Compile Data Set for Download or QSAR
Report error Found 14 Enz. Inhib. hit(s) with all data for entry = 50030527
TargetEstrogen receptor(Human)
University of Illinois

Curated by ChEMBL
LigandPNGBDBM50297518(trans-6-[1-ethyl-2-(4-hydroxy-phenyl)-butyl]-pyrid...)
Affinity DataEC50:  0.110nMAssay Description:Activity at human ERalpha expressed in HEC1 cells co-transfected with 2ERE-pS2-Luc assessed as relative transcriptional potency by luciferase reporte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
University of Illinois

Curated by ChEMBL
LigandPNGBDBM50297516(trans-6-[1-ethyl-2-(4-hydroxy-phenyl)-propyl]-pyri...)
Affinity DataEC50:  0.110nMAssay Description:Activity at human ERalpha expressed in HEC1 cells co-transfected with 2ERE-pS2-Luc assessed as relative transcriptional potency by luciferase reporte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
University of Illinois

Curated by ChEMBL
LigandPNGBDBM50297518(trans-6-[1-ethyl-2-(4-hydroxy-phenyl)-butyl]-pyrid...)
Affinity DataEC50:  0.610nMAssay Description:Activity at human ERbeta expressed in HEC1 cells co-transfected with 2ERE-pS2-Luc assessed as relative transcriptional potency by luciferase reporter...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
University of Illinois

Curated by ChEMBL
LigandPNGBDBM50297516(trans-6-[1-ethyl-2-(4-hydroxy-phenyl)-propyl]-pyri...)
Affinity DataEC50:  1.10nMAssay Description:Activity at human ERbeta expressed in HEC1 cells co-transfected with 2ERE-pS2-Luc assessed as relative transcriptional potency by luciferase reporter...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
University of Illinois

Curated by ChEMBL
LigandPNGBDBM50297519(4,4'-(propane-1,2-diyl)diphenol | (+/-)-1,2-Bis-(4...)
Affinity DataEC50:  1.20nMAssay Description:Activity at human ERbeta expressed in HEC1 cells co-transfected with 2ERE-pS2-Luc assessed as relative transcriptional potency by luciferase reporter...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
University of Illinois

Curated by ChEMBL
LigandPNGBDBM50297519(4,4'-(propane-1,2-diyl)diphenol | (+/-)-1,2-Bis-(4...)
Affinity DataEC50:  6.5nMAssay Description:Activity at human ERalpha expressed in HEC1 cells co-transfected with 2ERE-pS2-Luc assessed as relative transcriptional potency by luciferase reporte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
University of Illinois

Curated by ChEMBL
LigandPNGBDBM50297517(cis-6-[1-ethyl-2-(4-hydroxy-phenyl)-butyl]-pyridin...)
Affinity DataEC50:  16nMAssay Description:Activity at human ERalpha expressed in HEC1 cells co-transfected with 2ERE-pS2-Luc assessed as relative transcriptional potency by luciferase reporte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
University of Illinois

Curated by ChEMBL
LigandPNGBDBM50297514(6-[1-(4-Hydroxy-benzyl)-propyl]-pyridin-3-ol | CHE...)
Affinity DataEC50:  17nMAssay Description:Activity at human ERbeta expressed in HEC1 cells co-transfected with 2ERE-pS2-Luc assessed as relative transcriptional potency by luciferase reporter...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
University of Illinois

Curated by ChEMBL
LigandPNGBDBM50297517(cis-6-[1-ethyl-2-(4-hydroxy-phenyl)-butyl]-pyridin...)
Affinity DataEC50:  26nMAssay Description:Activity at human ERbeta expressed in HEC1 cells co-transfected with 2ERE-pS2-Luc assessed as relative transcriptional potency by luciferase reporter...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
University of Illinois

Curated by ChEMBL
LigandPNGBDBM50297513(6-[2-(4-Hydroxy-phenyl)-1-methyl-ethyl]-pyridin-3-...)
Affinity DataEC50:  60nMAssay Description:Activity at human ERbeta expressed in HEC1 cells co-transfected with 2ERE-pS2-Luc assessed as relative transcriptional potency by luciferase reporter...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
University of Illinois

Curated by ChEMBL
LigandPNGBDBM50297514(6-[1-(4-Hydroxy-benzyl)-propyl]-pyridin-3-ol | CHE...)
Affinity DataEC50:  65nMAssay Description:Activity at human ERalpha expressed in HEC1 cells co-transfected with 2ERE-pS2-Luc assessed as relative transcriptional potency by luciferase reporte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetEstrogen receptor beta(Human)
University of Illinois

Curated by ChEMBL
LigandPNGBDBM50297515(6-[2-(4-Hydroxy-phenyl)-propyl]-pyridin-3-ol | CHE...)
Affinity DataEC50:  170nMAssay Description:Activity at human ERbeta expressed in HEC1 cells co-transfected with 2ERE-pS2-Luc assessed as relative transcriptional potency by luciferase reporter...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
University of Illinois

Curated by ChEMBL
LigandPNGBDBM50297513(6-[2-(4-Hydroxy-phenyl)-1-methyl-ethyl]-pyridin-3-...)
Affinity DataEC50:  330nMAssay Description:Activity at human ERalpha expressed in HEC1 cells co-transfected with 2ERE-pS2-Luc assessed as relative transcriptional potency by luciferase reporte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
University of Illinois

Curated by ChEMBL
LigandPNGBDBM50297515(6-[2-(4-Hydroxy-phenyl)-propyl]-pyridin-3-ol | CHE...)
Affinity DataEC50:  440nMAssay Description:Activity at human ERalpha expressed in HEC1 cells co-transfected with 2ERE-pS2-Luc assessed as relative transcriptional potency by luciferase reporte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed