Compile Data Set for Download or QSAR
Report error Found 24 Enz. Inhib. hit(s) with all data for entry = 50028692
LigandPNGBDBM50258540(N-((7R,8R)-7-hydroxy-8-(4-pentylphenylsulfonamido)...)
Affinity DataIC50: 70nMAssay Description:Inhibition of human Kv1.5 channel expressed in mouse L929 cells by patch-clamp electrophysiology methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50258501(N-((7R,8R)-7-hydroxy-8-(4-propylphenylsulfonamido)...)
Affinity DataIC50: 90nMAssay Description:Inhibition of human Kv1.5 channel expressed in mouse L929 cells by patch-clamp electrophysiology methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50240481(N-((7R,8R)-8-(4-butylphenylsulfonamido)-7-hydroxy-...)
Affinity DataIC50: 140nMAssay Description:Inhibition of human Kv1.5 channel expressed in mouse L929 cells by patch-clamp electrophysiology methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50099581(N-[3-(4-Ethyl-benzenesulfonylamino)-2-hydroxy-inda...)
Affinity DataIC50: 160nMAssay Description:Inhibition of human Kv1.5 channel expressed in mouse L929 cells by patch-clamp electrophysiology methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50258503(N-((7R,8R)-8-(4-tert-butylphenylsulfonamido)-7-hyd...)
Affinity DataIC50: 160nMAssay Description:Inhibition of human Kv1.5 channel expressed in mouse L929 cells by patch-clamp electrophysiology methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50258755(N-((7R,8R)-8-(4-ethylphenylsulfonamido)-7-hydroxy-...)
Affinity DataIC50: 200nMAssay Description:Inhibition of human Kv1.5 channel expressed in mouse L929 cells by patch-clamp electrophysiology methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50258410((R)-1-(3-chlorobenzyl)-N-((7R,8R)-8-(4-ethylphenyl...)
Affinity DataIC50: 220nMAssay Description:Inhibition of human Kv1.5 channel expressed in mouse L929 cells by patch-clamp electrophysiology methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50258758(benzyl (7R,8R)-8-(4-ethylphenylsulfonamido)-7-hydr...)
Affinity DataIC50: 230nMAssay Description:Inhibition of human Kv1.5 channel expressed in mouse L929 cells by patch-clamp electrophysiology methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50258728(N-((7R,8R)-8-(4-ethylphenylsulfonamido)-7-hydroxy-...)
Affinity DataIC50: 250nMAssay Description:Inhibition of human Kv1.5 channel expressed in mouse L929 cells by patch-clamp electrophysiology methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50258801((S)-N-(8-(4-ethylphenylsulfonamido)-5,6,7,8-tetrah...)
Affinity DataIC50: 280nMAssay Description:Inhibition of human Kv1.5 channel expressed in mouse L929 cells by patch-clamp electrophysiology methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50258411((R)-N-((7R,8R)-8-(4-ethylphenylsulfonamido)-7-hydr...)
Affinity DataIC50: 290nMAssay Description:Inhibition of human Kv1.5 channel expressed in mouse L929 cells by patch-clamp electrophysiology methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50258412((R)-N-((7R,8R)-8-(4-ethylphenylsulfonamido)-7-hydr...)
Affinity DataIC50: 300nMAssay Description:Inhibition of human Kv1.5 channel expressed in mouse L929 cells by patch-clamp electrophysiology methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50258702(4-chloro-N-((7R,8R)-8-(4-ethylphenylsulfonamido)-7...)
Affinity DataIC50: 340nMAssay Description:Inhibition of human Kv1.5 channel expressed in mouse L929 cells by patch-clamp electrophysiology methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50258757((1S,2S)-N-((7R,8R)-8-(4-ethylphenylsulfonamido)-7-...)
Affinity DataIC50: 350nMAssay Description:Inhibition of human Kv1.5 channel expressed in mouse L929 cells by patch-clamp electrophysiology methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50258502(N-((7R,8R)-7-hydroxy-8-(4-isopropylphenylsulfonami...)
Affinity DataIC50: 430nMAssay Description:Inhibition of human Kv1.5 channel expressed in mouse L929 cells by patch-clamp electrophysiology methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50258756(N-((7R,8R)-8-(4-ethylphenylsulfonamido)-7-hydroxy-...)
Affinity DataIC50: 430nMAssay Description:Inhibition of human Kv1.5 channel expressed in mouse L929 cells by patch-clamp electrophysiology methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50207907(N-((7R,8R)-8-(4-ethylphenylsulfonamido)-7-hydroxy-...)
Affinity DataIC50: 440nMAssay Description:Inhibition of human Kv1.5 channel expressed in mouse L929 cells by patch-clamp electrophysiology methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50258671(N-((7R,8R)-8-(4-ethylphenylsulfonamido)-7-hydroxy-...)
Affinity DataIC50: 450nMAssay Description:Inhibition of human Kv1.5 channel expressed in mouse L929 cells by patch-clamp electrophysiology methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50258670(N-((7R,8R)-8-(4-ethylphenylsulfonamido)-7-hydroxy-...)
Affinity DataIC50: 450nMAssay Description:Inhibition of human Kv1.5 channel expressed in mouse L929 cells by patch-clamp electrophysiology methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50258800((S)-N-(8-(4-ethylphenylsulfonamido)-5,6,7,8-tetrah...)
Affinity DataIC50: 590nMAssay Description:Inhibition of human Kv1.5 channel expressed in mouse L929 cells by patch-clamp electrophysiology methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50258799(N-((1R,2R)-7-(3-benzylureido)-2-hydroxy-1,2,3,4-te...)
Affinity DataIC50: 610nMAssay Description:Inhibition of human Kv1.5 channel expressed in mouse L929 cells by patch-clamp electrophysiology methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50258703(N-((7R,8R)-8-(4-ethylphenylsulfonamido)-7-hydroxy-...)
Affinity DataIC50: 640nMAssay Description:Inhibition of human Kv1.5 channel expressed in mouse L929 cells by patch-clamp electrophysiology methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50258701(3-chloro-N-((7R,8R)-8-(4-ethylphenylsulfonamido)-7...)
Affinity DataIC50: 710nMAssay Description:Inhibition of human Kv1.5 channel expressed in mouse L929 cells by patch-clamp electrophysiology methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandPNGBDBM50258580(N-((7R,8R)-7-hydroxy-8-(4-methoxyphenylsulfonamido...)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of human Kv1.5 channel expressed in mouse L929 cells by patch-clamp electrophysiology methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed