Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50030382
TargetCyclin-dependent kinase 5(Human)
Cnrs Usr-3151

Curated by ChEMBL
LigandPNGBDBM7377(CHEMBL75680 | aloisine A | 7-n-Butyl-6-(4-hydroxyp...)
Affinity DataIC50: 200nMAssay Description:Inhibition of GST-fused recombinant CDK5/p25 expressed in Escherichia coli after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5(Human)
Cnrs Usr-3151

Curated by ChEMBL
LigandPNGBDBM50295352(2-(2-{2-[4-(7-Butyl-5H-pyrrolo[2,3-b]pyrazin-6-yl)...)
Affinity DataIC50: 660nMAssay Description:Inhibition of GST-fused recombinant CDK5/p25 expressed in Escherichia coli after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Baker's yeast)
Cnrs Usr-3151

Curated by ChEMBL
LigandPNGBDBM7377(CHEMBL75680 | aloisine A | 7-n-Butyl-6-(4-hydroxyp...)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of hemagglutininin-tagged Saccharomyces cerevisiae MNY629 Cdc28/Clb2More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5(Human)
Cnrs Usr-3151

Curated by ChEMBL
LigandPNGBDBM50295354(2-(1-{2-[2-(2-Aminoethoxy)ethoxy]ethyl}-1H-[1,2,3]...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of GST-fused recombinant CDK5/p25 expressed in Escherichia coli after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5(Human)
Cnrs Usr-3151

Curated by ChEMBL
LigandPNGBDBM50295355(2-(1-{2-[2-(2-Aminoethoxy)ethoxy]ethyl}-1H-[1,2,3]...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of GST-fused recombinant CDK5/p25 expressed in Escherichia coli after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Baker's yeast)
Cnrs Usr-3151

Curated by ChEMBL
LigandPNGBDBM50295351(N-methyl-aloisine A | CHEMBL560452)
Affinity DataIC50: 3.30E+4nMAssay Description:Inhibition of hemagglutininin-tagged Saccharomyces cerevisiae MNY629 Cdc28/Clb2More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5(Human)
Cnrs Usr-3151

Curated by ChEMBL
LigandPNGBDBM50295353(2-(2-{2-[4-(7-Butyl-5-methyl-5H-pyrrolo[2,3-b]pyra...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of GST-fused recombinant CDK5/p25 expressed in Escherichia coli after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5(Human)
Cnrs Usr-3151

Curated by ChEMBL
LigandPNGBDBM50295351(N-methyl-aloisine A | CHEMBL560452)
Affinity DataIC50: 1.60E+5nMAssay Description:Inhibition of GST-fused recombinant CDK5/p25 expressed in Escherichia coli after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed