Compile Data Set for Download or QSAR
Report error Found 37 Enz. Inhib. hit(s) with all data for entry = 50030379
TargetNeuropeptide Y receptor type 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50423655(CHEMBL2307889)
Affinity DataIC50: 3.30nMAssay Description:Antagonist activity at human neuropeptide Y2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50140506((E)-N-(1-acetylindolin-6-yl)-3-(3-cyanophenyl)-N-(...)
Affinity DataIC50: 63.1nMAssay Description:Antagonist activity at human neuropeptide Y2 receptor by [35]GTPgammaS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50140506((E)-N-(1-acetylindolin-6-yl)-3-(3-cyanophenyl)-N-(...)
Affinity DataIC50: 100nMAssay Description:Binding affinity to neuropeptide Y2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50135642(N-(2-(benzylthio)phenyl)-N-(3-(dimethylamino)propy...)
Affinity DataIC50: 450nMAssay Description:Binding affinity to neuropeptide Y2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50414468(CHEMBL1196581 | CHEMBL557502)
Affinity DataIC50: 5.01E+4nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50414466(CHEMBL550583)
Affinity DataKi:  2.51nMAssay Description:Antagonist activity at human neuropeptide Y2 receptor in KAN-TS cells by [35]GTPgammaS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50414465(CHEMBL550559)
Affinity DataKi:  3.98nMAssay Description:Antagonist activity at human neuropeptide Y2 receptor in KAN-TS cells by [35]GTPgammaS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50414470(CHEMBL551311)
Affinity DataKi:  5.01nMAssay Description:Antagonist activity at human neuropeptide Y2 receptor in KAN-TS cells by [35]GTPgammaS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50414458(CHEMBL562725)
Affinity DataKi:  6.31nMAssay Description:Antagonist activity at human neuropeptide Y2 receptor in KAN-TS cells by [35]GTPgammaS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50414459(CHEMBL549771)
Affinity DataKi:  10nMAssay Description:Antagonist activity at human neuropeptide Y2 receptor in KAN-TS cells by [35]GTPgammaS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50414461(CHEMBL556481)
Affinity DataKi:  12.6nMAssay Description:Antagonist activity at human neuropeptide Y2 receptor in KAN-TS cells by [35]GTPgammaS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50414467(CHEMBL552112)
Affinity DataKi:  12.6nMAssay Description:Antagonist activity at human neuropeptide Y2 receptor in KAN-TS cells by [35]GTPgammaS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50414455(CHEMBL560914)
Affinity DataKi:  19.9nMAssay Description:Antagonist activity at human neuropeptide Y2 receptor in KAN-TS cells by [35]GTPgammaS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50414468(CHEMBL1196581 | CHEMBL557502)
Affinity DataKi:  25.1nMAssay Description:Antagonist activity at human neuropeptide Y2 receptor in KAN-TS cells by [35]GTPgammaS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50414453(CHEMBL563650)
Affinity DataKi:  50.1nMAssay Description:Antagonist activity at human neuropeptide Y2 receptor in KAN-TS cells by [35]GTPgammaS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50414472(CHEMBL561719)
Affinity DataKi:  63.1nMAssay Description:Antagonist activity at human neuropeptide Y2 receptor in KAN-TS cells by [35]GTPgammaS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50414469(CHEMBL549565)
Affinity DataKi:  79.4nMAssay Description:Antagonist activity at human neuropeptide Y2 receptor in KAN-TS cells by [35]GTPgammaS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50414449(CHEMBL563568)
Affinity DataKi:  79.4nMAssay Description:Antagonist activity at human neuropeptide Y2 receptor in KAN-TS cells by [35]GTPgammaS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50414450(CHEMBL549895)
Affinity DataKi:  126nMAssay Description:Antagonist activity at human neuropeptide Y2 receptor in KAN-TS cells by [35]GTPgammaS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50414451(CHEMBL560716)
Affinity DataKi:  158nMAssay Description:Antagonist activity at human neuropeptide Y2 receptor in KAN-TS cells by [35]GTPgammaS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50414454(CHEMBL550504)
Affinity DataKi:  158nMAssay Description:Antagonist activity at human neuropeptide Y2 receptor in KAN-TS cells by [35]GTPgammaS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50414447(CHEMBL560117)
Affinity DataKi:  200nMAssay Description:Antagonist activity at human neuropeptide Y2 receptor in KAN-TS cells by [35]GTPgammaS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50414448(CHEMBL564159)
Affinity DataKi:  316nMAssay Description:Antagonist activity at human neuropeptide Y2 receptor in KAN-TS cells by [35]GTPgammaS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50414462(CHEMBL562179)
Affinity DataKi:  316nMAssay Description:Antagonist activity at human neuropeptide Y2 receptor in KAN-TS cells by [35]GTPgammaS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50414460(CHEMBL561313)
Affinity DataKi:  316nMAssay Description:Antagonist activity at human neuropeptide Y2 receptor in KAN-TS cells by [35]GTPgammaS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50414456(CHEMBL561577)
Affinity DataKi:  316nMAssay Description:Antagonist activity at human neuropeptide Y2 receptor in KAN-TS cells by [35]GTPgammaS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50414446(CHEMBL539730)
Affinity DataKi:  501nMAssay Description:Antagonist activity at human neuropeptide Y2 receptor in KAN-TS cells by [35]GTPgammaS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50414471(CHEMBL563037)
Affinity DataKi:  631nMAssay Description:Antagonist activity at human neuropeptide Y2 receptor in KAN-TS cells by [35]GTPgammaS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50414464(CHEMBL551715)
Affinity DataKi:  1.58E+3nMAssay Description:Antagonist activity at human neuropeptide Y2 receptor in KAN-TS cells by [35]GTPgammaS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50414463(CHEMBL557098)
Affinity DataKi:  2.51E+3nMAssay Description:Antagonist activity at human neuropeptide Y2 receptor in KAN-TS cells by [35]GTPgammaS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50414452(CHEMBL552393)
Affinity DataKi:  2.51E+3nMAssay Description:Antagonist activity at human neuropeptide Y2 receptor in KAN-TS cells by [35]GTPgammaS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50414473(CHEMBL549976)
Affinity DataKi:  3.16E+3nMAssay Description:Antagonist activity at human neuropeptide Y2 receptor in KAN-TS cells by [35]GTPgammaS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50414446(CHEMBL539730)
Affinity DataKi: >5.01E+3nMAssay Description:Antagonist activity at human neuropeptide Y5 receptor expressed in HEK293 cells by FLIPR/Ca2+ methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50414446(CHEMBL539730)
Affinity DataKi: >6.31E+3nMAssay Description:Antagonist activity at human neuropeptide Y1 receptor expressed in CHO cells by [35]GTPgammaS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50414468(CHEMBL1196581 | CHEMBL557502)
Affinity DataKi: >6.31E+3nMAssay Description:Antagonist activity at human neuropeptide Y1 receptor expressed in CHO cells by [35]GTPgammaS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50414457(CHEMBL559662)
Affinity DataKi: >6.31E+3nMAssay Description:Antagonist activity at human neuropeptide Y2 receptor in KAN-TS cells by [35]GTPgammaS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50414468(CHEMBL1196581 | CHEMBL557502)
Affinity DataKi: >1.00E+4nMAssay Description:Antagonist activity at human neuropeptide Y5 receptor expressed in HEK293 cells by FLIPR/Ca2+ methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed