Compile Data Set for Download or QSAR
Report error Found 49 Enz. Inhib. hit(s) with all data for entry = 50030802
TargetProtein kinase C theta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50301693(5-(5-((4-(dimethylamino)piperidin-1-yl)methyl)fura...)
Affinity DataIC50: 1.30nMAssay Description:Inhibition of human PKCtheta by IMAP kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50301694(5-(5-((4-isopropylpiperazin-1-yl)methyl)furan-3-yl...)
Affinity DataIC50: 2.40nMAssay Description:Inhibition of human PKCtheta by IMAP kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50301679(4-(4-methyl-1H-indol-5-ylamino)-5-(3-((4-methylpip...)
Affinity DataIC50: 3nMAssay Description:Inhibition of human PKCtheta by IMAP kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50301695(5-(5-((4-cyclopentylpiperazin-1-yl)methyl)furan-3-...)
Affinity DataIC50: 3.5nMAssay Description:Inhibition of human PKCtheta by IMAP kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50301686(1-((5-(3-ethynyl-2-((4-methyl-1H-inden-5-yl)methyl...)
Affinity DataIC50: 4.5nMAssay Description:Inhibition of human PKCtheta by IMAP kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50301685(1-((4-(3-ethynyl-2-((4-methyl-1H-inden-5-yl)methyl...)
Affinity DataIC50: 4.90nMAssay Description:Inhibition of human PKCtheta by IMAP kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50301678(4-(4-methyl-1H-indol-5-ylamino)-5-(4-((4-methylpip...)
Affinity DataIC50: 5nMAssay Description:Inhibition of human PKCtheta by IMAP kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50301684(4-(4-methyl-1H-indol-5-ylamino)-5-(5-((4-methylpip...)
Affinity DataIC50: 6.10nMAssay Description:Inhibition of human PKCtheta by IMAP kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50301676(5-(3-((dimethylamino)methyl)phenyl)-4-(4-methyl-1H...)
Affinity DataIC50: 6.90nMAssay Description:Inhibition of human PKCtheta by IMAP kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50301689(4-(4-methyl-1H-indol-5-ylamino)-5-(5-(thiomorpholi...)
Affinity DataIC50: 7.5nMAssay Description:Inhibition of human PKCtheta by IMAP kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50301688(4-(4-methyl-1H-indol-5-ylamino)-5-(5-(morpholinome...)
Affinity DataIC50: 7.80nMAssay Description:Inhibition of human PKCtheta by IMAP kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50301693(5-(5-((4-(dimethylamino)piperidin-1-yl)methyl)fura...)
Affinity DataIC50: 8.20nMAssay Description:Inhibition of human PKCdelta by IMAP kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50301675(5-(4-((dimethylamino)methyl)phenyl)-4-(4-methyl-1H...)
Affinity DataIC50: 8.40nMAssay Description:Inhibition of human PKCtheta by IMAP kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50301680(4-(4-methyl-1H-indol-5-ylamino)-5-(4-(morpholinome...)
Affinity DataIC50: 9nMAssay Description:Inhibition of human PKCtheta by IMAP kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50301685(1-((4-(3-ethynyl-2-((4-methyl-1H-inden-5-yl)methyl...)
Affinity DataIC50: 9.70nMAssay Description:Inhibition of human PKCdelta by IMAP kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50301687(4-(4-methyl-1H-indol-5-ylamino)-5-(5-((4-methylpip...)
Affinity DataIC50: 12nMAssay Description:Inhibition of human PKCtheta by IMAP kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetProtein kinase C epsilon type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50301686(1-((5-(3-ethynyl-2-((4-methyl-1H-inden-5-yl)methyl...)
Affinity DataIC50: 12nMAssay Description:Inhibition of PKCepsilon by IMAP kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50301694(5-(5-((4-isopropylpiperazin-1-yl)methyl)furan-3-yl...)
Affinity DataIC50: 14nMAssay Description:Inhibition of human PKCdelta by IMAP kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50301695(5-(5-((4-cyclopentylpiperazin-1-yl)methyl)furan-3-...)
Affinity DataIC50: 18nMAssay Description:Inhibition of human PKCdelta by IMAP kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50301679(4-(4-methyl-1H-indol-5-ylamino)-5-(3-((4-methylpip...)
Affinity DataIC50: 22nMAssay Description:Inhibition of human PKCdelta by IMAP kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50301681(4-(4-methyl-1H-indol-5-ylamino)-5-(3-(morpholinome...)
Affinity DataIC50: 23nMAssay Description:Inhibition of human PKCtheta by IMAP kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50301676(5-(3-((dimethylamino)methyl)phenyl)-4-(4-methyl-1H...)
Affinity DataIC50: 25nMAssay Description:Inhibition of human PKCdelta by IMAP kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50301678(4-(4-methyl-1H-indol-5-ylamino)-5-(4-((4-methylpip...)
Affinity DataIC50: 25nMAssay Description:Inhibition of human PKCdelta by IMAP kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50301691(4-(4-methyl-1H-indol-5-ylamino)-5-(5-(pyrrolidin-1...)
Affinity DataIC50: 35nMAssay Description:Inhibition of human PKCtheta by IMAP kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50301687(4-(4-methyl-1H-indol-5-ylamino)-5-(5-((4-methylpip...)
Affinity DataIC50: 36nMAssay Description:Inhibition of human PKCdelta by IMAP kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50301682(4-(4-methyl-1H-indol-5-ylamino)-6'-((4-methylpiper...)
Affinity DataIC50: 38nMAssay Description:Inhibition of human PKCtheta by IMAP kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50301690(4-(4-methyl-1H-indol-5-ylamino)-5-(5-(piperidin-1-...)
Affinity DataIC50: 41nMAssay Description:Inhibition of human PKCtheta by IMAP kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50301692(5-(5-((diethylamino)methyl)furan-2-yl)-4-(4-methyl...)
Affinity DataIC50: 42nMAssay Description:Inhibition of human PKCtheta by IMAP kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50301686(1-((5-(3-ethynyl-2-((4-methyl-1H-inden-5-yl)methyl...)
Affinity DataIC50: 45nMAssay Description:Inhibition of human PKCdelta by IMAP kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50301684(4-(4-methyl-1H-indol-5-ylamino)-5-(5-((4-methylpip...)
Affinity DataIC50: 50nMAssay Description:Inhibition of human PKCdelta by IMAP kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50301675(5-(4-((dimethylamino)methyl)phenyl)-4-(4-methyl-1H...)
Affinity DataIC50: 58nMAssay Description:Inhibition of human PKCdelta by IMAP kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50301680(4-(4-methyl-1H-indol-5-ylamino)-5-(4-(morpholinome...)
Affinity DataIC50: 70nMAssay Description:Inhibition of human PKCdelta by IMAP kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50301681(4-(4-methyl-1H-indol-5-ylamino)-5-(3-(morpholinome...)
Affinity DataIC50: 84nMAssay Description:Inhibition of human PKCdelta by IMAP kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50301688(4-(4-methyl-1H-indol-5-ylamino)-5-(5-(morpholinome...)
Affinity DataIC50: 86nMAssay Description:Inhibition of human PKCdelta by IMAP kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50301689(4-(4-methyl-1H-indol-5-ylamino)-5-(5-(thiomorpholi...)
Affinity DataIC50: 94nMAssay Description:Inhibition of human PKCdelta by IMAP kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetProtein kinase C eta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50301686(1-((5-(3-ethynyl-2-((4-methyl-1H-inden-5-yl)methyl...)
Affinity DataIC50: 140nMAssay Description:Inhibition of PKCeta by IMAP kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50301692(5-(5-((diethylamino)methyl)furan-2-yl)-4-(4-methyl...)
Affinity DataIC50: 190nMAssay Description:Inhibition of human PKCdelta by IMAP kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50301683(4-(4-methyl-1H-indol-5-ylamino)-5'-((4-methylpiper...)
Affinity DataIC50: 190nMAssay Description:Inhibition of human PKCtheta by IMAP kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetProtein kinase C theta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50301677(5-(2-((dimethylamino)methyl)phenyl)-4-(4-methyl-1H...)
Affinity DataIC50: 200nMAssay Description:Inhibition of human PKCtheta by IMAP kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50301682(4-(4-methyl-1H-indol-5-ylamino)-6'-((4-methylpiper...)
Affinity DataIC50: 250nMAssay Description:Inhibition of human PKCdelta by IMAP kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50301691(4-(4-methyl-1H-indol-5-ylamino)-5-(5-(pyrrolidin-1...)
Affinity DataIC50: 300nMAssay Description:Inhibition of human PKCdelta by IMAP kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50301690(4-(4-methyl-1H-indol-5-ylamino)-5-(5-(piperidin-1-...)
Affinity DataIC50: 390nMAssay Description:Inhibition of human PKCdelta by IMAP kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lck(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50301686(1-((5-(3-ethynyl-2-((4-methyl-1H-inden-5-yl)methyl...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of LckMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50301677(5-(2-((dimethylamino)methyl)phenyl)-4-(4-methyl-1H...)
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of human PKCdelta by IMAP kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetProtein kinase C beta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50301686(1-((5-(3-ethynyl-2-((4-methyl-1H-inden-5-yl)methyl...)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of PKCbeta by IMAP kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lyn(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50301686(1-((5-(3-ethynyl-2-((4-methyl-1H-inden-5-yl)methyl...)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of LynMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetMAP kinase-activated protein kinase 2(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50301686(1-((5-(3-ethynyl-2-((4-methyl-1H-inden-5-yl)methyl...)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of MK2More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetRho-associated protein kinase 1(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50301686(1-((5-(3-ethynyl-2-((4-methyl-1H-inden-5-yl)methyl...)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of ROCK1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetProtein kinase C zeta type(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50301686(1-((5-(3-ethynyl-2-((4-methyl-1H-inden-5-yl)methyl...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of PKCzeta by IMAP kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed