Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50030790
TargetEpidermal growth factor receptor(Human)
Mcgill University/Royal Victoria Hospital

Curated by ChEMBL
LigandPNGBDBM5447(ZD1839 | N-(3-chloro-4-fluorophenyl)-7-methoxy-6-[...)
Affinity DataIC50: 33nMAssay Description:Inhibition of EGFR-mediated poly(L-glutamic acid L-tyrosine) phosphorylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetEpidermal growth factor receptor(Human)
Mcgill University/Royal Victoria Hospital

Curated by ChEMBL
LigandPNGBDBM50301422(vinyl 3-(4-(3-chlorophenylamino)quinazolin-6-yl)-1...)
Affinity DataIC50: 180nMAssay Description:Inhibition of EGFR-mediated poly(L-glutamic acid L-tyrosine) phosphorylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Mcgill University/Royal Victoria Hospital

Curated by ChEMBL
LigandPNGBDBM50301421((3-(4-(3-chlorophenylamino)quinazolin-6-yl)-1-meth...)
Affinity DataIC50: 240nMAssay Description:Inhibition of EGFR-mediated poly(L-glutamic acid L-tyrosine) phosphorylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Mcgill University/Royal Victoria Hospital

Curated by ChEMBL
LigandPNGBDBM50301426(chloromethyl 3-(4-(3-chlorophenylamino)quinazolin-...)
Affinity DataIC50: 390nMAssay Description:Inhibition of EGFR-mediated poly(L-glutamic acid L-tyrosine) phosphorylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Mcgill University/Royal Victoria Hospital

Curated by ChEMBL
LigandPNGBDBM50301424(2-chloroethyl 3-(4-(3-chlorophenylamino)quinazolin...)
Affinity DataIC50: 500nMAssay Description:Inhibition of EGFR-mediated poly(L-glutamic acid L-tyrosine) phosphorylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Mcgill University/Royal Victoria Hospital

Curated by ChEMBL
LigandPNGBDBM50301425(acetoxymethyl 3-(4-(3-chlorophenylamino)quinazolin...)
Affinity DataIC50: 630nMAssay Description:Inhibition of EGFR-mediated poly(L-glutamic acid L-tyrosine) phosphorylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Mcgill University/Royal Victoria Hospital

Curated by ChEMBL
LigandPNGBDBM50301423(vinyl 3-(4-(3-chlorophenylamino)quinazolin-6-yl)-1...)
Affinity DataIC50: 720nMAssay Description:Inhibition of EGFR-mediated poly(L-glutamic acid L-tyrosine) phosphorylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Mcgill University/Royal Victoria Hospital

Curated by ChEMBL
LigandPNGBDBM50301427(4-nitrophenyl 3-(4-(3-chlorophenylamino)quinazolin...)
Affinity DataIC50: 770nMAssay Description:Inhibition of EGFR-mediated poly(L-glutamic acid L-tyrosine) phosphorylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed