Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 50028604
TargetBeta-secretase 1(Human)
Kyoto Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50277598(N-((2S,3S)-4-(3-(2H-tetrazol-5-yl)phenylamino)-3-h...)
Affinity DataIC50: 9nMAssay Description:Inhibition of human recombinant Arg235 region of BACE1 by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Kyoto Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50277599(N-((2S,3S)-4-(3-(2H-tetrazol-5-yl)phenylamino)-3-h...)
Affinity DataIC50: 10nMAssay Description:Inhibition of human recombinant Arg235 region of BACE1 by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Kyoto Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50277597(N-((2S,3S)-4-(3-(2H-tetrazol-5-yl)phenylamino)-3-h...)
Affinity DataIC50: 13nMAssay Description:Inhibition of human recombinant Arg235 region of BACE1 by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Kyoto Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50277595(N-((2S,3S)-4-(3-(2H-tetrazol-5-yl)phenylamino)-3-h...)
Affinity DataIC50: 15nMAssay Description:Inhibition of human recombinant Arg235 region of BACE1 by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Kyoto Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50277594(N-((2S,3S)-4-(3-(2H-tetrazol-5-yl)phenylamino)-3-h...)
Affinity DataIC50: 22nMAssay Description:Inhibition of human recombinant Arg235 region of BACE1 by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Kyoto Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50277596(N-((2S,3S)-4-(3-(2H-tetrazol-5-yl)phenylamino)-3-h...)
Affinity DataIC50: 24nMAssay Description:Inhibition of human recombinant Arg235 region of BACE1 by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Kyoto Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50234644(N-((2S,3S)-4-(3-(2H-tetrazol-5-yl)phenylamino)-3-h...)
Affinity DataIC50: 50nMAssay Description:Inhibition of human recombinant Arg235 region of BACE1 by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Kyoto Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50234646(2-(((2S,3S)-4-(3-(2H-tetrazol-5-yl)phenylamino)-3-...)
Affinity DataIC50: 96nMAssay Description:Inhibition of human recombinant Arg235 region of BACE1 by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Kyoto Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50234643(N-((2S,3S)-4-(3-(2H-tetrazol-5-yl)phenylamino)-3-h...)
Affinity DataIC50: 140nMAssay Description:Inhibition of human recombinant Arg235 region of BACE1 by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Kyoto Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50234645(N-((2S,3S)-4-(3-(2H-tetrazol-5-yl)phenylamino)-3-h...)
Affinity DataIC50: 360nMAssay Description:Inhibition of human recombinant Arg235 region of BACE1 by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed