Compile Data Set for Download or QSAR
Report error Found 104 Enz. Inhib. hit(s) with all data for entry = 50028587
TargetGlycogen synthase kinase-3 beta(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50267760(3-Benzofuran-3-yl-4-(7-methoxymethyl-1-methyl-1H-i...)
Affinity DataIC50: 0.230nMAssay Description:Inhibition of human GSK3-beta by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50267461(3-(5-Fluoro-1-methyl-1H-indol-3-yl)-4-(6-hydroxyme...)
Affinity DataIC50: 0.350nMAssay Description:Inhibition of human GSK3-beta by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Chk1(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of CHK1More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50267607(3-(5-Bromo-1-methyl-1H-indol-3-yl)-4-(6-hydroxymet...)
Affinity DataIC50: 0.510nMAssay Description:Inhibition of human GSK3-beta by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetRAC-gamma serine/threonine-protein kinase(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 0.640nMAssay Description:Inhibition of AKT3More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50267800(3-(6-Hydroxymethylbenzofuran-3-yl)-4-(7-methoxymet...)
Affinity DataIC50: 0.730nMAssay Description:Inhibition of human GSK3-beta by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50267523(3-(6-Chloro-5-fluoro-1-methyl-1H-indol-3-yl)-4-(6-...)
Affinity DataIC50: 0.950nMAssay Description:Inhibition of human GSK3-beta by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50267802(3-[3-(4-Benzofuran-3-yl-2,5-dioxo-2,5-dihydro-1H-p...)
Affinity DataIC50: 1.20nMAssay Description:Inhibition of human GSK3-beta by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 1.40nMAssay Description:Inhibition of CDK2/Cyclin AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 9(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 3.30nMAssay Description:Inhibition of CDK9/cyclin T1More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 3.30nMAssay Description:Inhibition of CDK1/Cyclin BMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50267520(3-(5-Fluoro-1-methyl-1H-indol-3-yl)-4-(6-hydroxybe...)
Affinity DataIC50: 3.5nMAssay Description:Inhibition of human GSK3-beta by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 3.80nMAssay Description:Inhibition of CDK5/P35More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 3.80nMAssay Description:Inhibition of CDK2/Cyclin EMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 4nMAssay Description:Inhibition of CDK5/P25More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50267759(3-(6-Hydroxymethylbenzofuran-3-yl)-4-(7-hydroxymet...)
Affinity DataIC50: 5.10nMAssay Description:Inhibition of human GSK3-beta by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50267758(3-Benzofuran-3-yl-4-(7-hydroxymethyl-1-methyl-1H-i...)
Affinity DataIC50: 5.40nMAssay Description:Inhibition of human GSK3-beta by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 3(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 6.90nMAssay Description:Inhibition of CDK3/Cyclin EMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50267605(3-(benzofuran-3-yl)-4-(5-bromo-1-methyl-1H-indol-3...)
Affinity DataIC50: 7nMAssay Description:Inhibition of human GSK3-beta by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50267606(3-(5-Bromo-1-methyl-1H-indol-3-yl)-4-(7-methoxyben...)
Affinity DataIC50: 7.5nMAssay Description:Inhibition of human GSK3-beta by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50267801(3-[3-(4-Benzofuran-3-yl-2,5-dioxo-2,5-dihydro-1H-p...)
Affinity DataIC50: 10nMAssay Description:Inhibition of human GSK3-beta by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50267678(3-[4-(6-Hydroxymethylbenzofuran-3-yl)-2,5-dioxo-2,...)
Affinity DataIC50: 13nMAssay Description:Inhibition of human GSK3-beta by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50267367(3-(benzofuran-3-yl)-4-(6-hydroxy-1-methyl-1H-indol...)
Affinity DataIC50: 15nMAssay Description:Inhibition of human GSK3-beta by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50267715(3-(5-Cyclopropylethynyl-1-methyl-1H-indol-3-yl)-4-...)
Affinity DataIC50: 16nMAssay Description:Inhibition of human GSK3-beta by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 4(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 18nMAssay Description:Inhibition of CDK4/Cyclin D1More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50267462(3-(5-Fluoro-1-methyl-1H-indol-3-yl)-4-(6-methoxyme...)
Affinity DataIC50: 24nMAssay Description:Inhibition of human GSK3-beta by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50267639(3-(5-Bromo-1-methyl-1H-indol-3-yl)-4-(6-prop-2-yny...)
Affinity DataIC50: 25nMAssay Description:Inhibition of human GSK3-beta by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50267759(3-(6-Hydroxymethylbenzofuran-3-yl)-4-(7-hydroxymet...)
Affinity DataIC50: 27nMAssay Description:Inhibition of CDK2/Cyclin EMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM2600(3-(1-benzofuran-3-yl)-4-(1-methyl-1H-indol-3-yl)-2...)
Affinity DataIC50: 35nMAssay Description:Inhibition of human GSK3-beta by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50267676(3-Benzofuran-3-yl-4-(5-iodo-1-methyl-1H-indol-3-yl...)
Affinity DataIC50: 35nMAssay Description:Inhibition of human GSK3-beta by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50229962(N-(4-METHOXYBENZYL)-N'-(5-NITRO-1,3-THIAZOL-2-YL)U...)
Affinity DataIC50: 42nMAssay Description:Inhibition of human GSK3-beta by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetGlycogen synthase kinase-3 beta(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50267642(3-(5-chloro-1-methyl-1H-indol-3-yl)-4-(5-fluoroben...)
Affinity DataIC50: 42nMAssay Description:Inhibition of human GSK3-beta by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50267640(3-(6-Allyloxybenzofuran-3-yl)-4-(5-bromo-1-methyl-...)
Affinity DataIC50: 48nMAssay Description:Inhibition of human GSK3-beta by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM8296(CHEMBL102714 | cid_176158 | 3-(2,4-dichlorophenyl)...)
Affinity DataIC50: 50nMAssay Description:Inhibition of human GSK3-beta by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50267803(3-(benzofuran-3-yl)-4-(7-hydroxy-1-methyl-1H-indol...)
Affinity DataIC50: 55nMAssay Description:Inhibition of human GSK3-beta by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50267675(3-(5,7-Dibromo-1-methyl-1H-indol-3-yl)-4-(7-methox...)
Affinity DataIC50: 89nMAssay Description:Inhibition of human GSK3-beta by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 6(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 116nMAssay Description:Inhibition of CDK6/cyclin D3More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50267758(3-Benzofuran-3-yl-4-(7-hydroxymethyl-1-methyl-1H-i...)
Affinity DataIC50: 149nMAssay Description:Inhibition of CDK2/Cyclin EMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50267677(3-(5-Fluorobenzofuran-3-yl)-4-(5-iodo-1-methyl-1H-...)
Affinity DataIC50: 180nMAssay Description:Inhibition of human GSK3-beta by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50267522(3-Benzofuran-3-yl-4-(6-chloro-5-fluoro-1-methyl-1H...)
Affinity DataIC50: 184nMAssay Description:Inhibition of human GSK3-beta by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50267718(3-Benzofuran-3-yl-4-(6-iodo-5-methoxy-1-methyl-1H-...)
Affinity DataIC50: 223nMAssay Description:Inhibition of human GSK3-beta by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit alpha(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 233nMAssay Description:Inhibition of IKKalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50267679(3-(benzofuran-3-yl)-4-(5-cyclopropyl-1-methyl-1H-i...)
Affinity DataIC50: 235nMAssay Description:Inhibition of human GSK3-beta by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50267461(3-(5-Fluoro-1-methyl-1H-indol-3-yl)-4-(6-hydroxyme...)
Affinity DataIC50: 237nMAssay Description:Inhibition of CDK2/Cyclin EMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50267521(3-(5-Fluoro-6-iodo-1-methyl-1H-indol-3-yl)-4-(7-me...)
Affinity DataIC50: 247nMAssay Description:Inhibition of human GSK3-beta by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetGlycogen synthase kinase-3 beta(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50267565(3-(6-Chloro-5-fluoro-1-methyl-1H-indol-3-yl)-4-(7-...)
Affinity DataIC50: 260nMAssay Description:Inhibition of human GSK3-beta by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50267845(3-(5,6-Difluorobenzofuran-3-yl)-4-(1-methyl-1H-ben...)
Affinity DataIC50: 314nMAssay Description:Inhibition of human GSK3-beta by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50267641(3-(5-Bromo-1-methyl-1H-indol-3-yl)-4-[6-(4-methoxy...)
Affinity DataIC50: 335nMAssay Description:Inhibition of human GSK3-beta by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 2(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50267607(3-(5-Bromo-1-methyl-1H-indol-3-yl)-4-(6-hydroxymet...)
Affinity DataIC50: 337nMAssay Description:Inhibition of CDK2/Cyclin EMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50267717(3-Benzofuran-3-yl-4-(6-chloro-5-methoxy-1-methyl-1...)
Affinity DataIC50: 440nMAssay Description:Inhibition of human GSK3-beta by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
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