Compile Data Set for Download or QSAR
Report error Found 116 Enz. Inhib. hit(s) with all data for entry = 50039018
TargetDelta-type opioid receptor(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM50001683(CHEMBL294616 | 13-[2-Amino-3-(4-hydroxy-phenyl)-pr...)
Affinity DataEC50:  15nMAssay Description:Activity at delta opioid receptor expressed in HEK293 cells assessed as stimulation of [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetNociceptin receptor(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM50304173(3,4-dichloro-N-[(1S,5R,13R,14R,17S)-4-(cyclopropyl...)
Affinity DataEC50:  0.100nMAssay Description:Inverse agonist activity at NOP expressed in HEK293 cells assessed as inhibition of [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM50304176(17-Cyclopropylmethyl-3,14beta-dihydroxy-4,5alpha-e...)
Affinity DataEC50: >1.00E+4nMAssay Description:Inverse agonist activity at kappa opioid receptor expressed in HEK293 cells assessed as inhibition of [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetNociceptin receptor(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM50304174(4-chloro-N-[(1S,5R,13R,14R,17S)-4-(cyclopropylmeth...)
Affinity DataEC50:  88nMAssay Description:Inverse agonist activity at NOP expressed in HEK293 cells assessed as inhibition of [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM50304170(17-Cyclopropylmethyl-3,14beta-dihydroxy-4,5alpha-e...)
Affinity DataEC50: >1.00E+4nMAssay Description:Inverse agonist activity at kappa opioid receptor expressed in HEK293 cells assessed as inhibition of [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetNociceptin receptor(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM50304171(17-Cyclopropylmethyl-3,14beta-dihydroxy-4,5alpha-e...)
Affinity DataEC50:  3.60nMAssay Description:Inverse agonist activity at NOP expressed in HEK293 cells assessed as inhibition of [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM50304171(17-Cyclopropylmethyl-3,14beta-dihydroxy-4,5alpha-e...)
Affinity DataEC50: >1.00E+4nMAssay Description:Inverse agonist activity at kappa opioid receptor expressed in HEK293 cells assessed as inhibition of [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetNociceptin receptor(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM50304172(17-Cyclopropylmethyl-3,14beta-dihydroxy-4,5alpha-e...)
Affinity DataEC50:  15nMAssay Description:Inverse agonist activity at NOP expressed in HEK293 cells assessed as inhibition of [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM50304172(17-Cyclopropylmethyl-3,14beta-dihydroxy-4,5alpha-e...)
Affinity DataEC50:  0.400nMAssay Description:Inverse agonist activity at kappa opioid receptor expressed in HEK293 cells assessed as inhibition of [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetNociceptin receptor(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM50304176(17-Cyclopropylmethyl-3,14beta-dihydroxy-4,5alpha-e...)
Affinity DataEC50:  20nMAssay Description:Inverse agonist activity at NOP expressed in HEK293 cells assessed as inhibition of [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetNociceptin receptor(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM50304170(17-Cyclopropylmethyl-3,14beta-dihydroxy-4,5alpha-e...)
Affinity DataEC50:  94nMAssay Description:Inverse agonist activity at NOP expressed in HEK293 cells assessed as inhibition of [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetNociceptin receptor(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM50304175(17-Cyclopropylmethyl-3,14beta-dihydroxy-4,5alpha-e...)
Affinity DataEC50:  135nMAssay Description:Inverse agonist activity at NOP expressed in HEK293 cells assessed as inhibition of [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM50304175(17-Cyclopropylmethyl-3,14beta-dihydroxy-4,5alpha-e...)
Affinity DataEC50:  2.40nMAssay Description:Inverse agonist activity at kappa opioid receptor expressed in HEK293 cells assessed as inhibition of [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM50304176(17-Cyclopropylmethyl-3,14beta-dihydroxy-4,5alpha-e...)
Affinity DataEC50:  16nMAssay Description:Activity at mu opioid receptor expressed in HEK293 cells assessed as stimulation of [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM50304170(17-Cyclopropylmethyl-3,14beta-dihydroxy-4,5alpha-e...)
Affinity DataEC50:  4.5nMAssay Description:Activity at mu opioid receptor expressed in HEK293 cells assessed as stimulation of [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM50304175(17-Cyclopropylmethyl-3,14beta-dihydroxy-4,5alpha-e...)
Affinity DataEC50: >1.00E+4nMAssay Description:Activity at mu opioid receptor expressed in HEK293 cells assessed as stimulation of [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM50304173(3,4-dichloro-N-[(1S,5R,13R,14R,17S)-4-(cyclopropyl...)
Affinity DataEC50:  2.30nMAssay Description:Activity at mu opioid receptor expressed in HEK293 cells assessed as stimulation of [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM50304174(4-chloro-N-[(1S,5R,13R,14R,17S)-4-(cyclopropylmeth...)
Affinity DataEC50:  6.80nMAssay Description:Activity at mu opioid receptor expressed in HEK293 cells assessed as stimulation of [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM50304171(17-Cyclopropylmethyl-3,14beta-dihydroxy-4,5alpha-e...)
Affinity DataEC50:  8.80nMAssay Description:Activity at mu opioid receptor expressed in HEK293 cells assessed as stimulation of [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM50304172(17-Cyclopropylmethyl-3,14beta-dihydroxy-4,5alpha-e...)
Affinity DataEC50: >1.00E+4nMAssay Description:Activity at mu opioid receptor expressed in HEK293 cells assessed as stimulation of [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM50304171(17-Cyclopropylmethyl-3,14beta-dihydroxy-4,5alpha-e...)
Affinity DataEC50: >1.00E+4nMAssay Description:Inverse agonist activity at mu opioid receptor expressed in HEK293 cells assessed as inhibition of [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM50304171(17-Cyclopropylmethyl-3,14beta-dihydroxy-4,5alpha-e...)
Affinity DataEC50:  5.10nMAssay Description:Activity at delta opioid receptor expressed in HEK293 cells assessed as stimulation of [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM50304170(17-Cyclopropylmethyl-3,14beta-dihydroxy-4,5alpha-e...)
Affinity DataEC50: >1.00E+4nMAssay Description:Inverse agonist activity at mu opioid receptor expressed in HEK293 cells assessed as inhibition of [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM50304170(17-Cyclopropylmethyl-3,14beta-dihydroxy-4,5alpha-e...)
Affinity DataEC50:  0.200nMAssay Description:Activity at delta opioid receptor expressed in HEK293 cells assessed as stimulation of [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM50304174(4-chloro-N-[(1S,5R,13R,14R,17S)-4-(cyclopropylmeth...)
Affinity DataEC50: >1.00E+4nMAssay Description:Inverse agonist activity at delta opioid receptor expressed in HEK293 cells assessed as inhibition of [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM50304176(17-Cyclopropylmethyl-3,14beta-dihydroxy-4,5alpha-e...)
Affinity DataEC50: >1.00E+4nMAssay Description:Inverse agonist activity at mu opioid receptor expressed in HEK293 cells assessed as inhibition of [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM50304173(3,4-dichloro-N-[(1S,5R,13R,14R,17S)-4-(cyclopropyl...)
Affinity DataEC50:  1.40nMAssay Description:Activity at delta opioid receptor expressed in HEK293 cells assessed as stimulation of [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM50304175(17-Cyclopropylmethyl-3,14beta-dihydroxy-4,5alpha-e...)
Affinity DataEC50:  8.90nMAssay Description:Inverse agonist activity at mu opioid receptor expressed in HEK293 cells assessed as inhibition of [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM50304172(17-Cyclopropylmethyl-3,14beta-dihydroxy-4,5alpha-e...)
Affinity DataEC50: >1.00E+4nMAssay Description:Activity at delta opioid receptor expressed in HEK293 cells assessed as stimulation of [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM50304176(17-Cyclopropylmethyl-3,14beta-dihydroxy-4,5alpha-e...)
Affinity DataEC50:  5.10nMAssay Description:Activity at delta opioid receptor expressed in HEK293 cells assessed as stimulation of [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM50304175(17-Cyclopropylmethyl-3,14beta-dihydroxy-4,5alpha-e...)
Affinity DataEC50:  0.140nMAssay Description:Activity at delta opioid receptor expressed in HEK293 cells assessed as stimulation of [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM50304175(17-Cyclopropylmethyl-3,14beta-dihydroxy-4,5alpha-e...)
Affinity DataEC50: >1.00E+4nMAssay Description:Activity at kappa opioid receptor expressed in HEK293 cells assessed as stimulation of [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM50304176(17-Cyclopropylmethyl-3,14beta-dihydroxy-4,5alpha-e...)
Affinity DataEC50:  9.90nMAssay Description:Activity at kappa opioid receptor expressed in HEK293 cells assessed as stimulation of [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM50304176(17-Cyclopropylmethyl-3,14beta-dihydroxy-4,5alpha-e...)
