-phenyl}-1-(2-...)
Affinity DataIC50: 126nMAssay Description:Inhibition of AChE in rat cortex after 15 mins by modified Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetAcetylcholinesterase(Rat)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50304231(6,7-Dimethoxy-3-{4-[(ethylmethylamino)-methyl]-phe...)
Affinity DataIC50: 171nMAssay Description:Inhibition of AChE in rat cortex after 15 mins by modified Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetAcetylcholinesterase(Rat)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50304232(6,7-Dimethoxy-2-[4-(piperidin-1-ylmethyl)-phenyl]-...)
Affinity DataIC50: 248nMAssay Description:Inhibition of AChE in rat cortex after 15 mins by modified Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetAcetylcholinesterase(Rat)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50304233(6,7-Dimethoxy-2-{4-[(ethylmethylamino)-methyl)-phe...)
Affinity DataIC50: 336nMAssay Description:Inhibition of AChE in rat cortex after 15 mins by modified Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetAcetylcholinesterase(Rat)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50304234(3-{3-[(Diethylamino)-methyl]-phenyl}-6,7-dimethoxy...)
Affinity DataIC50: 560nMAssay Description:Inhibition of AChE in rat cortex after 15 mins by modified Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetAcetylcholinesterase(Rat)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50304235(3-{4-[(Diethylamino)-methyl]-phenyl}-6,7-dimethoxy...)
Affinity DataIC50: 599nMAssay Description:Inhibition of AChE in rat cortex after 15 mins by modified Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetAcetylcholinesterase(Rat)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50304236(2-[4-(Diethylamino-methyl)-phenyl]-6,7-dimethoxy-4...)
Affinity DataIC50: 639nMAssay Description:Inhibition of AChE in rat cortex after 15 mins by modified Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetAcetylcholinesterase(Rat)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50304237(6,7-Dimethoxy-2-[3-(pyrrolidin-1-ylmethyl)-phenyl]...)
Affinity DataIC50: 704nMAssay Description:Inhibition of AChE in rat cortex after 15 mins by modified Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetAcetylcholinesterase(Rat)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50304238(6,7-Dimethoxy-2-[4-(pyrrolidin-1-ylmethyl)-phenyl]...)
Affinity DataIC50: 1.24E+3nMAssay Description:Inhibition of AChE in rat cortex after 15 mins by modified Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetAcetylcholinesterase(Rat)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50304239((E)-3-{3-[(Diethylamino)-methyl]-phenyl}-1-(2-hydr...)
Affinity DataIC50: 1.61E+3nMAssay Description:Inhibition of AChE in rat cortex after 15 mins by modified Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Rat)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM10620(3-[(1S)-1-(dimethylamino)ethyl]phenyl N-ethyl-N-me...)
Affinity DataIC50: 1.66E+3nMAssay Description:Inhibition of BChE in rat serum after 15 mins by modified Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetAcetylcholinesterase(Rat)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM10620(3-[(1S)-1-(dimethylamino)ethyl]phenyl N-ethyl-N-me...)
Affinity DataIC50: 2.25E+3nMAssay Description:Inhibition of AChE in rat cortex after 15 mins by modified Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetAcetylcholinesterase(Rat)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50304240(6,7-Dimethoxy-2-{4-[(ethylmethylamino)-methyl]-phe...)
Affinity DataIC50: 4.67E+3nMAssay Description:Inhibition of AChE in rat cortex after 15 mins by modified Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Rat)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM8960(2-[(1-benzylpiperidin-4-yl)methyl]-5,6-dimethoxy-2...)
Affinity DataIC50: 4.67E+3nMAssay Description:Inhibition of BChE in rat serum after 15 mins by modified Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetAcetylcholinesterase(Rat)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50304241(2-{4-[(Diethylamino)-methyl]-phenyl}-6,7-dimethoxy...)
Affinity DataIC50: 4.97E+3nMAssay Description:Inhibition of AChE in rat cortex after 15 mins by modified Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetAcetylcholinesterase(Rat)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50304242(6,7-Dimethoxy-2-[3-(pyrrolidin-1-ylmethyl)-phenyl]...)
Affinity DataIC50: 5.36E+3nMAssay Description:Inhibition of AChE in rat cortex after 15 mins by modified Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetAcetylcholinesterase(Rat)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50304243(2-{3-[(Diethylamino)-methyl]-phenyl}-6,7-dimethoxy...)
Affinity DataIC50: 5.99E+3nMAssay Description:Inhibition of AChE in rat cortex after 15 mins by modified Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Rat)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50304245(6,7-Dimethoxy-3-[4-(pyrrolidin-1-ylmethyl)-phenyl]...)
Affinity DataIC50: 1.83E+4nMAssay Description:Inhibition of BChE in rat serum after 15 mins by modified Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Rat)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50304232(6,7-Dimethoxy-2-[4-(piperidin-1-ylmethyl)-phenyl]-...)
Affinity DataIC50: 4.80E+4nMAssay Description:Inhibition of BChE in rat serum after 15 mins by modified Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Rat)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50304231(6,7-Dimethoxy-3-{4-[(ethylmethylamino)-methyl]-phe...)
Affinity DataIC50: 6.10E+4nMAssay Description:Inhibition of BChE in rat serum after 15 mins by modified Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Rat)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50304236(2-[4-(Diethylamino-methyl)-phenyl]-6,7-dimethoxy-4...)
Affinity DataIC50: 6.46E+4nMAssay Description:Inhibition of BChE in rat serum after 15 mins by modified Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Rat)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50304238(6,7-Dimethoxy-2-[4-(pyrrolidin-1-ylmethyl)-phenyl]...)
Affinity DataIC50: 6.82E+4nMAssay Description:Inhibition of BChE in rat serum after 15 mins by modified Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Rat)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50304246(6,7-Dimethoxy-2-[4-(piperidin-1-ylmethyl)-phenyl]-...)
Affinity DataIC50: 7.52E+4nMAssay Description:Inhibition of BChE in rat serum after 15 mins by modified Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Rat)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50304247((E)-1-(2-Hydroxy-4,5-dimethoxyphenyl)-3-[3-(pyrrol...)
Affinity DataIC50: 7.73E+4nMAssay Description:Inhibition of BChE in rat serum after 15 mins by modified Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Rat)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50304248(6,7-Dimethoxy-2-[4-(pyrrolidin-1-ylmethyl)-phenyl]...)
Affinity DataIC50: 8.97E+4nMAssay Description:Inhibition of BChE in rat serum after 15 mins by modified Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Rat)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50304250(6,7-Dimethoxy-3-[4-(piperidin-1-ylmethyl)-phenyl]-...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of BChE in rat serum after 15 mins by modified Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Rat)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50304237(6,7-Dimethoxy-2-[3-(pyrrolidin-1-ylmethyl)-phenyl]...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of BChE in rat serum after 15 mins by modified Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Rat)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50304227(6,7-Dimethoxy-3-[3-(pyrrolidin-1-ylmethyl)-phenyl]...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of BChE in rat serum after 15 mins by modified Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Rat)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50304234(3-{3-[(Diethylamino)-methyl]-phenyl}-6,7-dimethoxy...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of BChE in rat serum after 15 mins by modified Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Rat)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50304235(3-{4-[(Diethylamino)-methyl]-phenyl}-6,7-dimethoxy...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of BChE in rat serum after 15 mins by modified Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Rat)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50304242(6,7-Dimethoxy-2-[3-(pyrrolidin-1-ylmethyl)-phenyl]...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of BChE in rat serum after 15 mins by modified Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Rat)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50304244(2-{3-[(Diethylamino)-methyl]-phenyl}-6,7-dimethoxy...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of BChE in rat serum after 15 mins by modified Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Rat)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50304241(2-{4-[(Diethylamino)-methyl]-phenyl}-6,7-dimethoxy...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of BChE in rat serum after 15 mins by modified Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Rat)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50304240(6,7-Dimethoxy-2-{4-[(ethylmethylamino)-methyl]-phe...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of BChE in rat serum after 15 mins by modified Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Rat)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50304243(2-{3-[(Diethylamino)-methyl]-phenyl}-6,7-dimethoxy...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of BChE in rat serum after 15 mins by modified Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Rat)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50304233(6,7-Dimethoxy-2-{4-[(ethylmethylamino)-methyl)-phe...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of BChE in rat serum after 15 mins by modified Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Rat)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50304229((E)-1-(2-Hydroxy-4,5-dimethoxyphenyl)-3-[4-(piperi...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of BChE in rat serum after 15 mins by modified Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Rat)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50304249((E)-1-(2-Hydroxy-4,5-dimethoxyphenyl)-3-[4-(pyrrol...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of BChE in rat serum after 15 mins by modified Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Rat)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50304239((E)-3-{3-[(Diethylamino)-methyl]-phenyl}-1-(2-hydr...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of BChE in rat serum after 15 mins by modified Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetCarboxylic ester hydrolase(Rat)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50304228((E)-3-{4-[(Diethylamino)-methyl]-phenyl}-1-(2-hydr...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of BChE in rat serum after 15 mins by modified Ellman's methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
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