Compile Data Set for Download or QSAR
Report error Found 55 Enz. Inhib. hit(s) with all data for entry = 50028494
TargetAdenosine receptor A3(Human)
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM50257074(N-(2-(4-methoxyphenyl)-1-oxo-1,2-dihydropyrido[2,3...)
Affinity DataEC50:  36.3nMAssay Description:Antagonist activity at human adenosine A3 receptor expressed in CHO cells assessed as blockade of NECA-mediated inhibition of forskolin-stimulated cA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A1(Bovine)
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM50257025(4-(cyclohexylamino)-2-phenylpyrido[2,3-e][1,2,4]tr...)
Affinity DataKi:  0.380nMAssay Description:Displacement of [3H]DPCPX from bovine brain cortical membrane adenosine A1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A1(Bovine)
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM50257026(4-(cyclopentylamino)-2-phenylpyrido[2,3-e][1,2,4]t...)
Affinity DataKi:  0.470nMAssay Description:Displacement of [3H]DPCPX from bovine brain cortical membrane adenosine A1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A1(Bovine)
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM21173(DPCPX | CHEMBL183 | 8-cyclopentyl-1,3-dipropyl-2,3...)
Affinity DataKi:  0.5nMAssay Description:Displacement of [3H]DPCPX from bovine brain cortical membrane adenosine A1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A1(Bovine)
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM50256972(4-amino-2-phenylpyrido[2,3-e][1,2,4]triazolo[4,3-a...)
Affinity DataKi:  3.10nMAssay Description:Displacement of [3H]DPCPX from bovine brain cortical membrane adenosine A1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM21173(DPCPX | CHEMBL183 | 8-cyclopentyl-1,3-dipropyl-2,3...)
Affinity DataKi:  3.20nMAssay Description:Displacement of [3H]DPCPX from human cloned adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM50256925(2-(4-methoxyphenyl)pyrido[2,3-e][1,2,4]triazolo[4,...)
Affinity DataKi:  3.30nMAssay Description:Displacement of [125I]AB-MECA from human cloned adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM50257074(N-(2-(4-methoxyphenyl)-1-oxo-1,2-dihydropyrido[2,3...)
Affinity DataKi:  4.54nMAssay Description:Displacement of [125I]AB-MECA from human cloned adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM50149357(2-(4-methoxyphenyl)-6-nitro-[1,2,4]triazolo[4,3-a]...)
Affinity DataKi:  4.70nMAssay Description:Displacement of [125I]AB-MECA from human cloned adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM50149358(4-amino-6-nitro-2-phenyl-[1,2,4]triazolo[4,3-a]qui...)
Affinity DataKi:  4.75nMAssay Description:Displacement of [125I]AB-MECA from human cloned adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A1(Bovine)
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM50189820(N-(6-nitro-1-oxo-2-phenyl-1,2-dihydro-[1,2,4]triaz...)
Affinity DataKi:  6nMAssay Description:Displacement of [3H]DPCPX from bovine brain cortical membrane adenosine A1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A1(Bovine)
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM50257072(N-(1-oxo-2-phenyl-1,2-dihydropyrido[2,3-e][1,2,4]t...)
Affinity DataKi:  7.15nMAssay Description:Displacement of [3H]DPCPX from bovine brain cortical membrane adenosine A1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM50257113(N-benzoyl-N-(2-(4-methoxyphenyl)-1-oxo-1,2-dihydro...)
Affinity DataKi:  7.75nMAssay Description:Displacement of [125I]AB-MECA from human cloned adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM50257026(4-(cyclopentylamino)-2-phenylpyrido[2,3-e][1,2,4]t...)
Affinity DataKi:  8.40nMAssay Description:Displacement of [125I]AB-MECA from human cloned adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM50257072(N-(1-oxo-2-phenyl-1,2-dihydropyrido[2,3-e][1,2,4]t...)
Affinity DataKi:  11.7nMAssay Description:Displacement of [125I]AB-MECA from human cloned adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A1(Bovine)
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM50257027(N-(1-oxo-2-phenyl-1,2-dihydropyrido[2,3-e][1,2,4]t...)
Affinity DataKi:  14nMAssay Description:Displacement of [3H]DPCPX from bovine brain cortical membrane adenosine A1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM50257025(4-(cyclohexylamino)-2-phenylpyrido[2,3-e][1,2,4]tr...)
Affinity DataKi:  15.5nMAssay Description:Displacement of [125I]AB-MECA from human cloned adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM50189813(4-benzamido-6-nitro-2-phenyl-1,2-dihydro-1,2,4-tri...)
Affinity DataKi:  22nMAssay Description:Displacement of [125I]AB-MECA from human cloned adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM50257073(N-(2-(4-methoxyphenyl)-1-oxo-1,2-dihydropyrido[2,3...)
Affinity DataKi:  41nMAssay Description:Displacement of [125I]AB-MECA from human cloned adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM50149370(4-Amino-2-(4-methoxy-phenyl)-6-nitro-2H-[1,2,4]tri...)
Affinity DataKi:  47nMAssay Description:Displacement of [125I]AB-MECA from human cloned adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM50257028(N-(1-oxo-2-phenyl-1,2-dihydropyrido[2,3-e][1,2,4]t...)
Affinity DataKi:  70.3nMAssay Description:Displacement of [125I]AB-MECA from human cloned adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A1(Bovine)
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM50257075(N-benzoyl-N-(1-oxo-2-phenyl-1,2-dihydropyrido[2,3-...)
Affinity DataKi:  70.7nMAssay Description:Displacement of [3H]DPCPX from bovine brain cortical membrane adenosine A1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A1(Bovine)
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM50257024(4-amino-2-(4-hydroxyphenyl)pyrido[2,3-e][1,2,4]tri...)
Affinity DataKi:  112nMAssay Description:Displacement of [3H]DPCPX from bovine brain cortical membrane adenosine A1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM50256925(2-(4-methoxyphenyl)pyrido[2,3-e][1,2,4]triazolo[4,...)
Affinity DataKi:  114nMAssay Description:Displacement of [3H]DPCPX from human cloned adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM50257152(4-(cyclopentylamino)-6-nitro-2-phenyl-[1,2,4]triaz...)
Affinity DataKi:  116nMAssay Description:Displacement of [125I]AB-MECA from human cloned adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM50257027(N-(1-oxo-2-phenyl-1,2-dihydropyrido[2,3-e][1,2,4]t...)
Affinity DataKi:  138nMAssay Description:Displacement of [125I]AB-MECA from human cloned adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A1(Bovine)
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM50256924(2-phenylpyrido[2,3-e][1,2,4]triazolo[4,3-a]pyrazin...)
Affinity DataKi:  145nMAssay Description:Displacement of [3H]DPCPX from bovine brain cortical membrane adenosine A1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A1(Bovine)
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM50257028(N-(1-oxo-2-phenyl-1,2-dihydropyrido[2,3-e][1,2,4]t...)
Affinity DataKi:  152nMAssay Description:Displacement of [3H]DPCPX from bovine brain cortical membrane adenosine A1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM50256973(4-amino-2-(4-methoxyphenyl)pyrido[2,3-e][1,2,4]tri...)
Affinity DataKi:  158nMAssay Description:Displacement of [125I]AB-MECA from human cloned adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A1(Bovine)
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM50256974(4-amino-2-(4-fluorophenyl)pyrido[2,3-e][1,2,4]tria...)
Affinity DataKi:  181nMAssay Description:Displacement of [3H]DPCPX from bovine brain cortical membrane adenosine A1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM50257026(4-(cyclopentylamino)-2-phenylpyrido[2,3-e][1,2,4]t...)
Affinity DataKi:  208nMAssay Description:Displacement of [3H]NECA from human cloned adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM50257072(N-(1-oxo-2-phenyl-1,2-dihydropyrido[2,3-e][1,2,4]t...)
Affinity DataKi:  208nMAssay Description:Displacement of [3H]NECA from human cloned adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM50257025(4-(cyclohexylamino)-2-phenylpyrido[2,3-e][1,2,4]tr...)
Affinity DataKi:  211nMAssay Description:Displacement of [3H]NECA from human cloned adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM50189816(N-(2-(4-methoxyphenyl)-6-nitro-1-oxo-1,2-dihydro-[...)
Affinity DataKi:  217nMAssay Description:Displacement of [125I]AB-MECA from human cloned adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM50256924(2-phenylpyrido[2,3-e][1,2,4]triazolo[4,3-a]pyrazin...)
Affinity DataKi:  251nMAssay Description:Displacement of [125I]AB-MECA from human cloned adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Human)
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM21173(DPCPX | CHEMBL183 | 8-cyclopentyl-1,3-dipropyl-2,3...)
Affinity DataKi:  260nMAssay Description:Displacement of [3H]NECA from human cloned adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM50257114(6-nitro-2-phenyl-[1,2,4]triazolo[4,3-a]quinoxaline...)
Affinity DataKi:  279nMAssay Description:Displacement of [125I]AB-MECA from human cloned adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM50257151(4-(cyclohexylamino)-6-nitro-2-phenyl-[1,2,4]triazo...)
Affinity DataKi:  281nMAssay Description:Displacement of [125I]AB-MECA from human cloned adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A1(Bovine)
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM50256926(2-(4-fluorophenyl)pyrido[2,3-e][1,2,4]triazolo[4,3...)
Affinity DataKi:  306nMAssay Description:Displacement of [3H]DPCPX from bovine brain cortical membrane adenosine A1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM50257075(N-benzoyl-N-(1-oxo-2-phenyl-1,2-dihydropyrido[2,3-...)
Affinity DataKi:  335nMAssay Description:Displacement of [125I]AB-MECA from human cloned adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM50189821(N-benzoyl-N-(2-(4-methoxyphenyl)-6-nitro-1-oxo-1,2...)
Affinity DataKi:  342nMAssay Description:Displacement of [125I]AB-MECA from human cloned adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A1(Bovine)
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM50257074(N-(2-(4-methoxyphenyl)-1-oxo-1,2-dihydropyrido[2,3...)
Affinity DataKi:  355nMAssay Description:Displacement of [3H]DPCPX from bovine brain cortical membrane adenosine A1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A1(Bovine)
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM50256971(2-(4-Hydroxyphenyl)-1,2-dihydropyrido[2,3-e]-1,2,4...)
Affinity DataKi:  449nMAssay Description:Displacement of [3H]DPCPX from bovine brain cortical membrane adenosine A1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM50256974(4-amino-2-(4-fluorophenyl)pyrido[2,3-e][1,2,4]tria...)
Affinity DataKi:  490nMAssay Description:Displacement of [125I]AB-MECA from human cloned adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM50257074(N-(2-(4-methoxyphenyl)-1-oxo-1,2-dihydropyrido[2,3...)
Affinity DataKi:  587nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in Wistar rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM50256926(2-(4-fluorophenyl)pyrido[2,3-e][1,2,4]triazolo[4,3...)
Affinity DataKi:  590nMAssay Description:Displacement of [125I]AB-MECA from human cloned adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM50256972(4-amino-2-phenylpyrido[2,3-e][1,2,4]triazolo[4,3-a...)
Affinity DataKi:  656nMAssay Description:Displacement of [125I]AB-MECA from human cloned adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A1(Bovine)
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM50256973(4-amino-2-(4-methoxyphenyl)pyrido[2,3-e][1,2,4]tri...)
Affinity DataKi:  1.10E+3nMAssay Description:Displacement of [3H]DPCPX from bovine brain cortical membrane adenosine A1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM21173(DPCPX | CHEMBL183 | 8-cyclopentyl-1,3-dipropyl-2,3...)
Affinity DataKi:  1.30E+3nMAssay Description:Displacement of [125I]AB-MECA from human cloned adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Universita Di Firenze

Curated by ChEMBL
LigandPNGBDBM50257024(4-amino-2-(4-hydroxyphenyl)pyrido[2,3-e][1,2,4]tri...)
Affinity DataKi:  1.34E+3nMAssay Description:Displacement of [125I]AB-MECA from human cloned adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
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