Compile Data Set for Download or QSAR
Report error Found 28 Enz. Inhib. hit(s) with all data for entry = 50028737
TargetHistone deacetylase 6(Human)
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM19149(Zolinza | suberoylanilide hydroxamic acid | CHEMBL...)
Affinity DataIC50: 28nMAssay Description:Inhibition of human recombinant HDAC6 by fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetHistone deacetylase 6(Human)
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50250101((S)-7-(Biphenyl-3-ylamino)-7-oxo-6-(thiazole-5-car...)
Affinity DataIC50: 110nMAssay Description:Inhibition of human recombinant HDAC6 by fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetHistone deacetylase 2(Human)
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM19149(Zolinza | suberoylanilide hydroxamic acid | CHEMBL...)
Affinity DataIC50: 250nMAssay Description:Inhibition of human recombinant HDAC2 by fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetHistone deacetylase 6(Human)
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50250099((S)-7-(Biphenyl-3-ylamino)-7-oxo-6-(pyridine-3-car...)
Affinity DataIC50: 320nMAssay Description:Inhibition of human recombinant HDAC6 by fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM19149(Zolinza | suberoylanilide hydroxamic acid | CHEMBL...)
Affinity DataIC50: 350nMAssay Description:Inhibition of human recombinant HDAC1 by fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetHistone deacetylase 2(Human)
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50250101((S)-7-(Biphenyl-3-ylamino)-7-oxo-6-(thiazole-5-car...)
Affinity DataIC50: 530nMAssay Description:Inhibition of human recombinant HDAC2 by fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetHistone deacetylase 2(Human)
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50250099((S)-7-(Biphenyl-3-ylamino)-7-oxo-6-(pyridine-3-car...)
Affinity DataIC50: 830nMAssay Description:Inhibition of human recombinant HDAC2 by fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetHistone deacetylase 6(Human)
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50249973((S)-6-(Benzenecarbonylamino)-7-(biphenyl-3-ylamino...)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of human recombinant HDAC6 by fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetHistone deacetylase 8(Human)
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM19149(Zolinza | suberoylanilide hydroxamic acid | CHEMBL...)
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of human recombinant HDAC8 by fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetHistone deacetylase 1(Human)
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50250101((S)-7-(Biphenyl-3-ylamino)-7-oxo-6-(thiazole-5-car...)
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of human recombinant HDAC1 by fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50250099((S)-7-(Biphenyl-3-ylamino)-7-oxo-6-(pyridine-3-car...)
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibition of human recombinant HDAC1 by fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetHistone deacetylase 2(Human)
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50249973((S)-6-(Benzenecarbonylamino)-7-(biphenyl-3-ylamino...)
Affinity DataIC50: 3.60E+3nMAssay Description:Inhibition of human recombinant HDAC2 by fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetHistone deacetylase 6(Human)
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50250151((R)-7-(Biphenyl-3-ylamino)-7-oxo-6-(thiazole-5-car...)
Affinity DataIC50: 5.60E+3nMAssay Description:Inhibition of human recombinant HDAC6 by fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetHistone deacetylase 8(Human)
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50250101((S)-7-(Biphenyl-3-ylamino)-7-oxo-6-(thiazole-5-car...)
Affinity DataIC50: 6.60E+3nMAssay Description:Inhibition of human recombinant HDAC8 by fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50249973((S)-6-(Benzenecarbonylamino)-7-(biphenyl-3-ylamino...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant HDAC1 by fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetHistone deacetylase 6(Human)
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50250100((R)-7-(Biphenyl-3-ylamino)-7-oxo-6-(pyridine-3-car...)
Affinity DataIC50: 1.40E+4nMAssay Description:Inhibition of human recombinant HDAC6 by fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetHistone deacetylase 8(Human)
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50250099((S)-7-(Biphenyl-3-ylamino)-7-oxo-6-(pyridine-3-car...)
Affinity DataIC50: 2.30E+4nMAssay Description:Inhibition of human recombinant HDAC8 by fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetHistone deacetylase 6(Human)
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50250098((R)-6-(Benzenecarbonylamino)-7-(biphenyl-3-ylamino...)
Affinity DataIC50: 2.40E+4nMAssay Description:Inhibition of human recombinant HDAC6 by fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetHistone deacetylase 2(Human)
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50250100((R)-7-(Biphenyl-3-ylamino)-7-oxo-6-(pyridine-3-car...)
Affinity DataIC50: 9.90E+4nMAssay Description:Inhibition of human recombinant HDAC2 by fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetHistone deacetylase 8(Human)
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50249973((S)-6-(Benzenecarbonylamino)-7-(biphenyl-3-ylamino...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human recombinant HDAC8 by fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50250098((R)-6-(Benzenecarbonylamino)-7-(biphenyl-3-ylamino...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human recombinant HDAC1 by fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetHistone deacetylase 2(Human)
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50250098((R)-6-(Benzenecarbonylamino)-7-(biphenyl-3-ylamino...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human recombinant HDAC2 by fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetHistone deacetylase 8(Human)
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50250098((R)-6-(Benzenecarbonylamino)-7-(biphenyl-3-ylamino...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human recombinant HDAC8 by fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50250100((R)-7-(Biphenyl-3-ylamino)-7-oxo-6-(pyridine-3-car...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human recombinant HDAC1 by fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetHistone deacetylase 8(Human)
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50250100((R)-7-(Biphenyl-3-ylamino)-7-oxo-6-(pyridine-3-car...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human recombinant HDAC8 by fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50250151((R)-7-(Biphenyl-3-ylamino)-7-oxo-6-(thiazole-5-car...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human recombinant HDAC1 by fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetHistone deacetylase 2(Human)
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50250151((R)-7-(Biphenyl-3-ylamino)-7-oxo-6-(thiazole-5-car...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human recombinant HDAC2 by fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetHistone deacetylase 8(Human)
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50250151((R)-7-(Biphenyl-3-ylamino)-7-oxo-6-(thiazole-5-car...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human recombinant HDAC8 by fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed