Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 50004254
TargetIntegrase(Human immunodeficiency virus type 1)
Facult£S Universitaires Notre-Dame De La Paix

Curated by ChEMBL
LigandPNGBDBM50184349((Z)-4-[6-((Z)-3-carboxy-3-hydroxy-acryloyl)-1-(4-f...)
Affinity DataIC50: 17nMAssay Description:Inhibition of HIV1 integrase strand transfer activity expressed in Escherichia coli BL21 (DE3) by gel based assay in presence of magnesiumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Facult£S Universitaires Notre-Dame De La Paix

Curated by ChEMBL
LigandPNGBDBM50480767(CHEMBL562899)
Affinity DataIC50: 30nMAssay Description:Inhibition of HIV1 integrase strand transfer activity expressed in Escherichia coli BL21 (DE3) by gel based assay in presence of magnesiumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Facult£S Universitaires Notre-Dame De La Paix

Curated by ChEMBL
LigandPNGBDBM50480768(CHEMBL559753)
Affinity DataIC50: 120nMAssay Description:Inhibition of HIV1 integrase strand transfer activity expressed in Escherichia coli BL21 (DE3) by gel based assay in presence of magnesiumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Facult£S Universitaires Notre-Dame De La Paix

Curated by ChEMBL
LigandPNGBDBM50184349((Z)-4-[6-((Z)-3-carboxy-3-hydroxy-acryloyl)-1-(4-f...)
Affinity DataIC50: 440nMAssay Description:Inhibition of HIV1 integrase 3'-processing activity expressed in Escherichia coli BL21 (DE3) by gel based assay in presence of magnesiumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Facult£S Universitaires Notre-Dame De La Paix

Curated by ChEMBL
LigandPNGBDBM50480767(CHEMBL562899)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of HIV1 integrase 3'-processing activity expressed in Escherichia coli BL21 (DE3) by gel based assay in presence of magnesiumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Facult£S Universitaires Notre-Dame De La Paix

Curated by ChEMBL
LigandPNGBDBM50480768(CHEMBL559753)
Affinity DataIC50: 7.80E+4nMAssay Description:Inhibition of HIV1 integrase 3'-processing activity expressed in Escherichia coli BL21 (DE3) by gel based assay in presence of magnesiumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed