Compile Data Set for Download or QSAR
Report error Found 24 Enz. Inhib. hit(s) with all data for entry = 50030779
TargetD(1A) dopamine receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 82247BDBM82247(SCH 23390,R(+) | CAS_87134-87-0 | CHEMBL2158641 | ...)
Affinity DataKi:  1nMAssay Description:Displacement of [3H]SCH23390 from human D1 receptor expressed in Ltk cellMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50280442BDBM50280442(8-Chloro-3-methyl-2,3,4,5-tetrahydro-1H-benzo[d]az...)
Affinity DataKi:  50nMAssay Description:Displacement of [3H]SCH23390 from human D1 receptor expressed in Ltk cellMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50301259BDBM50301259(7-chloro-2-methyl-1-(thiophen-3-yl)-4,5-dihydro-1H...)
Affinity DataKi:  87nMAssay Description:Displacement of [3H]SCH23390 from human D1 receptor expressed in Ltk cellMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50301272BDBM50301272(7-chloro-2-(cyclohexylamino)-4,5-dihydro-1H-benzo[...)
Affinity DataKi:  129nMAssay Description:Displacement of [3H]SCH23390 from human D1 receptor expressed in Ltk cellMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50301262BDBM50301262(7-chloro-2-(4-(dimethylamino)styryl)-1-phenyl-4,5-...)
Affinity DataKi:  154nMAssay Description:Displacement of [3H]SCH23390 from human D1 receptor expressed in Ltk cellMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50301260BDBM50301260(7-chloro-2-methyl-1-p-tolyl-4,5-dihydro-1H-benzo[d...)
Affinity DataKi:  181nMAssay Description:Displacement of [3H]SCH23390 from human D1 receptor expressed in Ltk cellMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50301264BDBM50301264(7-chloro-2-(6-methoxynaphthalen-2-yl)-4,5-dihydro-...)
Affinity DataKi:  198nMAssay Description:Displacement of [3H]SCH23390 from human D1 receptor expressed in Ltk cellMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50301257BDBM50301257(7-chloro-2-methyl-1-phenyl-4,5-dihydro-1H-benzo[d]...)
Affinity DataKi:  200nMAssay Description:Displacement of [3H]SCH23390 from human D1 receptor expressed in Ltk cellMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50301268BDBM50301268(7-chloro-2-(4-methoxystyryl)-4,5-dihydro-1H-benzo[...)
Affinity DataKi:  206nMAssay Description:Displacement of [3H]SCH23390 from human D1 receptor expressed in Ltk cellMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50301267BDBM50301267(7-chloro-2-cyclohexyl-4,5-dihydro-1H-benzo[d][1,3]...)
Affinity DataKi:  284nMAssay Description:Displacement of [3H]SCH23390 from human D1 receptor expressed in Ltk cellMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50301269BDBM50301269(7-chloro-2-(2-(4-methoxyphenyl)cyclopropyl)-4,5-di...)
Affinity DataKi:  311nMAssay Description:Displacement of [3H]SCH23390 from human D1 receptor expressed in Ltk cellMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50301261BDBM50301261(7-chloro-2-methyl-1-o-tolyl-4,5-dihydro-1H-benzo[d...)
Affinity DataKi:  321nMAssay Description:Displacement of [3H]SCH23390 from human D1 receptor expressed in Ltk cellMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50301263BDBM50301263(7-chloro-1-cyclohexyl-2-(4-(dimethylamino)styryl)-...)
Affinity DataKi:  370nMAssay Description:Displacement of [3H]SCH23390 from human D1 receptor expressed in Ltk cellMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50301273BDBM50301273(7-chloro-2-(cyclopentylamino)-4,5-dihydro-1H-benzo...)
Affinity DataKi:  391nMAssay Description:Displacement of [3H]SCH23390 from human D1 receptor expressed in Ltk cellMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50301265BDBM50301265(7-chloro-2-isobutyl-4,5-dihydro-1H-benzo[d][1,3]di...)
Affinity DataKi:  442nMAssay Description:Displacement of [3H]SCH23390 from human D1 receptor expressed in Ltk cellMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50301275BDBM50301275(2-(benzylthio)-7-chloro-4,5-dihydro-1H-benzo[d][1,...)
Affinity DataKi:  445nMAssay Description:Displacement of [3H]SCH23390 from human D1 receptor expressed in Ltk cellMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50301274BDBM50301274(7-chloro-2-(phenethylamino)-4,5-dihydro-1H-benzo[d...)
Affinity DataKi:  465nMAssay Description:Displacement of [3H]SCH23390 from human D1 receptor expressed in Ltk cellMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50301266BDBM50301266(7-chloro-2-phenyl-4,5-dihydro-1H-benzo[d][1,3]diaz...)
Affinity DataKi:  475nMAssay Description:Displacement of [3H]SCH23390 from human D1 receptor expressed in Ltk cellMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50301276BDBM50301276(7-chloro-2-(cyclopropylamino)-4,5-dihydro-1H-benzo...)
Affinity DataKi:  575nMAssay Description:Displacement of [3H]SCH23390 from human D1 receptor expressed in Ltk cellMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50301277BDBM50301277(7-chloro-2-(methylamino)-4,5-dihydro-1H-benzo[d][1...)
Affinity DataKi:  783nMAssay Description:Displacement of [3H]SCH23390 from human D1 receptor expressed in Ltk cellMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50301278BDBM50301278(7-chloro-2-(methylthio)-4,5-dihydro-1H-benzo[d][1,...)
Affinity DataKi:  900nMAssay Description:Displacement of [3H]SCH23390 from human D1 receptor expressed in Ltk cellMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50301258BDBM50301258(1-benzyl-7-chloro-2-methyl-4,5-dihydro-1H-benzo[d]...)
Affinity DataKi:  930nMAssay Description:Displacement of [3H]SCH23390 from human D1 receptor expressed in Ltk cellMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50301270BDBM50301270(7-chloro-2-cyclopropyl-4,5-dihydro-1H-benzo[d][1,3...)
Affinity DataKi:  1.50E+3nMAssay Description:Displacement of [3H]SCH23390 from human D1 receptor expressed in Ltk cellMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50301271BDBM50301271(2-amino-7-chloro-4,5-dihydro-1H-benzo[d][1,3]diaze...)
Affinity DataKi:  1.02E+4nMAssay Description:Displacement of [3H]SCH23390 from human D1 receptor expressed in Ltk cellMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2010
Entry Details Article
PubMed