Affinity DataEC50: >1.00E+4nMAssay Description:Inverse agonist activity at delta opioid receptor expressed in HEK293 cells assessed as inhibition of [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM50304170(17-Cyclopropylmethyl-3,14beta-dihydroxy-4,5alpha-e...)
Affinity DataEC50:  0.100nMAssay Description:Activity at kappa opioid receptor expressed in HEK293 cells assessed as stimulation of [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM50304175(17-Cyclopropylmethyl-3,14beta-dihydroxy-4,5alpha-e...)
Affinity DataEC50: >1.00E+4nMAssay Description:Inverse agonist activity at delta opioid receptor expressed in HEK293 cells assessed as inhibition of [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM50304171(17-Cyclopropylmethyl-3,14beta-dihydroxy-4,5alpha-e...)
Affinity DataEC50:  29nMAssay Description:Activity at kappa opioid receptor expressed in HEK293 cells assessed as stimulation of [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM50304171(17-Cyclopropylmethyl-3,14beta-dihydroxy-4,5alpha-e...)
Affinity DataEC50: >1.00E+4nMAssay Description:Inverse agonist activity at delta opioid receptor expressed in HEK293 cells assessed as inhibition of [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM50304172(17-Cyclopropylmethyl-3,14beta-dihydroxy-4,5alpha-e...)
Affinity DataEC50: >1.00E+4nMAssay Description:Activity at kappa opioid receptor expressed in HEK293 cells assessed as stimulation of [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM50304174(4-chloro-N-[(1S,5R,13R,14R,17S)-4-(cyclopropylmeth...)
Affinity DataEC50: >1.00E+4nMAssay Description:Inverse agonist activity at mu opioid receptor expressed in HEK293 cells assessed as inhibition of [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM50304174(4-chloro-N-[(1S,5R,13R,14R,17S)-4-(cyclopropylmeth...)
Affinity DataEC50:  42nMAssay Description:Activity at delta opioid receptor expressed in HEK293 cells assessed as stimulation of [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM50304170(17-Cyclopropylmethyl-3,14beta-dihydroxy-4,5alpha-e...)
Affinity DataEC50:  66nMAssay Description:Inverse agonist activity at delta opioid receptor expressed in HEK293 cells assessed as inhibition of [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM50304173(3,4-dichloro-N-[(1S,5R,13R,14R,17S)-4-(cyclopropyl...)
Affinity DataEC50:  0.900nMAssay Description:Activity at kappa opioid receptor expressed in HEK293 cells assessed as stimulation of [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM50304173(3,4-dichloro-N-[(1S,5R,13R,14R,17S)-4-(cyclopropyl...)
Affinity DataEC50: >1.00E+4nMAssay Description:Inverse agonist activity at mu opioid receptor expressed in HEK293 cells assessed as inhibition of [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM50304173(3,4-dichloro-N-[(1S,5R,13R,14R,17S)-4-(cyclopropyl...)
Affinity DataEC50: >1.00E+4nMAssay Description:Inverse agonist activity at delta opioid receptor expressed in HEK293 cells assessed as inhibition of [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM50304174(4-chloro-N-[(1S,5R,13R,14R,17S)-4-(cyclopropylmeth...)
Affinity DataEC50:  7.10nMAssay Description:Activity at kappa opioid receptor expressed in HEK293 cells assessed as stimulation of [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM50304172(17-Cyclopropylmethyl-3,14beta-dihydroxy-4,5alpha-e...)
Affinity DataEC50:  4.00E+3nMAssay Description:Inverse agonist activity at mu opioid receptor expressed in HEK293 cells assessed as inhibition of [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM50304172(17-Cyclopropylmethyl-3,14beta-dihydroxy-4,5alpha-e...)
Affinity DataEC50:  0.300nMAssay Description:Inverse agonist activity at delta opioid receptor expressed in HEK293 cells assessed as inhibition of [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM50304173(3,4-dichloro-N-[(1S,5R,13R,14R,17S)-4-(cyclopropyl...)
Affinity DataEC50: >1.00E+4nMAssay Description:Inverse agonist activity at kappa opioid receptor expressed in HEK293 cells assessed as inhibition of [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM50304174(4-chloro-N-[(1S,5R,13R,14R,17S)-4-(cyclopropylmeth...)
Affinity DataEC50: >1.00E+4nMAssay Description:Inverse agonist activity at kappa opioid receptor expressed in HEK293 cells assessed as inhibition of [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
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