Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50028764
TargetProtein kinase C delta type(Human)
University of Helsinki

Curated by ChEMBL
LigandPNGBDBM50258529(CHEMBL449158 | bryostatin 1)
Affinity DataKi:  0.440nMAssay Description:Displacement of [3H]PDBu from human recombinant PKCdelta expressed in Sf9 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Human)
University of Helsinki

Curated by ChEMBL
LigandPNGBDBM50015677(CHEMBL55267 | 1,2-dioctanoyl-sn-glycerol | 1,2-Dio...)
Affinity DataKi:  40nMAssay Description:Displacement of [3H]PDBu from human recombinant PKCalpha expressed in Sf9 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Human)
University of Helsinki

Curated by ChEMBL
LigandPNGBDBM50258472(bis(3-(trifluoromethyl)benzyl)5-(hydroxymethyl)iso...)
Affinity DataKi:  205nMAssay Description:Displacement of [3H]PDBu from human recombinant PKCalpha expressed in Sf9 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Human)
University of Helsinki

Curated by ChEMBL
LigandPNGBDBM50258322(diheptan-3-yl 5-(hydroxymethyl)isophthalate | CHEM...)
Affinity DataKi:  319nMAssay Description:Displacement of [3H]PDBu from human recombinant PKCalpha expressed in Sf9 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
University of Helsinki

Curated by ChEMBL
LigandPNGBDBM50258322(diheptan-3-yl 5-(hydroxymethyl)isophthalate | CHEM...)
Affinity DataKi:  529nMAssay Description:Displacement of [3H]PDBu from human recombinant PKCdelta expressed in Sf9 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
University of Helsinki

Curated by ChEMBL
LigandPNGBDBM50258472(bis(3-(trifluoromethyl)benzyl)5-(hydroxymethyl)iso...)
Affinity DataKi:  590nMAssay Description:Displacement of [3H]PDBu from human recombinant PKCdelta expressed in Sf9 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Human)
University of Helsinki

Curated by ChEMBL
LigandPNGBDBM50258321(dihexan-3-yl 5-(hydroxymethyl)isophthalate | CHEMB...)
Affinity DataKi:  661nMAssay Description:Displacement of [3H]PDBu from human recombinant PKCalpha expressed in Sf9 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
University of Helsinki

Curated by ChEMBL
LigandPNGBDBM50258321(dihexan-3-yl 5-(hydroxymethyl)isophthalate | CHEMB...)
Affinity DataKi:  915nMAssay Description:Displacement of [3H]PDBu from human recombinant PKCdelta expressed in Sf9 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed